搜索页_+Kappa+antagonist

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在“Elsevier电子期刊”中，命中：488条，耗时：0.0119946 秒

在所有数据库中总计命中：632条

1.N-[¹⁸F]-FluoropropylJDTic for κ-opioid receptor PET imaging: Radiosynthesis, pre-clinical evaluation, and metabolic investigation in comparison with parent JDTic

作者：Sé ; bastien Schmitt ; Jé ; rô ; me Delamare ; Olivier Tirel ; Fabien Fillesoye ; Martine Dhilly ; Cé ; cile Perrio ; ^{perrio@cyceron.fr}

关键词：kappa Opioid receptor ; PET imaging ; JDTic ; Fluorine-18 ; Metabolism ; N-fluoroalkylation

刊名：Nuclear Medicine and Biology

出版年：2017

2.Evaluation of CERC-501, a selective kappa opioid antagonist in preclinical models of alcoholism

刊名：Drug and Alcohol Dependence

出版年：2017

3.Synergistic antidepressant-like effects between a kappa opioid antagonist (LY2444296) and a delta opioid agonist (ADL5859) in the mouse forced swim test

作者：Peng Huang ; Julia Tunis ; Christopher Parry ; Ronald Tallarida ; Lee-Yuan. Liu-Chen ; ^{lliuche@temple.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：Kappa opioid antagonist ; Delta opioid agonist ; Antidepressant ; Synergy ; Forced swim test

刊名：European Journal of Pharmacology

出版年：2016

4.Two short-acting kappa opioid receptor antagonists (zyklophin and LY2444296) exhibited different behavioral effects from the long-acting antagonist norbinaltorphimine in mouse anxiety tests

作者：Peng Huang^a ; Tatyana Yakovleva^b ; Jane V. Aldrich^b ; Julia Tunis^a ; Christopher Parry^a ; Lee-Yuan Liu-Chen^a ; ^{lliuche@temple.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：5&prime ; -GNTI ; 5&prime ; -guanidinonaltrindole ; ANOVA ; analysis of variance ; AZ-ECPC ; ethyl 4-(3-carbamoylbenzyl)-1-(cyclohexylmethyl)piperidine-4-carboxylate ; AZ-MTAB ; 3-((1R ; 3r ; 5S)-8-((5-methylthiophen-2-yl)methyl)-8-azabicyclo[3.2.1]octan-3-yloxy)benzamide ; DOPR ; delta opioid receptor ; EPM ; elevated plus maze ; FST ; forced swim test ; i.p. ; intraperitoneal (ly) ; JDTic ; (3R)-7-hydroxy-N-[(2S)-1-[(3R ; 4R)-4-(3-hydroxyphenyl)-3 ; 4-dimethylpiperidin-1-yl]-3-methylbutan-2-yl]-123 ; 4-tetrahydroisoquinol

刊名：Neuroscience Letters

出版年：2016

5.Development of a robust, sensitive and selective liquid chromatography-tandem mass spectrometry assay for the quantification of the novel macrocyclic peptide kappa opioid receptor antagonist [D-Trp]CJ-15,208 in plasma and application to an initial pharmacokinetic study

作者：Tanvir Khaliq^a ; ^c ; Todd D. Williams^b ; Sanjeewa N. Senadheera^a ; ¹ ; Jane V. Aldrich^a ; ^c ; ^{janealdrich@ufl.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：CV ; coefficient of variation ; [D-Trp]CJ-15 ; 208 ; cyclo[Phe-d-Pro-Phe-d-Trp] ; KOR ; kappa opioid receptor ; LLQ ; lower limit of quantitation ; MRM ; multiple reaction monitoring ; MS/MS ; tandem mass spectrometry ; QC ; quality control

刊名：Journal of Chromatography B, Analytical Technologies in the Biomedical and Life Sciences

出版年：2016

6.Potent ameliorating effect of Hypoxia-inducible factor 1α (HIF-1α) antagonist YC-1 on combined allergic rhinitis and asthma syndrome (CARAS) in Rats

作者：Xu Wang ; Chun Liu ; Liucheng Wu ; Shunxing Zhu ; ^{zsx@ntu.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：HIF-1α ; Combined allergic rhinitis and asthma syndrome ; YC-1 ; Inflammation ; Rat

刊名：European Journal of Pharmacology

出版年：2016

7.Bisphenol A exposure alters release of immune and developmental modulators and expression of estrogen receptors in human fetal lung fibroblasts

作者：Laziyan Mahemuti¹ ; ⁵ ; ^{Mahemuti_Laziyan@hc-sc.gc.ca" class="auth_mail" title="E-mail the corresponding author} ; Qixuan Chen¹ ; Melanie C. Coughlan¹ ; Min Zhang¹ ; Maria Florian¹ ; ⁵ ; Ryan J. Mailloux¹ ; ⁵ ; Xu-Liang Cao² ; Kylie A. Scoggan³ ; ⁴ ; William G. Willmore⁵ ; Xiaolei Jin¹ ; ^{Dawn_Jin@hc-sc.gc.ca" class="auth_mail" title="E-mail the corresponding author} ; ^{jxnc329@gmail.com" class="auth_mail" title="E-mail the corresponding author}

关键词：Bisphenol A ; Human fetal lung fibroblasts ; Estrogen receptors ; Antagonists ; Cytokines ; Chemokines ; Immune and developmental modulators

刊名：Journal of Environmental Sciences

出版年：2016

8.Resveratrol inhibits inflammatory signaling implicated in ionizing radiation-induced premature ovarian failure through antagonistic crosstalk between silencing information regulator 1 (SIRT1) and poly(ADP-ribose) polymerase 1 (PARP-1)

作者：Riham Soliman Said^a ; Ebtehal El-Demerdash^b ; ^{ebtehal_dm@yahoo.com" class="auth_mail" title="E-mail the corresponding author} ; ^{ebtehal_dm@pharma.asu.edu.eg" class="auth_mail" title="E-mail the corresponding author} ; Ahmed Shafik Nada^a ; Mohamed M. Kamal^c

关键词：AMH ; anti-Mü ; llerian hormone ; COX-2 ; cyclooxygenase-2 ; IL ; interleukin ; iNOS ; inducible nitric oxide synthase ; NF-κB ; nuclear factor kappa-B ; PARP ; poly(ADP-ribose) polymerase ; POF ; premature ovarian failure ; PPARs ; peroxisome proliferator-activated receptors ; Sir2 ; silent information regulator 2 ; SIRT1 ; silencing information regulator 1 ; TBS ; Tris buffered saline

刊名：Biochemical Pharmacology

出版年：2016

9.Species differences in the effects of the κ-opioid receptor antagonist zyklophin

作者：Sunil Sirohi^a ; ^b ; Jane V. Aldrich^e ; Brendan M. Walker^a ; ^b ; ^c ; ^d ; ^{b_walker@wsu.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：Alcohol dependence and withdrawal ; GTPyS coupling ; Kappa-opioid receptor ; Alcohol self-administration ; Zyklophin

刊名：Alcohol

出版年：2016

10.The effect of some immunomodulatory and anti-inflammatory drugs on Li-pilocarpine-induced epileptic disorders in Wistar rats

作者：Layla E. Borham^a ; ^b ; ^{borhaml@hotmail.com" class="auth_mail" title="E-mail the corresponding author} ; Amal M. Mahfoz^a ; ^c ; Ibrahim A.A. Ibrahim^a ; Naiyer Shahzad^a ; Abeer Ahmed ALrefai^d ; Amira A. Labib^e ; Bassam Bin Sef^f ; Abdulrahmman Alshareef^f ; Meshal Khan^f ; Ali Milibary^f ; Saeed Al Ghamdi^a

关键词：BBB ; blood brain barrier ; CA ; catecholamine ; IFN-γ ; interferon-gamma ; IL ; interleukin ; IL-1R ; interleukin-1 receptor ; IL-1Ra ; interleukin-1 receptor antagonist ; IL-6R ; IL-6 receptor ; IP ; intraperitoneal ; NF-kB ; nuclear factor kappaB ; NMDA ; N-methyl-d-aspartic acid ; PBMCs ; peripheral blood mononuclear cells ; PTZ ; Pentylenetetrazol ; PO ; oral ; SC ; subcutaneous ; SE ; status epilepticus ; SNS ; sympathetic nervous system ; TLE ; temporal lobe epilepsy ; TNFα ; tumor necrosis factor α ; AEDs ; antiepileptic dr

刊名：Brain Research

出版年：2016

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