Ni-catalyzed Suzuki-Miyaura coupling reactions of pyrimidin-2-yl phosphates, tosylates and pivalates with arylboronic acids
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- 作者：Ting Xing ; Zhang Zhang ; Yu-Xia Da ; Zheng-Jun Quan ; Xi-Cun Wang
- 关键词：RVAVWCHBMNDDQH-UHFFFAOYSA-N ; HDKKFMXVDFMUQS-UHFFFAOYSA-N ; CSDAUXAPGDRBSC-UHFFFAOYSA-N ; RKAAEZSKIBVVGC-UHFFFAOYSA-N ; UHKOXYQKXLAKDM-UHFFFAOYSA-N ; OPEJTCDVORPEPV-UHFFFAOYSA-N ; FXIVAVSVPUSHPA-UHFFFAOYSA-N ; IQEQUTOVOYWVKG-UHFFFAOYSA-N ; KHNLNBSXQJCTRT-UHFFFAOYSA-N ; XGQGZAHRDGDIKI-UHFFFAOYSA-N ; NHISUBGSMQKIAC-UHFFFAOYSA-N ; NZMSLESJAWZITD-UHFFFAOYSA-N ; YOZNFRWJCWLTJB-UHFFFAOYSA-N ; WMEKKCWMZWNGIN-UHFFFAOYSA-N ; RXQCUOMAYXDGFD-UHFFFAOYSA-N ; UAWNXFDECYZTBJ-UHFFFAOYSA-N ; SFBSIEMYLNJRGX-UHFFFAOYSA-N ; VPZGJDH
- 刊名：Tetrahedron Letters
- 出版年：2015
- 出版时间：18 November 2015
- 年：2015
- 卷：56
- 期：46
- 页码：6495-6498
- 全文大小：399 K
文摘
Ni-catalyzed Suzuki–Miyaura cross-coupling reactions of pyrimidin-2-yl phosphates, tosylates and pivalates with arylboronic acids were described. A wide array of functionalized pyrimidines have been prepared in impressive yields and show good tolerance towards wide substrate scope.