Multicomponent synthesis and antimicrobial activity of alkyl 4-arylamino-1,2,6-triaryl-1,2,5,6-tetrahydropyridine-3-carboxylates

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• 作者：A. N. Yankin ; N. V. Nosova ; V. L. Gein…
• 关键词：multicomponent synthesis ; tetrahydropyridines ; antimicrobial activity
• 刊名：Russian Journal of General Chemistry
• 出版年：2015
• 出版时间：April 2015
• 年：2015
• 卷：85
• 期：4
• 页码：844-850
• 全文大小：228 KB
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• 作者单位：A. N. Yankin (1)
  N. V. Nosova (1)
  V. L. Gein (1)
  M. V. Tomilov (1)
  
  1. Perm State Pharmaceutical Academy, ul. Polevaya 2, Perm, 614990, Russia
  
• 刊物类别：Chemistry and Materials Science
• 刊物主题：Chemistry
  Chemistry
  Russian Library of Science
  
• 出版者：MAIK Nauka/Interperiodica distributed exclusively by Springer Science+Business Media LLC.
• ISSN：1608-3350

文摘

Reaction of arylamines with aromatic aldehydes and β-ketoesters in the presence of bismuth nitrate or crystalline iodine as a catalyst afforded to alkyl 4-arylamino-1,2,6-triaryl-1,2,5,6-tetrahydropyridine-3-carboxy-lates. Antimicrobial activity of the obtained compounds was studied.