Morita-Baylis-Hillman reactions of isatins with allenoates

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• 作者：Qian-Yi Zhao^a ; Zhong Lian^b ; Yin Wei^b ; Min Shi^a ; ^b ; ^{mshi@mail.sioc.ac.cn}
• 关键词：4-(N ; N-Dimethylamino)pyridine (DMAP) ; Morita&ndash ; Baylis&ndash ; Hillman reaction ; Isatins ; 伪-Substituted allenoates
• 刊名：Tetrahedron
• 出版年：2012
• 期刊代码：107_00404020
• 类别：ch
• 出版时间：17 June, 2012
• 卷：68
• 期：24
• 页码：4899-4905
• 文件大小：528 K

摘要

4-(N,N-dimethylamino)pyridine (DMAP) was found to be a fairly efficient catalyst for the Morita-Baylis-Hillman reactions of isatins with 伪-substituted allenoates to give the corresponding products in good to high yields with moderate diastereoselectivities under mild conditions.