Ir-Catalyzed Functionalization of 2-Substituted Indoles at the 7-Position: Nitrogen-Directed Aromatic Borylation

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• 作者：Sulagna Paul ; Ghayoor A. Chotana ; Daniel Holmes ; Rebecca C. Reichle ; Robert E. Maleczka ; Jr. ; Milton R. Smith ; III
• 刊名：Journal of the American Chemical Society
• 出版年：2006
• 出版时间：December 13, 2006
• 年：2006
• 卷：128
• 期：49
• 页码：15552 - 15553
• 全文大小：72K
• 年卷期：v.128,no.49(December 13, 2006)
• ISSN：1520-5126

文摘

Ir-catalyzed borylation of 2-substituted indoles selectively yields 7-borylated products in good yields. N-Protection, required for previous functionalizations of 2-substituted indoles, is unnecessary.