A Novel Approach for Analyzing the Dissolution Mechanism of Solid Dispersions
详细信息    查看全文
  • 作者:Yuanhui Ji ; Raphael Paus ; Anke Prudic ; Christian Lübbert
  • 关键词:amorphous solid dispersions ; chemical ; potential ; gradient model ; drug release mechanism ; PC ; SAFT ; poorly water ; soluble pharmaceutical
  • 刊名:Pharmaceutical Research
  • 出版年:2015
  • 出版时间:August 2015
  • 年:2015
  • 卷:32
  • 期:8
  • 页码:2559-2578
  • 全文大小:2,660 KB
  • 参考文献:1.Newman A, Knipp G, Zografi G. Assessing the performance of amorphous solid dispersions. J Pharm Sci. 2012;101(4):1355-7.PubMed View Article
    2.Sun DD, Ju TC, Lee PI. Enhanced kinetic solubility profiles of indomethacin amorphous solid dispersions in poly(2-hydroxyethyl methacrylate) hydrogels. Eur J Pharm Biopharm. 2012;81(1):149-8.PubMed View Article
    3.Hancock BC, Parks M. What is the true solubility advantage for amorphous pharmaceuticals? Pharm Res. 2000;17(4):397-04.PubMed View Article
    4.Vasconcelos T, Sarmento B, Costa P. Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs. Drug Discov Today. 2007;12(23-4):1068-5.PubMed View Article
    5.Sivert A, Bérard V, Andrès C. New binary solid dispersion of indomethacin with surfactant polymer: from physical characterization to in vitro dissolution enhancement. J Pharm Sci. 2010;99(3):1399-13.PubMed View Article
    6.Mura P, Faucci MT, Manderioli A, Bramanti G, Parrini P. Thermal behavior and dissolution properties of naproxen from binary and ternary solid dispersions. Drug Dev Ind Pharm. 1999;25(3):257-4.PubMed View Article
    7.Kogermann K, Penkina A, Predbannikova K, Jeeger K, Veski P, Rantanen J, et al. Dissolution testing of amorphous solid dispersions. Int J Pharm. 2013;444(1-):40-.PubMed View Article
    8.Alonzo DE, Gao Y, Zhou D, Mo H, Zhang GG, Taylor LS. Dissolution and precipitation behavior of amorphous solid dispersions. J Pharm Sci. 2011;100(8):3316-1.PubMed View Article
    9.Arthur AN, Willis RW. The rate of solution of solid substances in their own solutions. J Am Chem Soc. 1897;19(12):930-.View Article
    10.Lu AT, Frisella ME, Johnson KC. Dissolution modeling: factors affecting the dissolution rates of polydisperse powders. Pharm Res. 1993;10(9):1308-4.PubMed View Article
    11.Vudathala GK, Rogers JA. Dissolution of fludrocortisone from phospholipid coprecipitates. J Pharm Sci. 1992;81(3):282-.PubMed View Article
    12.Higuchi T. Rate of release of medicaments from ointment bases containing drugs in suspension. J Pharm Sci. 1961;50(10):874-.PubMed View Article
    13.Higuchi T. Mechanism of sustained-action medication. Theoretical analysis of rate of release of solid drugs dispersed in solid matrices. J Pharm Sci. 1963;52(12):1145-.PubMed View Article
    14.Hixson AW, Crowell JH. Dependence of reaction velocity upon surface and agitation. Ind Eng Chem. 1931;23(8):923-1.View Article
    15.de Almeida LP, Sim?es S, Brito P, Portugal A, Figueiredo M. Modeling dissolution of sparingly soluble multisized powders. J Pharm Sci. 1997;86(6):726-2.PubMed View Article
    16.Korsmeyer RW, Gurny R, Doelker E, Buri P, Peppas NA. Mechanisms of solute release from porous hydrophilic polymers. Int J Pharm. 1983;15(1):25-5.View Article
    17.Baker RW, Lonsdale HK. Controlled release: mechanisms and rates. In: Tanquary AC, Lacey RE, editors. Controlled release of biologically active agents. Advances in experimental medicine and biology. New York: Plenum; 1974. p. 15-2.View Article
    18.Craig DQM. The mechanisms of drug release from solid dispersions in water-soluble polymers. Int J Pharm. 2002;231(2):131-4.PubMed View Article
    19.Siepmann J, Kranz H, Bodmeier R, Peppas NA. HPMC-matrices for controlled drug delivery: a new model combining diffusion, swelling, and dissolution mechanisms and predicting the release kinetics. Pharm Res. 1999;16(11):1748-6.PubMed View Article
    20.Langham ZA, Booth J, Hughes LP, Reynolds GK, Wren SA. Mechanistic insights into the dissolution of spray-dried amorphous solid dispersions. J Pharm Sci. 2012;101(8):2798-10.PubMed View Article
    21.Costa P, Sousa Lobo JM. Modeling and comparison of dissolution profiles. Eur J Pharm Sci. 2001;13(2):123-3.PubMed View Article
    22.Alonzo DE, Zhang GG, Zhou D, Gao Y, Taylor LS. Understanding the behavior of amorphous pharmaceutical systems during dissolution. Pharm Res. 2010;27(4):608-8.PubMed View Article
    23.Lu XH, Ji YH, Liu HL. Non–equilibrium thermodynamics analysis and its application in interfacial mass transfer. Sci China Chem. 2011;54(10):1659-6.View Article
    24.Liu C, Ji Y, Shao Q, Feng X, Lu X. Thermodynamic analysis for synthesis of advanced materials. In: Lu XH, Hu Y, editors. Molecular thermodynamics of complex systems, Struct Bond. Berlin: Springer–Verlag; 2009. p. 193-70.View Article
    25.Ji YH, Ji XY, Liu C, Feng X, Lu XH. Modelling of mass transfer coupling with crystallization kinetics in microscale. Chem Eng Sci. 2010;65:2649-5.View Article
    26.Ruether F, Sadowski G. Modeling the solubility of pharmaceuticals in pure solvents and solvent mixtures for drug process design. J Pharm Sci. 2009;98(11):4205-5.
    27.Cassens J, Prudic A, Ruether F, Sadowski G. Solubility of pharmaceuticals and their salts as a function of pH. Ind Eng Chem Res. 2013;52(7):2721-1.
    28.Fuchs D, Fischer J, Tumakaka F, Sadowski G. Solubility of amino acids: influence of the pH value and the a
  • 作者单位:Yuanhui Ji (1)
    Raphael Paus (1)
    Anke Prudic (1)
    Christian Lübbert (1)
    Gabriele Sadowski (1)

    1. TU Dortmund, Department of Biochemical and Chemical Engineering, Laboratory of Thermodynamics, Emil-Figge-Str. 70, 44227, Dortmund, Germany
  • 刊物类别:Biomedical and Life Sciences
  • 刊物主题:Biomedicine
    Pharmacology and Toxicology
    Pharmacy
    Biochemistry
    Medical Law
    Biomedical Engineering
  • 出版者:Springer Netherlands
  • ISSN:1573-904X
文摘

© 2004-2018 中国地质图书馆版权所有 京ICP备05064691号 京公网安备11010802017129号

地址:北京市海淀区学院路29号 邮编:100083

电话:办公室:(+86 10)66554848;文献借阅、咨询服务、科技查新:66554700