An efficient synthesis of 1-thioamidoalkyl-2-naphthol derivatives

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• 作者：Hamid Reza Shaterian ; Kobra Azizi ; Nafiseh Fahimi
• 关键词：P2O5–SiO2 ; 1 ; Thioamidoalkyl ; 2 ; naphthol ; N ; Phenylthiourea ; Heterogeneous catalyst ; Solvent ; free
• 刊名：Research on Chemical Intermediates
• 出版年：2014
• 出版时间：October 2014
• 年：2014
• 卷：40
• 期：8
• 页码：2613-2620
• 全文大小：246 KB
• 参考文献：1. T. Dingermann, D. Steinhilber, G. Folkers, / Molecular Biology in Medicinal Chemistry (Wiley–VCH, Weinheim, 2004)
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• 作者单位：Hamid Reza Shaterian (1)
  Kobra Azizi (1)
  Nafiseh Fahimi (1)
  
  1. Department of Chemistry, Faculty of Sciences, University of Sistan and Baluchestan, PO Box 98135-674, Zahedan, Iran
  
• ISSN：1568-5675

文摘

The discovery and development of phosphorus pentoxide supported on silica gel (P2O5-a href='/search?dc.title=SiO&facet-content-type=ReferenceWorkEntry&sortOrder=relevance' class='reference-link webtrekk-track' gaCategory="Internal link" gaLabel="SiO" gaAction="reference keyword">SiO2) as an efficient catalyst has led to an efficient method for the direct preparation of 1-thioamidoalkyl-2-naphthol derivatives in high yields by one-pot, three-component reaction of β-naphthol, aryl aldehydes, and thiourea or N-phenylthiourea at 100?°C under solvent-free conditions. In addition to its simplicity, this method has the ability to prepare a wide variety of the desired products.