Expedient and Rapid Synthesis of 1,2,3-Triazolo[5,1-c]morpholines through Palladium−Copper Catalysis

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• 作者：Chinmay Chowdhury ; Sanjukta Mukherjee ; Bimolendu Das ; Basudeb Achari
• 刊名：Journal of Organic Chemistry
• 出版年：2009
• 出版时间：May 1, 2009
• 年：2009
• 卷：74
• 期：9
• 页码：3612-3615
• 全文大小：162K
• 年卷期：v.74,no.9(May 1, 2009)
• ISSN：1520-6904

文摘

A one-pot approach using palladium−copper as catalyst has been developed for the synthesis of morpholines fused with 1,2,3-triazole. Good regioselectivity, mild reaction conditions, high yields and short reaction time are the hallmarks of this method.