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在“Elsevier电子期刊”中，命中：3,984条，耗时：0.0839591 秒

在所有数据库中总计命中：9,809条

1.Cocaine self-administration, extinction training and drug-induced relapse change metabotropic glutamate mGlu5 receptors expression: Evidence from radioligand binding and immunohistochemistry assays

作者：Lucyna Pomierny-Chamiolo^a ; ^{lpomiern@cm-uj.krakow.pl} ; Joanna Miszkiel^b ; Malgorzata Frankowska^b ; Beata Bystrowska^a ; Malgorzata Filip^b

关键词：Cocaine self-administration ; Extinction training ; Drug-induced relapse ; MGlu5 receptor binding ; MGlu5 receptor immunohistochemistry

刊名：Brain Research

出版年：2017

2.Pharmacological studies on the NOP and opioid receptor agonist PWT2-[Dmt¹]N/OFQ(1-13)

作者：Maria Camilla Cerlesi^a ; Huiping Ding^b ; Mark F. Bird^c ; Norikazu Kiguchi^b ; Federica Ferrari^a ; Davide Malfacini^a ; Anna Rizzi^a ; Chiara Ruzza^a ; David G. Lambert^c ; Mei-Chuan Ko^b ; Girolamo Calo^a ; ; Remo Guerrini^d

关键词：PWT2-[Dmt1]N/OFQ(1&ndash ; 13) ; NOP and opioid receptors ; Receptor binding ; Stimulation of [35S]GTPγS binding ; Calcium mobilization ; Monkey spinal analgesia

刊名：European Journal of Pharmacology

出版年：2017

3.High affinity binding of the peptide agonist TIP-39 to the parathyroid hormone 2 (PTH₂) receptor requires the hydroxyl group of Tyr-318 on transmembrane helix 5

作者：Richard E. Weaver^a ; Juan C. Mobarec^c ; Mark J. Wigglesworth^b ; ¹ ; Christopher A. Reynolds^c ; Dan Donnelly^a ; ^{d.donnelly@leeds.ac.uk}

关键词：Parathyroid hormone ; PTH ; GPCR ; Agonist ; Receptor ; TIP39

刊名：Biochemical Pharmacology

出版年：2017

4.Characterization of P2X4 receptor agonists and antagonists by calcium influx and radioligand binding studies

作者：Aliaa Abdelrahman^a ; Vigneshwaran Namasivayam^a ; ^c ; Sonja Hinz^a ; Anke C. Schiedel^a ; Meryem Kö ; se^a ; Maggi Burton^b ; Ali El-Tayeb^a ; ¹ ; Michel Gillard^b ; Jü ; rgen Bajorath^c ; Marc de Ryck^b ; Christa E. Mü ; ller^a ; ^{christa.mueller@uni-bonn.de}

关键词：Ap3A ; diadenosine triphosphate ; Ap4A ; diadenosine tetraphosphate ; Ap5A ; diadenosine pentaphosphate ; AR-C67085MX ; 2-propylthio-β ; γ-dichloromethylene-ATP ; PSB0412 ; 2-propargylthio-β ; γ-dichloromethylene-ATP ; 5-BDBD ; 5-(3-bromophenyl)-1 ; 3-dihydro-2H-benzofuro[3 ; 2-e]-1 ; 4-diazepin-2-one ; BzATP ; 2&prime ; (3&prime ; )-O-(4-benzoylbenzoyl)adenosine 5&prime ; -triphosphate ; CHO-K1 cells ; Chinese hamster ovary cells ; HBSS ; Hank&rsquo ; s balanced salt solution ; HEPES ; 4-(2-hydroxyethyl)-1-piperazine ethanesulfoni

刊名：Biochemical Pharmacology

出版年：2017

5.A benzo[b]thiophene-based selective type 4 S1P receptor agonist

作者：Wooyoung Hur^a ; ¹ ; Hugh Rosen^b ; Nathanael S. Gray^a ; ^{Nathanael_Gray@dfci.harvard.edu}

关键词：Sphingosine-1-phosphate ; S1P receptor ; S1PR4 ; S1P4 ; Selective agonist

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

6.New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking

作者：Giulio Ragusa^a ; Marí ; a Gó ; mez-Cañ ; as^b ; ^c ; ^d ; Paula Morales^e ; Carmen Rodrí ; guez-Cueto^b ; ^c ; ^d ; Marí ; a R. Pazos^b ; ^c ; ^d ; Battistina Asproni^a ; Elena Cichero^f ; Paola Fossa^f ; Gerard A. Pinna^a ; Nadine Jagerovic^e ; Javier Ferná ; ndez-Ruiz^b ; ^c ; ^d ; Gabriele Murineddu^a ; ^{muri@uniss.it}

关键词：Scaffold hopping ; Synthesis ; Cannabinoid receptors ; CB2 antagonism ; ADME model ; Docking studies

刊名：European Journal of Medicinal Chemistry

出版年：2017

7.Critical and direct involvement of the CD23 stalk region in IgE binding

作者：Regina Selb ; PhD^a ; Julia Eckl-Dorna ; MD ; PhD^a ; Teresa E. Twaroch ; PhD^b ; Christian Lupinek ; MD^b ; Andrea Teufelberger ; MSc^c ; ^&lowast ; ; Gerhard Hofer ; MSc^c ; Margarete Focke-Tejkl ; PhD^b ; Barbara Gepp ; PhD^d ; Birgit Linhart ; PhD^b ; Heimo Breiteneder ; PhD^d ; Adolf Ellinger ; MD^e ; Walter Keller ; PhD^c ; Kenneth H. Roux ; PhD^f ; Rudolf Valenta ; MD^b ; ^{Rudolf.valenta@meduniwien.ac.at} ; Verena Niederberger ; MD^a

关键词：CD23 ; allergy ; IgE ; low-affinity IgE receptor ; B cell ; allergen

刊名：Journal of Allergy and Clinical Immunology

出版年：2017

8.Design, synthesis and biological evaluation of (E)-3,4-dihydroxystyryl 4-acylaminophenethyl sulfone, sulfoxide derivatives as dual inhibitors of HIV-1 CCR5 and integrase

作者：Yixing Sun^a ; ¹ ; Weisi Xu^b ; ¹ ; Ningning Fan^a ; Xuefeng Sun^a ; Xianling Ning^a ; Liying Ma^b ; ^{mal@chinaaids.cn} ; Junyi Liu^a ; ^c ; ^{jyliu@bjmu.edu.cn} ; Xiaowei Wang^a ; ^{xiaoweiwang@bjmu.edu.cn}

关键词：HIV dual inhibitors ; CCR5 receptor ; HIV integrase ; Sulfones ; Sulfoxides

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

9.In vitro antioxidative and anti-inflammatory effects of the compound K-rich fraction BIOGF1K, prepared from Panax ginseng

作者：Muhammad Jahangir Hossen¹ ; ² ; ^☆ ; Yong Deog Hong³ ; ^☆ ; Kwang-Soo Baek¹ ; Sulgi Yoo¹ ; Yo Han Hong¹ ; Ji Hye Kim¹ ; Jeong-Oog Lee⁴ ; Donghyun Kim³ ; Junseong Park³ ; ^{superbody@amorepacific.com} ; Jae Youl Cho¹ ; ^{jaecho@skku.edu}

关键词：anti-inflammatory activity ; antioxidative activity ; BIOGF1K ; compound K ; Panax ginseng

刊名：Journal of Ginseng Research

出版年：2017

10.Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1

作者：Karolina Grabowska^a ; Anna K. Puszko^a ; Piotr F.J. Lipiński^b ; Anna K. Laskowska^b ; Beata Wileńska^a ; Ewa Witkowska^a ; Gerard Y. Perret^c ; Aleksandra Misicka^a ; ^b ; ^{misicka@chem.uw.edu.pl}

关键词：ABTS ; 2 ; 2&prime ; -azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt ; ACN ; acetonitrile ; BSA ; bovine serum albumin ; (bt)-VEGF165 ; biotinylated-VEGF165 ; 6-Cl-HOBt ; 6-chloro-1-hydroxybenzotriazole dihydrate ; DIPEA ; N ; N-diisopropylethylamine ; DMEM ; Dulbecco&rsquo ; s Modified Eagle Medium ; EGM ; Endothelial Cell Growth Media ; ELISA ; enzyme-linked immunosorbent assay ; FA ; formic acid ; MDA-MB-231 ; human breast adenocarcinoma cells ; MTS ; 3-(4 ; 5-dimethylthiazol-2-yl)-5-(3-carboxymethoxypheny

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

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