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在“Elsevier电子期刊”中，命中：655条，耗时：0.0249877 秒

在所有数据库中总计命中：1,243条

1.New bimetallic dicyanidoargentate(I)-based coordination compounds: Synthesis, characterization, biological activities and DNA-BSA binding affinities

作者：Nesrin Korkmaz^a ; Ali Aydın^b ; Ahmet Karadağ^a ; ^{ahmet.karadag@gop.edu.tr} ; Yusuf Yanar^c ; Yelis Maaşoğlu^d ; Ertan Şahin^e ; Şaban Tekin^b

关键词：Dicyanidoargentat(I) ; 2 ; 2&prime ; -(ethylenedioxy)bis(ethylamine) ; Anticancer activity ; Antimicrobial activity ; Antifugal activity ; Apoptosis

刊名：Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy

出版年：2017

2.Design, synthesis and biological evaluation of (E)-3,4-dihydroxystyryl 4-acylaminophenethyl sulfone, sulfoxide derivatives as dual inhibitors of HIV-1 CCR5 and integrase

作者：Yixing Sun^a ; ¹ ; Weisi Xu^b ; ¹ ; Ningning Fan^a ; Xuefeng Sun^a ; Xianling Ning^a ; Liying Ma^b ; ^{mal@chinaaids.cn} ; Junyi Liu^a ; ^c ; ^{jyliu@bjmu.edu.cn} ; Xiaowei Wang^a ; ^{xiaoweiwang@bjmu.edu.cn}

关键词：HIV dual inhibitors ; CCR5 receptor ; HIV integrase ; Sulfones ; Sulfoxides

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

3.Chiral resolution of serial potent and selective σ₁ ligands and biological evaluation of (−)-[¹⁸F]TZ3108 in rodent and the nonhuman primate brain

作者：Xuyi Yue^a ; Hongjun Jin^a ; Zonghua Luo^a ; Hui Liu^a ; Xiang Zhang^a ; Ethan D. McSpadden^b ; Linlin Tian^c ; Hubert P. Flores^c ; Joel S. Perlmutter^a ; ^c ; Stanley M. Parsons^b ; Zhude Tu^a ; ^{tuz@mir.wustl.edu}

关键词：calcd ; calculated ; CH2Cl2 ; dichloromethane ; CNS ; central nervous system ; DMSO ; dimethyl sulfoxide ; [3H]DTG ; [3H]ditolylguanidine ; DTTA ; di-p-toluoyl tartaric acid ; EBP ; emopamil binding protein ; ee ; enantiomeric excess ; EOB ; end of bombardment ; EtOH ; ethanol ; [18F]FTC146 ; 18F-6-(3-fluoropropyl)-3-(2-(azepan-1-yl)ethyl)benzo[d]thiazol-2(3H)-one ; HPLC ; high performance liquid chromatography ; HRMS ; high resolution mass spectrometry ; IC50 ; half maximum inhibitory constant ; K2CO3 ; potassium carbonate

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

4.Array-based functional peptide screening and characterization of gold nanoparticle synthesis

作者：Masayoshi Tanaka^a ; ^b ; Shun Hikiba^a ; Kiyoto Yamashita^a ; Masaki Muto^a ; ^b ; Mina Okochi^a ; ^b ; ^{okochi.m.aa@m.titech.ac.jp}

关键词：AuNP ; gold nanoparticle ; SH ; sulfhydryl ; AuP ; AuNP binding peptides screened with a peptide array ; GRAVY ; grand average of hydropathy ; SEM ; scanning electron microscope ; SPR ; surface plasmon resonance ; TEM ; transmission electron microscopy

刊名：Acta Biomaterialia

出版年：2017

5.Synthesis and biological evaluation of novel 6,7-dihydro-5H-cyclopenta[d]pyrimidine and 5,6,7,8-tetrahydroquinazoline derivatives as sigma-1 (σ₁) receptor antagonists for the treatment of pain

作者：Yu Lan ; Yiyan Songyang ; Lingli Zhang ; Yan Peng ; Jinchun Song ; ^{songjcwhu@163.com" class="auth_mail" title="E-mail the corresponding author}

关键词：σ1R ; sigma-1 receptor ; σ2R ; sigma-2 receptor ; NMDA ; N-methyl-d-aspartate ; CNS ; central nervous system ; PNS ; peripheral nervous system ; KO ; knockout ; WT ; wild-type ; [3H]-DTG ; [3H]-di-o-tolylguanidine ; SAR ; structure-active relationship ; FRET ; fluorescence resonance energy transfer ; ip ; intraperitoneal injection

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

6.Comparison of the primary structures, cytotoxicities, and affinities to phospholipids of five kinds of cytotoxins from the venom of Indian cobra, Naja naja

作者：Mieko Suzuki-Matsubara^a ; ^{m.suzuki@nsc.nagoya-cu.ac.jp" class="auth_mail" title="E-mail the corresponding author} ; Senarath B.P. Athauda^b ; Yoshiyuki Suzuki^a ; Kazumi Matsubara^a ; ¹ ; Akihiko Moriyama^a

关键词：CTX ; cytotoxin ; PBS ; phosphate buffered saline ; PC ; phosphatidylcholine ; PS ; phosphatidylserine ; PE ; phosphatidylethanolanine ; PA ; phosphatidic acid ; SM ; sphingomyeline ; PE ; phosphatidylethanolamine ; dN ; number of nucleotide substitutions per nonsynonymous site ; dS ; number of nucleotide substitutions per synonymous site

刊名：Comparative Biochemistry and Physiology, Part C

出版年：2016

7.Binding affinities of Schiff base Fe(II) complex with BSA and calf-thymus DNA: Spectroscopic investigations and molecular docking analysis

作者：Suparna Rudra ; Somnath Dasmandal ; Chiranjit Patra ; Arjama Kundu ; Ambikesh Mahapatra

关键词：Schiff base ; Fe(II) complex ; Serum albumin ; ct-DNA

刊名：Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy

出版年：2016

8.Enkephalin analogues with N-phenyl-N-(piperidin-2-ylmethyl)propionamide derivatives: Synthesis and biological evaluations

作者：Srinivas Deekonda^a ; Jacob Cole^a ; Sydney Sunna^a ; David Rankin^b ; Tally M. Largent-Milnes^b ; Peg Davis^b ; Neemah M. BassiriRad^b ; Josephine Lai^b ; Todd W. Vanderah^b ; Frank Porecca^b ; Victor J. Hruby^a ; ^{hruby@email.arizona.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：ACN ; acetonitrile ; Boc ; tert-butyloxycarbonyl ; CHO ; Chinese hamster ovary ; DAMGO ; [D-Ala2 ; NMePhe4 ; Gly5-ol]enkephalin ; DALEA ; [D-Ala2 ; Leu5] enkephalin amide ; DCM ; dichloromethane ; DIPEA ; N ; N-diisopropylethylamine ; HBTU ; NN ; N&prime ; N&prime ; -tetra methyl-O-(1H-benzotriazol-1-yl)uronium hexafluorophosphate ; hDOR ; human δ opioid receptor ; Dmt ; 2 ; 6-dimethyltyrosine ; DPDPE ; c[D-Pen2 ; DPen5]enkephalin ; GPI ; guinea pig isolated ileum ; HATU ; 1-[bis(dimethylamino)methylene]-1H-12 ; 3-triazolo[4 ; 5-b]pyridi

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

9.Synthesis of 4-substituted nipecotic acid derivatives and their evaluation as potential GABA uptake inhibitors

作者：Tim Hellenbrand ; Georg Hö ; fner ; Thomas Wein ; Klaus T. Wanner ; ^{klaus.wanner@cup.uni-muenchen.de" class="auth_mail" title="E-mail the corresponding author}

关键词：GABA uptake ; mGAT1 ; Nipecotic acid ; Suzuki&ndash ; Miyaura reaction ; Biological evaluation

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

10.Synthesis and biological evaluation of ranitidine analogs as multiple-target-directed cognitive enhancers for the treatment of Alzheimer’s disease

作者：Jie Gao^a ; ^b ; Narasimha Midde^a ; Jun Zhu^a ; Alvin V. Terry^b ; Campbell McInnes^a ; ^{mcinnes@sccp.sc.edu" class="auth_mail" title="E-mail the corresponding author} ; James M. Chapman^a

关键词：Acetylcholinesterase ; Alzheimers Disease ; Multi-target ; Ranitidine

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

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