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在“Elsevier”中，命中：68条，耗时：0.076963 秒

1.Design and synthesis of 3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-quinolin-2-ones as VEGFR-2 kinase inhibitors

作者：Sun-Young Han^a ; ^b ; Jie Won Choi^a ; ^c ; Jeon Yang^a ; ^d ; Chong Hack Chae^a ; Jongkook Lee^a ; Heejung Jung^a ; Kwangho Lee^a ; Jae Du Ha^a ; ; Hyoung Rae Kim^a ; Sung Yun Cho^a ; ^{sycho@krict.re.kr}

关键词：Cancer ; VEGFR-2 ; KDR kinase ; Imidazo[4 ; 5-c]pyridine ; Quinolin-2-one

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2012

2.A new series of N⁵ derivatives of the 1,1,5-trimethyl furo[3,4-c]pyridine-3,4-dione (cerpegin) selectively inhibits the post-acid activity of mammalian 20S proteasomes

作者：The Hien Pham^a ; ^&dagger ; ; ^{hien_fr@yahoo.fr} ; Anna Hovhannisyan^b ; ^&dagger ; ; ^{annahovh@gmail.com} ; Dominique Bouvier^c ; ^{dbouvier@snv.jussieu.fr} ; Lei Tian^a ; ^{leon-0315@hotmail.com} ; Michè ; le Reboud-Ravaux^a ; ^{Michele.Reboud@upmc.fr} ; Gagik Melikyan^b ; ^{suren@netsys.am} ; Michelle Bouvier-Durand^a ; ^{mbouvier@snv.jussieu.fr}

关键词：DMF/DMA ; dimethylformamide/dimethylacetal ; DMSO ; dimethyl sulfoxide ; 20S ; 20S proteasome catalytic core ; CT-L ; chymotrypsin-like ; T-L ; trypsin-like ; PA ; post-acid or caspase-like ; AMC ; 7-amino-4-methyl-coumarin ; 尾-NA ; 尾-naphthylamide ; PDB ; Protein Data

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2012

3.Regulation of the surface expression of 伪4尾2未 GABA_A receptors by high efficacy states

作者：Aarti Kuver ; Hui Shen ; Sheryl S. Smith ; ^{Sheryl.smith@downstate.edu}

关键词：伪4F ; 伪4FLAG (3xFLAG tag) ; BDNF ; Brain-derived neurotrophic factor ; DMSO ; dimethyl sulfoxide ; FLAG ; DYKDDDDK epitope ; GABAR ; GABAA receptor ; GBX ; Gaboxadol ; 456 ; 7-tetrahydroisoxazolo(5 ; 4-c)pyridin-3-ol ; THIP ; HEK-293 ; human embryonic kidney cell-293 ; P

刊名：Brain Research

出版年：2012

4.1,3-Dipolar cycloaddition reaction of 3-trifluoromethyl-4-diazopyrazolinones with acetylenedicarboxylates

作者：Zhenhua Zhang^a ; Xiaowei Wang^a ; Song Tao^a ; ^b ; Shizheng Zhu^a ; ^{zhusz@mail.sioc.ac.cn}

关键词：3-Trifluoromethyl-4-diazopyrazolinone ; Acetylenedicarboxylate ; [3+2] Dipolar cycloaddition ; Furo[2 ; 3-c]pyrazole ; Pyrazolotriazine

刊名：Tetrahedron

出版年：2012

5.InCl₃-promoted a novel Prins cyclization for the synthesis of hexahydro-1H-furo[3,4-c]pyran derivatives

作者：B.V. Subba Reddy ; ^{basireddy@iict.res.in} ; Marepally Sreelatha ; Ch. Kishore ; Prashant Borkar ; J.S. Yadav

关键词：Indium(III) chloride ; Bicyclic ethers ; Prins cyclization ; cis-Fused furopyrans

刊名：Tetrahedron Letters

出版年：2012

6.Thieno[3,2-c]pyran-4-one based novel small molecules: Their synthesis, crystal structure analysis and in vitro evaluation as potential anticancer agents

作者：Ali Nakhi^a ; Raju Adepu^a ; D. Rambabu^a ; Ravada Kishore^b ; G.R. Vanaja^c ; Arunasree M. Kalle^c ; Manojit Pal^a ; ^{manojitpal@rediffmail.com}

关键词：Thienopyranone ; Alkynylation ; Iodocyclization ; Sonogashira ; Heck ; Suzuki

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2012

7.Design, synthesis, and antiproliferative activity of new 1H-pyrrolo[3,2-c]pyridine derivatives against melanoma cell lines. Part 2

作者：Myung-Ho Jung^a ; Mohammed I. El-Gamal^a ; ^b ; ^d ; Mohammed S. Abdel-Maksoud^a ; ^b ; Taebo Sim^c ; Kyung Ho Yoo^c ; Chang-Hyun Oh^a ; ^b ; ^{choh@kist.re.kr}

关键词：Pyrrolo[3 ; 2-c]pyridine ; A375P ; Antiproliferative activity ; Melanoma ; Diarylurea ; Diarylamide

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2012

8.Steroidal C-21 heteroaryl thioethers. Part 3: Pregn-4-eno-[3,2-c]pyrazole fused A ring modified steroids as selective glucocorticoid receptor modulators (dissociated steroids)

作者：Purakkattle Biju ; ^{purakkattle.biju@merck.com} ; Hongwu Wang ; John Anthes ; Kevin McCormick ; Robert Aslanian ; Michael Berlin ; Rema Bitar ; Yeon-Hee Lim ; Yoon Joo Lee ; Daniel Prelusky ; Robbie Mcleod ; Yanlin Jia ; Xiomora Fernandez ; Gissela Lieber ; Johanna Jimenez ; Steve Eckel ; Aileen House ; Richard Chapman ; Jonathan Phillips

关键词：Selective glucocorticoid receptor modulators ; Dissociated steroids ; Prednisolone ; Transactivation ; Transrepression ; Pyrazole

刊名：Bioorganic and Medicinal Chemistry Letters

出版年：2012

9.The selective metabotropic glutamate receptor 7 allosteric agonist AMN082 prevents reinstatement of extinguished ethanol-induced conditioned place preference in mice

作者：Amine Bahi ; ^{amine.bahi@uaeu.ac.ae}

关键词：AMN082 ; N ; N&prime ; -Bis(diphenylmethyl)-1 ; 2-ethanediamine dihydrochloride ; BEC ; blood ethanol concentrations ; CPP ; conditioned place preference ; mGluR ; metabotropic glutamate receptor ; MMPIP ; 6-(4-methoxyphenyl)-5-methyl-3-(4-pyridinyl)-isoxazolo[4 ; 5-c]pyr

刊名：Pharmacology Biochemistry and Behavior

出版年：2012

10.Synthesis of pyrrolo[3,4-b]pyrroles and perhydrothiazolo[3′,4′-2,3]pyrrolo[4,5-c]pyrroles

作者：Mahalingam Poornach ; ran ; Raghavachary Raghunathan

关键词：Pyrrolidine ; Pyrrolo[3 ; 4-b]pyrrole ; Cycloaddition ; Heterotricycle ; Perhydrothiazolo[3′ ; 4′ ; -2 ; 3]pyrrolo[4 ; 5-c]pyrrole ; Stereoselective ; Azomethine ylide ; Alkenyl aldehyde

刊名：Tetrahedron

出版年：2008

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