Broflanilide及其类似物研究进展
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摘要
Broflanilide是一种全新作用机制的双酰胺类杀虫剂,主要用于防治鳞翅目、鞘翅目、白蚁及蚊蝇等害虫。简要介绍了broflanilide及其市场开发状况和合成路线,根据其主要研发公司(MCAG、Syngenta、Agro-Kanesho、Bayer等)对该类化合物的研究进展进行了概述,并对其发展趋势和前景作了展望。
Broflanilide is a diamide insecticides with novel mechanism of action. It is mainly used for the control of Lepidopteran and Coleopteran pests as well as termites, mosquitoes, houseflies and so on. The business development state and synthetic methods of broflanilide from major research and development companies was introduced briefly in this article. The research progress of the analogues of broflanilide was reviewed and the development and prospects of this kind of insecticides were also predicted.
Broflanilide is a diamide insecticides with novel mechanism of action. It is mainly used for the control of Lepidopteran and Coleopteran pests as well as termites, mosquitoes, houseflies and so on. The business development state and synthetic methods of broflanilide from major research and development companies was introduced briefly in this article. The research progress of the analogues of broflanilide was reviewed and the development and prospects of this kind of insecticides were also predicted.
引文
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[47]冯启,袁静,张红敏.苯甲酰胺类衍生物、其制备方法及应用:CN,102993054[P].2013-03-27.
[2]NAKAO T,BANBA S.Broflanilide:A Meta-diamide Insecticide with a Novel Mode of Action[J].Bioorganic&Medicinal Chemistry,2016,24(3):372-377.
[3]JEANMART S,EDMUNDS A J,LAMBERTH C,et al.Synthetic Approaches to the 2010-2014 New Agrochemicals[J].Bioorganic&Medicinal Chemistry,2016,24(3):317-341.
[4]YOSHIDA K,WAKITA T,KATSUTA H,et al.Insecticide for Agricultural or Horticultural Use and Method of Use Thereof:WO,2005021488[P].2005-03-10.
[5]YOSHIDA K,WAKITA T,KATSUTA H,et al.Amide Derivatives,Process for Production of the Same and Method for Application Thereof as Insecticide:WO,2005073165[P].2005-08-11.
[6]TAKAHASHI K,KAI A,WAKITA T.Method for Producing Insecticide and Production Intermediate of the Same:JP,2006225340[P].2006-08-31.
[7]KAI A,WAKITA T,YOSHIDA K,et al.Agricultural/Horticultural Insecticide:JP,2006306771[P].2006-11-09.
[8]KAI A,WAKITA T,KATSUTA,et al.Amide Derivative and Pesticide Containing Such Compound:WO,2006137376[P].2006-12-28.
[9]YOSHIDA K,KOBAYASHI Y,NOMURA M,et al.Amide Derivative,Pesticide Containing Such Compound and Use Thereof:WO,2006137395[P].2006-12-28.
[10]KAWAHARA N,NOMURA M,DAIDO H.Pest Control Composition:WO,2007013150[P].2007-02-01.
[11]WAKITA T,DAIDO H,KAI A,et al.Amide Derivative and Application Method Thereof as Insecticide:JP,2007099761[P].2007-04-19.
[12]KOBAYASHI Y,KATSUTA H,NOMURA M,et al.Amide Derivative,Pest Control Agent Containing the Amide Derivative and Pest Controlling Method:WO,2010013567[P].2010-02-04.
[13]KOBAYASHI Y,DAIDO H,KATSUTA H,et al.Amide Derivative,Pest Control Agent Containing the Amide Derivative and Use of the Pest Control Agent:WO,2010018714[P].2010-02-18.
[14]FUKAZAWA Y.Amide Derivative and Insecticide:JP,2010138079[P].2010-06-24.
[15]HIRABAYASHI A,BANBA S,WAKITA T,et al.Amide Derivative and Harmful Organism-controlling Agent Containing the Amide Derivative:JP,2011063549[P].2011-03-31.
[16]FUKAZAWA Y,OKURA H,KOHNO T,et al.Imide Compound,Method for Manufacturing Same,and Use as Insecticide:WO,2014054158[P].2014-04-10.
[17]FUKAZAWA Y,OKURA H,KONO T,et al.Imide Compound,Process of Producing the Same,and Application Thereof as Insecticide:JP,5778091[P].2015-09-16.
[18]JUNG P,DURIEUX P,LUTZ W,et al.Insecticidal Compounds:WO,2007128410[P].2007-11-15.
[19]JUNG P,GODFREY C,LUTZ W,et al.Insecticidal Compounds:WO,2008074427[P].2008-06-26.
[20]JUNG P,GODFREY C,RICHARD A,et al.Insecticidal Compounds:WO,2008107091[P].2009-07-30.
[21]JUNG P,HUETER O,RANZRENOLD P.Insecticidal Compounds:WO,2012069366[P].2012-05-31.
[22]RENOLD P,MAIENFISCH P,JUNG P,et al.Insecticidal Compounds:WO,2008012027[P].2008-01-31.
[23]JUNG P,RENOLD P,GODFREY C,et al.Insecticidal Compounds:WO,2009049844[P].2009-04-23.
[24]STOLLER A,JUNG P,GODFREY C,et al.Insecticidal Compounds:WO,2009049845[P].2009-04-23.
[25]JUNG P,GODFREY C,HUETER O,et al.Insecticidal Compounds:WO,2011095462[P].2011-08-11.
[26]JUNG P,GODFREY C,HUETER O,et al.4-Cyano-3-benzoylamino-N-phenyl-benzamides for Use in Pest Control:WO,2010127926[P].2010-11-11.
[27]EDMUNDS A,STOLLER A,PITTERNA T.Insecticidal Compounds:WO,2015097091[P].2015-07-02.
[28]HUETER O,RENOLD P,MAIENFISCH P,et al.Insecticidal2-Methoxybenzamide Derivatives:WO,2013050261[P].2013-04-11.
[29]HUETER O,JUNG P,JOSEPH M,et al.Insecticidal Compounds:WO,2014067838[P].2014-05-08.
[30]THOMAS P,AYLES G,FRANZ H,et al.Insecticidal Compounds:GB,2520098[P].2015-05-13.
[31]STOLLER A,EDMUNDS A,PITTERNA T,et al.Insecticidal Compounds:WO,2014161848[P].2014-10-09.
[32]HUETER O,PITTERNA T,STOLLER A,et al.Insecticidal Compounds:WO,2014161849[P].2014-10-09.
[33]PITTERNA T,STOLLER A,EDMUNDS A.Insecticidal Compounds:WO,2015097094[P].2015-07-02.
[34]USUI S,FUKUCHI T,KINOSHITA Y.3-Aminoxalylaminobenzamide Derivatives,and Insecticidal and Miticidal Agents Containing Same as Active Ingredient:WO,2010090282[P].2010-08-12.
[35]USUI S,FUKUCHI T,KINOSHITA S.3-Aminooxalyl Aminobenzamide Derivative,and Insecticide and Miticide Using Same as Active Ingredient:WO,2012020483[P].2012-02-16.
[36]USUI S,KAKINUMA S,FUKUCHI T,et al.3-Aminooxalylaminobenzamide Derivative,and Insecticidal and Acaricidal Agent Containing Same as Active Ingredient:WO,2012077221[P].2012-06-14.
[37]USUI S,FUKUCHI T,KINOSHITA S.3-Aminooxalylaminobenzamide Derivative,and Insecticidal or Miticidal Agent Comprising Same as Active Ingredient:WO,2012164698[P].2012-12-06.
[38]YOSHIDA K,KOBAYASHI Y,NOMURA M,et al.Amide Derivative,Pesticide Containing such Compound and Use Thereof:WO,2006137395[P].2006-12-28.
[39]GOERGENS U,YANAGI A,WADA K,et al.Aminobenzamide Derivatives as Useful Agents for Controlling Animal Parasites:WO,2009080203[P].2009-07-02.
[40]MAUE M,ADELT I,GIENCKE W,et al.Halogen-substituted Compounds Used as Pesticides:WO,2010051926[P].2011-05-26.
[41]MAUE M,ADELT I,GIENCKE W,et al.Halogen-substituted Compounds as Pesticides:WO,2010133312[P].2010-11-25.
[42]MIHARA J,MURATA T,DOMON K,et al.Novel Acylaminobenzamide Derivatives:WO,2010015355[P].2010-02-11.
[43]TAKAHASHI M.3-Aminooxalylaminobenzamide Compound and Use for Controlling Harmful Arthropod:WO,2016143652[P].2016-09-15.
[44]TAKAHASHI M.3-Aminooxalylaminobenzamide Compound and Use for Controlling Harmful Arthropod:WO,2016143650[P].2016-09-15.
[45]TAKAHASHI M.Oxalyl Amide Compound and Use Thereof for Controlling Harmful Arthropods:WO,2017026298[P].2017-02-16.
[46]HEEMSTRA R.,ROSS R,DEKORVER,K,et al.Molecules Having Pesticidal Utility,and Intermediates,Compositions,and Processes,Related Thereto:WO,2016168059[P].2016-10-20.
[47]冯启,袁静,张红敏.苯甲酰胺类衍生物、其制备方法及应用:CN,102993054[P].2013-03-27.