Biological affinity evaluation of Lawsonia inermis origin Lawsone compound and its radioiodinated form via in vitro methods

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• 作者：Volkan Tekin ; F. Zumrut Biber Muftuler…
• 关键词：Lawsonia inermis ; Lawsone ; 131I ; Cell culture ; Wound healing ; Antibacterial and antifungal activity
• 刊名：Journal of Radioanalytical and Nuclear Chemistry
• 出版年：2015
• 出版时间：January 2015
• 年：2015
• 卷：303
• 期：1
• 页码：701-708
• 全文大小：898 KB
• 参考文献：1. Makhija IK, Dhananjaya, Kumar SV, Devkar R, Khamar D, Manglani N, Chandrakar S (2011) / Lawsonia inermis–from traditional use to scientific assessment. African J Pharm Sci Pharm 1(2):145-65
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• 作者单位：Volkan Tekin (1)
  F. Zumrut Biber Muftuler (1)
  Ozge Kozgus Guldu (1)
  Ayfer Yurt Kilcar (1)
  E. Ilker Medine (1)
  Murat Yavuz (2) (3)
  Perihan Unak (1)
  Suna Timur (3)
  
  1. Department of Nuclear Applications, Institute of Nuclear Science, Ege University, 35100, Bornova, Izmir, Turkey
  2. Department of Chemistry, Faculty of Science, Dicle University, 21280, Diyarbakir, Turkey
  3. Department of Biochemistry, Faculty of Sciences, Ege University, 35100, Bornova, Izmir, Turkey
  
• 刊物类别：Chemistry and Materials Science
• 刊物主题：Chemistry
  Nuclear Chemistry
  Physical Chemistry
  Nuclear Physics, Heavy Ions and Hadrons
  Diagnostic Radiology
  Inorganic Chemistry
  
• 出版者：Akad茅miai Kiad贸, co-published with Springer Science+Business Media B.V., Formerly Kluwer Academic
• ISSN：1588-2780

文摘

WST-1-based cytotoxicity assay of lawsone (LW) was performed on MCF7, Caco2, BJ and Keratinocyte cells and viabilities were found as over 90?% for all cells. Significant wound healing effect of LW was reported on Keratinocyte cells. Antibacterial and antifungal activities of LW were tested on seven microorganisms with three concentrations and 1,000?μg/disc of LW showed antibacterial effect on Bacillus subtilis. In vitro cell incorporation of radioiodinated LW (131I-LW) was evaluated on same cells. Keratinocyte cells uptake were 5 times more. Consequently, 131I-LW was found usable for researches about especially skin diseases in addition to breast and intestinal cancer.