Synthesis of novel N-aryl-4-[6-(2-fluoropyridin-3-yl)quinazolin-2-yl]-piperazine-1-carboxamide or -carbothioamide derivatives and their antimicrobial activity

详细信息    查看全文

• 作者：D. Suresh Babu (1)
  Doddaga Srinivasulu (1)
  Venkata S. Kotakadi (1)
  
  1. Sri Venkateswara University ; Tirupati ; 517502 ; Andhra Pradesh ; India
  
• 关键词：arylisocyanates ; arylisothiocyanates ; piperazine ; quinazoline ; Suzuki coupling ; antimicrobial activity
• 刊名：Chemistry of Heterocyclic Compounds
• 出版年：2015
• 出版时间：January 2015
• 年：2015
• 卷：51
• 期：1
• 页码：60-66
• 全文大小：488 KB
• 参考文献：1. L眉th, A, L枚we, W (2008) Eur. J. Med. Chem. 43: pp. 1478 CrossRef
  2. 艩pirkov谩, K, Stankovsk媒, S, Mrvov谩, A, 膶ip谩k, 墓 (1999) Chem. Pap. 53: pp. 272
  3. Tiwari, R, Chhabra, GA (2010) J. Chem. 22: pp. 5981
  4. Kumar, A, Sharma, P, Kumari, P, Kalal, BL (2011) Bioorg. Med. Chem. Lett. 21: pp. 4353 CrossRef
  5. Bartroli, J, Turmo, E, Alguer贸, M, Boncompte, E, Vericat, ML, Conte, L, Ramis, J, Merlos, M, Garc铆a-Rafanell, J, Forn, J (1998) J. Med. Chem. 41: pp. 1869 CrossRef
  6. Balakumar, C, Lamba, P, Kishore, DP, Narayana, BL, Rao, KV, Rajwinder, K, Rao, AR, Shireesha, B, Narsaiah, B (2010) Eur. J. Med. Chem. 45: pp. 4904 CrossRef
  7. Wakeling, AE, Guy, SP, Woodburn, JR, Ashton, SE, Curry, BJ, Barker, AJ, Gibson, KH (2002) Cancer Res. 62: pp. 5749
  8. Nandy, P, Vishalakshi, MT, Bhat, AR (2006) Indian J. Heterocycl. Chem. 15: pp. 293
  9. Kabri, Y, Azas, N, Dum猫tre, A, Hutter, S, Laget, M, Verhaeghe, P, Gellis, A, Vanelle, P (2010) Eur. J. Med. Chem. 45: pp. 616 CrossRef
  10. Aly, AA (2003) Chin. J. Chem. 21: pp. 339 CrossRef
  11. Saravanan, G, Alagarsamy, V, Prakash, CR (2010) Int. J. Pharm. Pharm. Sci. 2: pp. 83
  12. Kim, BM, Evans, BE, Gilbert, KF, Hanifin, CM, Vacca, JP, Michelson, SR, Darke, PL, Zugay, JA, Emini, EA, Schleif, W, Lin, JH, Anderson, PS, Huff, JR (1995) Bioorg. Med. Chem. Lett. 5: pp. 2707 CrossRef
  13. Askin, D, Eng, KK, Rossen, K, Purick, RM, Wells, KM, Volante, RP, Reider, PJ (1994) Tetrahedron Lett. 35: pp. 673 CrossRef
  14. Patrick, GL, Kinsmar, OS (1996) Eur. J. Med. Chem. 31: pp. 615 CrossRef
  15. Hishmat, OH, Abdel Galil, FM, Farrag, DS (1990) Pharmazie 45: pp. 793
  16. Patel, HS, Desai, HD, Mistry, HJ (2004) J. Chem. 1: pp. 93
  17. Gan, LL, Lu, YH, Zhou, CH (2009) Chin. J. Biochem. Pharm. 30: pp. 127
  18. Todorovic, A, Haskell-Luevano, C (2005) Peptides 26: pp. 2026 CrossRef
  19. Kundu, B (2003) Curr. Opin. Drug Discovery Dev. 6: pp. 815
  20. Myangar, KN, Akhaja, TN, Naik, DR, Raval, JP (2012) Chem. Sci. Trans. 1: pp. 688 CrossRef
  21. Fournier, J, Bruneau, C, Dixneuf, PH, L茅colier, S (1991) J. Org. Chem. 56: pp. 4456 CrossRef
  22. Abdel-Rahman, HM, Morsy, MA (2007) J. Enzyme Inhib. Med. Chem. 22: pp. 57 CrossRef
  23. Dom铆ngu茅z, JN, Le贸n, C, Rodrigues, J, Gamboa de Dom铆nguez, N, Gut, J, Rosenthal, PJ (2005) J. Med. Chem. 48: pp. 3654 CrossRef
  24. Suzuki, A (1991) Pure Appl. Chem. 63: pp. 419
  25. Suzuki, A (1999) J. Organomet. Chem. 576: pp. 147 CrossRef
  26. Miyaura, N, Suzuki, A (1995) Chem. Rev. 95: pp. 2457 CrossRef
  27. Kazmi, SU, Ali, SN, Jamal, SA, Atta-ur-Rahman, (1991) Pak. J. Pharm. Sci. 4: pp. 113
  28. Atta-ur-Rehman, , Choudhary, MI, Thomsen, WJ (2001) Bioassay Techniques for Drug Development. Harwood Academic Publishers, Amsterdam CrossRef
  29. Greenwood, D, Slack, R, Peutherer, J (1997) Medical Microbiology: A Guide to Microbial Infections: Pathogenesis, Immunity, Laboratory Diagnosis and Control, Edinburgh. ELST Publishers, Edinburgh
  30. Perez, C, Pauli, M, Bazevque, P (1990) Acta Biol. Med. Exp. 15: pp. 113
  31. Rasheed, S, Venkataramana, K, Chandrasekhar, K, Fareeda, G, Naga Raju, C (2012) Arch. Pharm. 345: pp. 294 CrossRef
  32. Vasbinder, MM, Aquila, B, Augustin, M, Chen, H, Cheung, T, Cook, D, Drew, L, Fauber, BP, Glossop, S, Grondine, M, Hennessy, E, Johannes, J, Lee, S, Lyne, P, M枚rtl, M, Omer, C, Palakurthi, S, Pontz, T, Read, J, Sha, L, Shen, M, Steinbacher, S, Wang, H, Allan, W, Minwei, Y (2013) J. Med. Chem. 56: pp. 1996 CrossRef
  33. DiMauro, EF, Newcomb, J, Nunes, JJ, Bemis, JE, Boucher, C, Buchanan, JL, Buckner, WH, Cee, VJ, Chai, L, Deak, HL, Epstein, LF, Faust, T, Gallant, P, Geuns-Meyer, SD, Gore, A, Yan, G, Henkle, B, Hodous, BL, Hsieh, F, Huang, X, Kim, JL, Lee, JH, Martin, MW, Masse, CE, McGowan, DC, Metz, D, Mohn, D, Morgenstern, KA, Oliveira-dos-Santos, A, Patel, VF, Powers, D, Rose, PE, Schneider, S, Tomlinson, SA, Tudor, Y-Y, Turci, SM, Welcher, AA, White, RD, Zhao, H, Zhu, L, Zhu, X (2006) J. Med. Chem. 49: pp. 5671 CrossRef
  
• 刊物类别：Chemistry and Materials Science
• 刊物主题：Chemistry
  Organic Chemistry
  Pharmacy
  Russian Library of Science
  
• 出版者：Springer New York
• ISSN：1573-8353

文摘