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Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors
详细信息
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作者:
Ashvinikumar V. Gavai
;
Claude Quesnelle
;
Derek Norris
;
Wen-Ching Han
;
Patrice Gill
;
Weifang Shan
;
Aaron Balog
;
Ke Chen
;
Andrew Tebben
;
Richard Rampulla
;
Dauh-Rurng Wu
;
Yingru Zhang
;
Arvind
Mathur
;
Ronald White
;
Anne Rose
;
Haiqing Wang
;
Zheng Yang
;
Asoka Ranasinghe
;
Celia D鈥橝rienzo
;
Victor Guarino
;
Lan Xiao
;
Ching Su
;
Gerry Everlof
;
Vinod Arora
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Krista Menard
;
Mei-Li Wen
;
Jere Meredith
;
George Trainor
;
Louis J. Lombardo
;
Richard Olson
;
Phil S. Baran
;
John T. Hunt
;
Gregory D. Vite
;
Bruce S. Fischer
;
Richard A. Westhouse
;
Francis Y. Lee
刊名:ACS Medicinal Chemistry Letters
出版年:2015
出版时间:May 14, 2015
年:2015
卷:6
期:5
页码:523-527
全文大小:316K
ISSN:1948-5875
文摘
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