搜索页_ 2-(1H-benzotriazol-1-yl)-1

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Elsevier电子期刊(42)

在“Elsevier电子期刊”中，命中：42条，耗时：小于0.01 秒

在所有数据库中总计命中：59条

1.Bivalent SIRT1 inhibitors

作者：Juan Wang¹ ; Wenwen Zang¹ ; Jiajia Liu¹ ; Weiping Zheng ; ^{wzheng@ujs.edu.cn}

关键词：β-NAD+ ; β-nicotinamide adenine dinucleotide ; NAM ; nicotinamide ; 2&prime ; -O-AADPR ; 2&prime ; -O-acyl-ADP-ribose ; RP-HPLC ; reversed-phase high performance liquid chromatography ; HRMS ; high-resolution mass spectrometry ; EDC-MeI ; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimide methiodide ; DIC ; N ; N&prime ; -diisopropylcarbodiimide ; HBTU ; 2-(1H-benzotriazole-1-yl)-113 ; 3-tetramethylaminium hexafluorophosphate ; HOBt ; N-hydroxybenzotriazole ; NMM ; N-methylmorpholine ; EDC-HCl ; 1-(3-dimethylaminopropyl)-3-ethyl

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

2.1-Heteroarylpropan-2-ones as inhibitors of fatty acid amide hydrolase: Studies on structure-activity relationships and metabolic stability

作者：Stefan Zahov ; David Garzinsky ; Walburga Hanekamp ; Matthias Lehr ; ^{lehrm@uni-muenster.de}

关键词：Propan-2-one ; Fatty acid amide hydrolase ; Enzyme inhibition ; Metabolic stability ; Aqueous solubility

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

3.Synthesis and preliminary evaluation of 5,7-dimethyl-2-aryl-3H-pyrrolizin-3-ones as angiogenesis inhibitors

作者：Nicholas S. Kirk^a ; Anna Bezos^b ; Anthony C. Willis^c ; Pichit Sudta^d ; ^e ; Sunit Suksamrarn^e ; Christopher R. Parish^b ; Marie Ranson^f ; Michael J. Kelso^a ; ^{mkelso@uow.edu.au" class="auth_mail" title="E-mail the corresponding author}

关键词：HBTU ; 2-(1H-benzotriazol-1-yl)-113 ; 3-tetramethyluronium hexafluorophosphate ; CSF-1R ; colony-stimulating factor-1 receptor ; DIPEA ; N ; N-diisopropylethylamine ; FLT-3 ; Fms-like tyrosine kinase 3 ; FOV ; field of view ; HUVEC ; human umbilical vein endothelial cell ; PDGFR ; platelet-derived growth factor receptor ; RTK ; receptor tyrosine kinase ; THF ; tetrahydrofuran ; VEGFR ; vascular endothelial growth factor receptor

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

4.Cyclic non-opioid dynorphin A analogues for the bradykinin receptors

作者：Yeon Sun Lee^a ; ^{yeon@email.arizona.edu" class="auth_mail" title="E-mail the corresponding author} ; Michael Remesic^a ; Cyf Ramos-Colon^a ; Sara M. Hall^a ; Alexander Kuzmin^a ; David Rankin^b ; Frank Porreca^b ; Josephine Lai^b ; Victor J. Hruby^a

关键词：BBB ; blood brain barrier ; BK ; bradykinin ; Boc ; t-butyloxycarbonyl ; BR ; bradykinin receptor ; CNS ; central nervous system ; DALKD ; [des-Arg10 ; Leu9]-kallidin ; DIPEA ; diisopropylethylamine ; DMF ; N ; N-dimethylformamide ; Dyn A ; dynorphin A ; Fmoc ; fluorenylmethyloxycarbonyl ; HBTU ; 2-(1H-benzotriazole-1-yl)-113 ; 3-tetramethylaminium hexafluorophosphate ; HOBt ; N-hydroxybenzotriazole ; i.pl. ; intraplantar ; MS ; mass spectroscopy ; Pbf ; 2246 ; 7-pentamethyldihydrobenzofuran-5-sulfonyl ; RP-HPLC ; reversed-phas

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

5.Cyclic peptide-based potent and selective SIRT1/2 dual inhibitors harboring N^ε-thioacetyl-lysine

作者：Di Chen ; Weiping Zheng ; ^{wzheng@ujs.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：β-NAD+ ; β-nicotinamide adenine dinucleotide ; MBHA ; 4-methylbenzhydrylamine ; SPPS ; solid phase peptide synthesis ; DMF ; N ; N-dimethylformamide ; TFA ; trifluoroacetic acid ; DCM ; dichloromethane ; HBTU ; 2-(1H-benzotriazole-1-yl)-113 ; 3-tetramethylaminium hexafluorophosphate ; NMM ; N-methylmorpholine ; RP-HPLC ; reversed-phase high performance liquid chromatography ; HRMS ; high-resolution mass spectrometry ; IC50 ; the inhibitor concentration at which an enzymatic reaction velocity is reduced by 50%

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

6.Design, synthesis and biological evaluation of multifunctional ligands targeting opioid and bradykinin 2 receptors

作者：Srinivas Deekonda^a ; David Rankin^b ; Peg Davis^b ; Josephine Lai^b ; Frank Porreca^b ; Victor J. Hruby^a ; ^{hruby@email.arizona.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：BK ; bradykinin ; BR ; bradykinin receptor ; CNS ; central nervous system ; DALKD ; [des-Arg10 ; Leu9]-kallidin ; Dap ; 2 ; 3-diaminopropionic acid ; DIPEA ; diisopropylethylamine ; DMF ; N ; N-dimethylformamide ; Fmoc ; 9-fluorenylmethoxycarbonyl ; GPI ; guinea pig ileum ; HBTU ; 2-(1H-benzotriazole-1-yl)-113 ; 3-tetramethylaminium hexafluorophosphate ; HCTU ; 2-(6-chloro-1H-benzotriazole-1-yl)-113 ; 3-tetramethylaminium hexafluorophosphate ; HOBt ; N-hydroxybenzotriazole ; PNS ; peripheral nervous system ; RP-HPLC ; reverse

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2015

7.Synthetic peptides for the immunodiagnosis of hepatitis A virus infection

关键词：NMP ; N-Methyl-2-pyrrolidone ; HOBt ; hydroxybenzotriazole ; DIC ; N ; N&prime ; -Diisopropylcarbodiimide ; TFA ; trifluoroacetic acid ; DCM ; dichloromethane ; TIPS ; triisopropylsilane ; TBTU ; 2-(1H-Benzotriazol-1-yl)-113 ; 3-tetramethyluroniumtetrafluoroborate ; DMSO ; dimethyl sulfoxide ; PBS ; phosphate buffered saline ; IMT ; Instituto de Medicina Tropical

刊名：Journal of Immunological Methods

出版年：2015

8.Design and synthesis of novel bivalent ligands (MOR and DOR) by conjugation of enkephalin analogues with 4-anilidopiperidine derivatives

作者：Srinivas Deekonda^a ; Lauren Wugalter^a ; David Rankin^b ; Tally M. Largent-Milnes^b ; Peg Davis^b ; Yue Wang^b ; Neemah M. Bassirirad^b ; Josephine Lai^b ; Vinod Kulkarni^a ; Todd W. Vanderah^b ; Frank Porreca^b ; Victor J. Hruby^a ; ^{hruby@email.arizona.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：ACN ; Acetonitrile ; Boc ; tert-butyloxycarbonyl ; CHO ; Chinese hamster ovary ; DCM ; Dichloromethane ; DIPEA ; N ; N-Diisopropylethylamine ; DALEA ; [D-Ala2 ; Leu5] enkephalin amide ; DAMGO ; [D-Ala2 ; NMePhe4 ; Gly5-ol]enkephalin ; Dmt ; 2 ; 6-dimethyltyrosine ; DPDPE ; c[D-Pen2 ; DPen5]enkephalin ; GPI ; guinea pig isolated ileum ; HBTU ; NN ; N&prime ; N&prime ; -Tetramethyl-O-(1H-benzotriazol-1-yl)uronium hexafluorophosphate ; HATU ; 1-[Bis(dimethylamino)methylene]-1H-12 ; 3-triazolo[4 ; 5-b]pyridinium3-oxid hexafluorophosphate

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2015

9.Potential anticancer activity of benzimidazole-based mono/dinuclear Zn(II) complexes towards human carcinoma cells

作者：Jin&rsquo ; an Zhao^a ; ^{zjinan@zzu.edu.cn" class="auth_mail" title="E-mail the corresponding author} ; Yan Guo^b ; Jiyong Hu^a ; Huaibin Yu^b ; Shuangcheng Zhi^b ; Junshuai Zhang^a

关键词：Zn(II) complexes ; DNA binding ; SHSY5Y cells ; Cytotoxic activity ; Apoptosis

刊名：Polyhedron

出版年：2015

10.Benzotriazoles and benzothiazoles in human urine from several countries: A perspective on occurrence, biotransformation, and human exposure

作者：Alex ; ros G. Asimakopoulos ; Lei Wang ; Nikolaos S. Thomaidis ; Kurunthachalam Kannan

关键词：1H-BTR ; 1H-benzotriazole ; 1-OH-BTR ; 1-hydroxy-benzotriazole ; 4-OH-BTR ; 4-hydroxy-benzotriazole ; 5-OH-BTR ; 5-hydroxy-benzotriazole ; TTR ; tolyltriazole ; 4-Me-1H-BTR ; 4-methyl-1H-benzotriazole ; 5-Me-1H-BTR ; 5-methyl-1H-benzotriazole ; XTR ; or 5 ; 6-diMe-1H-BTR

刊名：Environment International

出版年：2013

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