搜索页_benzodiazepine+derivative

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在“Elsevier电子期刊”中，命中：357条，耗时：0.0179886 秒

在所有数据库中总计命中：1,040条

1.Synthesis and fluorescence studies of nine 1,5-benzodiazepine-2,4-dione derivatives: Dual emission and excimer fluorescence

作者：Hamid Reza Qomi ; Azizollah Habibi ; ^{habibi@khu.ac.ir} ; Seyyed Mohammad Shahcheragh

关键词：1 ; 5-Benzodiazepine-2 ; 4-dione (BZD) ; Dual fluorescence ; Excimer emission ; Intramolecular charge transfer (ICT) ; Solvatochromism ; Phosphorescence

刊名：Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy

出版年：2017

2.Design and synthesis of benzodiazepine analogs as isoform-selective human lysine deacetylase inhibitors

作者：D. Rajasekhar Reddy ; Flavio Ballante ; Nancy J. Zhou ; Garland R. Marshall ; ^{garlandm@gmail.com}

关键词：Epigenetics ; Histone deacetylase (HDAC) ; Lysine deacetylase (KDAC) ; Benzodiazepine (BZD) ; Structure-based drug design (SBDD)

刊名：European Journal of Medicinal Chemistry

出版年：2017

3.Derivatives of the pyrazolo[1,5-a]pyrimidine acetamide DPA-713 as translocator protein (TSPO) ligands and pro-apoptotic agents in human glioblastoma

作者：Eryn L Werry^a ; ¹ ; Victoria A. King^b ; ¹ ; Melissa L Barron^a ; Samuel D. Banister^c ; Renee Sokias^c ; Michael Kassiou^c ; ^{michael.kassiou@sydney.edu.au}

关键词：BrdU ; 5-bromo-2&prime ; -deoxyuridine ; DMEM/F12 ; Dulbecco's modified eagle's medium ; Ham's nutrient mixture F-12 ; DMSO ; dimethyl sulfoxide ; EDTA ; ethylenediaminetetraacetic acid ; LLE ; lipophilic ligand efficiency ; MEM ; minimum essential medium ; PET ; positron emission tomography ; SPECT ; single-photon emission computed tomography ; TSPO ; translocator protein

刊名：European Journal of Pharmaceutical Sciences

出版年：2017

4.Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH₃ or 2-CH₃

作者：Agnieszka Gunia-Krzyżak^a ; ^{agnieszka.gunia@uj.edu.pl} ; Dorota Żelaszczyk^a ; Anna Rapacz^b ; Ewa Żesławska^c ; Anna M. Waszkielewicz^a ; Katarzyna Pańczyk^a ; Karolina Słoczyńska^d ; Elżbieta Pękala^d ; Wojciech Nitek^e ; Barbara Filipek^b ; Henryk Marona^a

关键词：Anticonvulsant ; Cinnamamide ; Crystal structure ; MES ; Pharmacophore ; scPTZ ; 6-Hz

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

5.Palladium-benzodiazepine derivatives as promising metallodrugs for the development of antiepileptic therapies

关键词：Palladacycles ; Diazepam ; Benzodiazepine ; Convulsion ; Epilepsy

刊名：Journal of Inorganic Biochemistry

出版年：2016

6.A novel 2,3-benzodiazepine-4-one derivative AMPA antagonist inhibits G₂/M transition and induces apoptosis in human leukemia Jurkat T cell line

作者：S. Parenti^a ; ^{sandra.parenti@unimore.it" class="auth_mail" title="E-mail the corresponding author} ; G. Casagrande^a ; ^{85570@studenti.unimore.it" class="auth_mail" title="E-mail the corresponding author} ; M. Montanari^a ; ^{monica.montanari@unimore.it" class="auth_mail" title="E-mail the corresponding author} ; M. Espahbodinia^b ; ^{mespahbodinia@unime.it" class="auth_mail" title="E-mail the corresponding author} ; R. Ettari^b ; ^{roberta.ettari@unime.it" class="auth_mail" title="E-mail the corresponding author} ; A. Grande^a ; ^{alexis.grande@unimore.it" class="auth_mail" title="E-mail the corresponding author} ; L. Corsi^a ; ^{corsi.lorenzo@unimore.it" class="auth_mail" title="E-mail the corresponding author}

关键词：AMPA ; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate ; CNS ; central nervous system ; DMSO ; dimethyl sulfoxide ; RK 1/2 ; extracellular-signal-regulated kinases 1/2 ; MAPK ; mitogen-activated protein kinase

刊名：Life Sciences

出版年：2016

7.An overview of emerging and new psychoactive substances in the United Kingdom

作者：Shruti Beharry ; Simon Gibbons ; ^{simon.gibbons@ucl.ac.uk" class="auth_mail" title="E-mail the corresponding author}

关键词：New psychoactive substances ; Psychostimulants ; Lefetamine ; Hallucinogens ; LSD derivatives ; Benzodiazepines

刊名：Forensic Science International

出版年：2016

8.A fatal intoxication related to MDPV and pentedrone combined with antipsychotic and antidepressant substances in Cyprus

作者：Katerina Liveri¹ ; ^{kliveri@sgl.moh.gov.cy" class="auth_mail" title="E-mail the corresponding author} ; ^{maconstantinou@sgl.moh.gov.cy" class="auth_mail" title="E-mail the corresponding author} ; Maria A. Constantinou¹ ; Maria Afxentiou ; Popi Kanari

关键词：Multidrug intoxication ; Bath salts ; Designer benzodiazepines ; Postmortem ; Gas chromatography-mass spectrometry

刊名：Forensic Science International

出版年：2016

9.Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agents

作者：Roberta Ettari^a ; Santo Previti^a ; Sandro Cosconati^b ; Santina Maiorana^a ; Tanja Schirmeister^c ; Silvana Grasso^a ; Maria Zappalà ; ^a ; ^{mzappala@unime.it" class="auth_mail" title="E-mail the corresponding author}

关键词：Trypanosoma ; Peptidomimetics ; Michael acceptors ; Microwave irradiation ; Pharmacokinetic parameters

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

10.Implication of coumarins towards central nervous system disorders

作者：Krystyna Skalicka-Woźniak^a ; ^{kskalicka@pharmacognosy.org" class="auth_mail" title="E-mail the corresponding author} ; Ilkay Erdogan Orhan^b ; Geoffrey A. Cordell^c ; ^d ; Seyed Mohammad Nabavi^e ; Barbara Budzyńska^f

关键词：Coumarins ; Central nervous system ; γ-Aminobutyric acid (GABA) ; Benzodiazepine receptors ; Monoamine oxidase (MAO) inhibitors ; Cholinesterase inhibitors

刊名：Pharmacological Research

出版年：2016

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