Synthesis of enantiomerically enriched (R)- and (S)-benzofuranyl- and benzo[b]thiophenyl-1,2-ethanediols via enantiopure cyanohydrins as intermediates

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• 作者：Lá ; szló ; Csaba Bencze ; Csaba Paizs ; Monica Ioana Toş ; a ; Elemé ; r Vass ; Florin Dan Irimie
• 刊名：Tetrahedron: Asymmetry
• 出版年：2010
• 出版时间：16 March 2010
• 年：2010
• 卷：21
• 期：4
• 页码：443-450
• 全文大小：473 K

文摘

The chemoenzymatic synthesis of highly enantiopure (R)- and (S)-benzofuranyl- and benzo[b]thiophenyl-cyanohydrins and their chemical transformation into the corresponding heteroaryl-1,2-ethanediols is described.