搜索页_μ-opioid receptor agonist

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在“Elsevier电子期刊”中，命中：26条，耗时：0.0429789 秒

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1.Discovery, structure-activity relationship studies, and anti-nociceptive effects of N-(1,2,3,4-tetrahydro-1-isoquinolinylmethyl)benzamides as novel opioid receptor agonists

作者：Sheng-Ren Chen^a ; ^c ; Yi-Yu Ke^a ; ¹ ; Teng-Kuang Yeh^a ; ¹ ; Shu-Yu Lin^a ; Li-Chin Ou^a ; Shu-Chun Chen^a ; Wan-Ting Chang^a ; Hsiao-Fu Chang^a ; Zih-Huei Wu^a ; Chih-Chien Hsieh^a ; Ping-Yee Law^b ; Horace H. Loh^b ; Chuan Shih^a ; Yiu-Kay Lai^c ; ^{yklai@life.nthu.edu.tw} ; Shiu-Hwa Yeh^a ; ^d ; ^{bau9763@bp.nhri.org.tw} ; Shau-Hua Ueng^a ; ^{shueng@nhri.org.tw}

关键词：μ-opioid receptor agonist ; κ-opioid receptor agonist ; Structure-activity relationship ; Blood-brain barrier ; Penetration ; Anti-nociceptive effects ; Tail-flick test

刊名：European Journal of Medicinal Chemistry

出版年：2017

2.Suppression of the acute upregulation of phosphorylated-extracellular regulated kinase in ventral tegmental area by a μ-opioid receptor agonist is related to resistance to rewarding effects in a mouse model of bone cancer

作者：Atsushi Nakamura ; ^{atsushi_nakamura@shionogi.co.jp} ; Hiroko Ono ; Azusa Ando ; Mikie Hinata ; Kazuki Niidome ; Shigeki Omachi ; Gaku Sakaguchi ; Shunji Shinohara

关键词：Antinociception ; Bone cancer pain ; Extracellular regulated kinase ; Opioid ; Rewarding effect

刊名：Journal of Pharmacological Sciences

出版年：2017

3.Distinguishing subgroups among μ-opioid receptor agonists using Na⁺,K⁺-ATPase as an effector mechanism

作者：Willias Masocha^a ; ¹ ; Luis G. Gonzá ; lez^b ; ¹ ; ^{lggonzal@ugr.es" class="auth_mail" title="E-mail the corresponding author} ; Ahmad Agil^b

关键词：Antinociception ; μ-opioid receptor agonists ; Ouabain ; Na+ ; K+-ATPase ; Synaptosomes

刊名：European Journal of Pharmacology

出版年：2016

4.NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids

作者：Nadja A. Simeth^a ; ^d ; Manuel Bause^a ; ^d ; Michael Dobmeier^a ; ^d ; Ralf C. Kling^b ; ^c ; Daniel Lachmann^a ; Harald Hü ; bner^b ; Jü ; rgen Einsiedel^b ; Peter Gmeiner^b ; ^{peter.gmeiner@fau.de} ; Burkhard Kö ; nig^a ; ^{burkhard.koenig@ur.de}

关键词：Neurotensin ; Peptides ; Non-natural amino acid

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

5.Nalfurafine hydrochloride, a selective κ opioid receptor agonist, has no reinforcing effect on intravenous self-administration in rhesus monkeys

作者：Kaoru Nakao^a ; ^{Kaoru_Nakao@nts.toray.co.jp" class="auth_mail" title="E-mail the corresponding author} ; Mikito Hirakata^a ; Yohei Miyamoto^a ; Mie Kainoh^a ; Yoshio Wakasa^b ; Tomoji Yanagita^c

关键词：Nalfurafine hydrochloride ; TRK-820 ; κ opioid receptor ; Self-administration ; Monkey

刊名：Journal of Pharmacological Sciences

出版年：2016

6.The antinociceptive effects of a δ-opioid receptor agonist in mice with painful diabetic neuropathy: Involvement of heme oxygenase 1

作者：Sí ; lvia Castany¹ ; Mireia Carcolé ; ¹ ; Sergi Leá ; nez ; Olga Pol ; ^{opol@santpau.es" class="auth_mail" title="E-mail the corresponding author}

关键词：CoPP ; cobalt protoporphyrin IX ; CORM-2 ; tricarbonyldichlororuthenium(II) dimer ; DOR ; δ-opioid receptor ; DPDPE ; [d-Pen(2) ; d-Pen(5)]-Enkephalin ; HO-1 ; inducible heme oxygenase ; MOR ; μ-opioid receptor ; SnPP ; tin protoporphyrin IX ; STZ ; streptozotocin

刊名：Neuroscience Letters

出版年：2016

7.Opioid mechanisms and opioid drugs

作者：John McDonald ; David G. Lambert

关键词：G-protein-coupled receptor ; MOP/DOP opioid receptor actions ; NOP-receptor antagonist

刊名：Anaesthesia & Intensive Care Medicine

出版年：2016

8.Design synthesis and structure-activity relationship of 5-substituted (tetrahydronaphthalen-2yl)methyl with N-phenyl-N-(piperidin-2-yl)propionamide derivatives as opioid ligands

作者：Srinivas Deekonda^a ; David Rankin^b ; Peg Davis^b ; Josephine Lai^b ; Todd. W. Vanderah^b ; Frank Porecca^b ; Victor J. Hruby^a ; ^{hruby@email.arizona.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：GPCR ; G protein-coupled receptor ; MOR ; Mu opioid receptor ; DOR ; delta opioid receptor ; Boc ; tert-butyloxycarbonyl ; NaOtBu ; sodium tert-butoxide ; Et3N ; triethylamine ; HCl ; hydrochloric acid ; BH3-SMe2 ; borane dimethylsulfide ; DHP ; dihydropyran ; PPTS ; pyridinium p-toluenesulfonate ; Ph3P ; triphenylphosphine ; Na(OAc)3BH ; sodium triacetoxyborohydride ; DCE ; dichloroethane ; DIPEA ; N ; N-diisopropylethylamine ; ACN ; acetonitrile ; DCM ; dichloromethane ; rt ; room temperature ; CHO ; Chinese hamster ovary ; dALEA

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

9.Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives

作者：Silvia Franchini^a ; Umberto Maria Battisti^a ; Adolfo Prandi^a ; Annalisa Tait^a ; Chiara Borsari^a ; Elena Cichero^b ; Paola Fossa^b ; Antonio Cilia^c ; Orazio Prezzavento^d ; Simone Ronsisvalle^d ; Giuseppina Aricò ; ^e ; Carmela Parenti^e ; Livio Brasili^a ; ^{livio.brasili@unimore.it" class="auth_mail" title="E-mail the corresponding author}

关键词：Sigma receptors ligands ; Sigma-1 ; Sigma-2 ; Piperidine ; Piperazine ; 1 ; 3-Dioxolane ; Receptor-mediated analgesia

刊名：European Journal of Medicinal Chemistry

出版年：2016

10.Peripheral interactions between cannabinoid and opioid receptor agonists in a model of inflammatory mechanical hyperalgesia

作者：Q-Schick Auh^b ; Yang Hyun Chun^b ; Ohannes K. Melemedjian^a ; Youping Zhang^a ; Jin Y. Ro^a ; ^b ; ^{jro@umaryland.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：DAMGO ; ACPA ; μ Opioid receptor ; CB1 ; Dorsal root ganglia ; Isobologram ; Complete freund&rsquo ; s adjuvant

刊名：Brain Research Bulletin

出版年：2016

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