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在“Elsevier电子期刊”中，命中：63,703条，耗时：0.0579733 秒

在所有数据库中总计命中：74,653条

1.The efficacy and safety of adrenergic alpha-antagonists in treatment of distal ureteral stones in pediatric patients: A systematic review and meta-analysis

作者：Daxue Tian ; Nan Li ; Wei Huang ; Huantao Zong ; Yong Zhang ; ^{758980179@qq.com}

关键词：Adrenergic alpha-antagonists ; Pediatrics ; Distal ureteral stones ; Meta-analysis ; Randomized controlled trials

刊名：Journal of Pediatric Surgery

出版年：2017

2.A novel and selective melanin-concentrating hormone receptor 1 antagonist ameliorates obesity and hepatic steatosis in diet-induced obese rodent models

作者：Yayoi Kawata^a ; ^{yayoi.kawata@takeda.com} ; Shoki Okuda^a ; Natsu Hotta^a ; Hideyuki Igawa^a ; Masashi Takahashi^a ; Minoru Ikoma^a ; Shizuo Kasai^a ; Ayumi Ando^a ; Yoshinori Satomi^a ; Mayumi Nishida^a ; Masaharu Nakayama^a ; Syunsuke Yamamoto^a ; Yasutaka Nagisa^a ; ¹ ; Shiro Takekawa^a

关键词：Melanin-concentrating hormone 1 receptor antagonist ; Obesity ; Non-alcoholic fatty liver disease

刊名：European Journal of Pharmacology

出版年：2017

3.Approaches to improve metabolic stability of a statine-based GRP receptor antagonist

作者：Ilinca Popp^a ; Luigi Del Pozzo^a ; ^b ; ^c ; Beatrice Waser^d ; Jean Claude Reubi^d ; Philipp T. Meyer^a ; ^b ; ^c ; Helmut R. Maecke^a ; Eleni Gourni^a ; ^b ; ^c ; ^{eleni.gourni@medisin.uio.no}

关键词：Gastrin-releasing peptide receptor antagonists ; Metabolic stability ; 68Ga ; PET-imaging

刊名：Nuclear Medicine and Biology

出版年：2017

4.Synthesis and optimization of novel α-phenylglycinamides as selective TRPM8 antagonists

作者：Jun-ichi Kobayashi ; ^{jun-ichi_kobayashi@pharm.kissei.co.jp} ; Hideaki Hirasawa ; Tetsuji Ozawa^a ; Tomonaga Ozawa ; Hiroo Takeda ; Yoshikazu Fujimori ; Osamu Nakanishi ; Noboru Kamada ; Tetsuya Ikeda^b

关键词：TRPM8 ; TRPM8 antagonist ; Phenylglycinamide ; KPR-2579 ; Ugi reaction ; OAB

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

5.Structure-activity relationships of benzothiazole GPR35 antagonists

作者：Manahil M. Abdalhameed^a ; Pingwei Zhao^b ; Dow P. Hurst^a ; Patricia H. Reggio^a ; ^{phreggio@uncg.edu} ; Mary E. Abood^b ; ^{mabood@temple.edu} ; Mitchell P. Croatt^a ; ^{mpcroatt@uncg.edu}

关键词：GPR35 ; Antagonist ; G protein-coupled receptor ; Benzothiazole ; SAR

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

6.Combined effect of antagonistic yeast and modified atmosphere to control Penicillium expansum infection in sweet cherries cv. Ambrunés

作者：E. de Paiva^a ; ^b ; M.J. Serradilla^c ; S. Ruiz-Moyano^a ; ^b ; M.G. Có ; rdoba^a ; ^b ; M.C. Villalobos^a ; ^b ; R. Casquete^a ; ^b ; A. Herná ; ndez^a ; ^b ; ^{ahernandez@unex.es} ;

关键词：Antagonistic yeast ; Disease incidence ; Disease severity ; Modified atmospheres ; Penicillium expansum

刊名：International Journal of Food Microbiology

出版年：2017

7.Escape from adamantane: Scaffold optimization of novel P2X7 antagonists featuring complex polycycles

作者：Marta Barniol-Xicota^a ; Seung-Hwa Kwak^b ; So-Deok Lee^b ; Emily Caseley^c ; Elena Valverde^a ; Lin-Hua Jiang^c ; Yong-Chul Kim^b ; ^{yongchul@gist.ac.kr} ; Santiago Vá ; zquez^a ; ^{svazquez@ub.edu}

关键词：Adamantane ; Drug discovery ; Homology models ; P2X7 antagonists ; Scaffold replacement

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

8.An evaluation of central penetration from a peripherally administered oxytocin receptor selective antagonist in nonhuman primates

作者：Aaron L. Smith^a ; ^b ; ^c ; ^{asmit53@emory.edu} ; Hasse Walum^a ; Fawn Connor-Stroud^d ; Sara M. Freeman^e ; Kiyoshi Inoue^a ; Lisa A. Parr^a ; Mark M. Goodman^a ; ^b ; ^c ; Larry J. Young^a

关键词：Oxytocin antagonist ; Oxytocin receptor ; PET imaging ; Rhesus macaque ; Cerebrospinal fluid

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

9.Imidazo[1,2-a]pyrazin-8-amine core for the design of new adenosine receptor antagonists: Structural exploration to target the A₃ and A_2A subtypes

作者：Daniela Poli^a ; Matteo Falsini^a ; Flavia Varano^a ; Marco Betti^a ; Katia Varani^b ; Fabrizio Vincenzi^b ; Anna Maria Pugliese^c ; Felicita Pedata^c ; Diego Dal Ben^d ; Ajiroghene Thomas^d ; Ilaria Palchetti^e ; ^f ; Francesca Bettazzi^e ; Daniela Catarzi^a ; ^{daniela.catarzi@unifi.it} ; Vittoria Colotta^a

关键词：G protein-coupled receptors ; Adenosine receptor antagonists ; Imidazopyrazines ; Bicyclic heteroaromatic systems ; Ligand-receptor modeling studies

刊名：European Journal of Medicinal Chemistry

出版年：2017

10.Influence of chain length on the activity of tripeptidomimetic antagonists for CXC chemokine receptor 4 (CXCR4)

作者：Markus Baumann^a ; Mohammad Musarraf Hussain^a ; ¹ ; Nina Henne^a ; Daniel Moya Garrote^a ; Stefanie Karlshø ; j^b ; Torgils Fossen^a ; Mette M. Rosenkilde^b ; Jon Vå ; benø ; ^c ; ^{jon.vabeno@uit.no} ; Bengt Erik Haug^a ; ^{bengt-erik.haug@farm.uib.no}

关键词：CXCR4 antagonist ; Peptidomimetic ; Scaffold

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

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