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Elsevier电子期刊(567)
在“
Elsevier电子期刊
”中,
命中:
567
条,耗时:小于0.01 秒
在所有数据库中总计命中:
567
条
1.
Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline
antiplasmodial
scaffold
作者:
Justine Desroches
a
;
1
;
Charline Kieffer
a
;
1
;
Nicolas Primas
a
;
Sé
;
bastien Hutter
b
;
Armand Gellis
a
;
Hussein El-Kashef
c
;
Pascal Rathelot
a
;
Pierre Verhaeghe
d
;
pierre.verhaeghe@univ-tlse3.fr
;
Nadine Azas
b
;
Patrice Vanelle
a
;
patrice.vanelle@univ-amu.fr
关键词:
Quinazoline
;
Quinoline
;
Quinoxaline
;
Thienopyrimidine
;
Trichloromethyl goup
;
Plasmodium falciparum
;
In vitro
antiplasmodial
activity
;
In vitro HepG2 cytotoxicity
;
Structure-activity relationships
刊名:European Journal of Medicinal Chemistry
出版年:2017
2.
Design, synthesis and evaluation of 4-aminoquinoline-purine hybrids as potential
antiplasmodial
agents
作者:
P. Linga Reddy
a
;
Shabana I. Khan
b
;
Prija Ponnan
a
;
Mohit Tripathi
a
;
Diwan S. Rawat
a
;
dsrawat@chemistry.du.ac.in
关键词:
Antimalarial hybrids
;
Aminoquinoline
;
Antiplasmodial
activity
;
Heme binding activity
;
Docking studies
刊名:European Journal of Medicinal Chemistry
出版年:2017
3.
Synthesis and biological characterisation of ester and amide derivatives of fusidic acid as
antiplasmodial
agents
作者:
Marlene Espinoza-Moraga
a
;
Kawaljit Singh
a
;
Mathew Njoroge
a
;
Gurminder Kaur
a
;
John Okombo
a
;
Carmen De Kock
c
;
Peter J. Smith
c
;
Sergio Wittlin
d
;
e
;
Kelly Chibale
a
;
b
;
f
;
Kelly.Chibale@uct.ac.za
关键词:
Fusidic acid
;
Malaria
;
Antiplasmodial
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
4.
Synthesis and evaluation of naphthyl bearing 1,2,3-triazole analogs as
antiplasmodial
agents, cytotoxicity and docking studies
作者:
Saikrishna Balabadra
a
;
MeenaKumari Kotni
a
;
Vijjulatha Manga
a
;
vijjulathamanga@gmail.com
;
Aparna Devi Allanki
b
;
Rajesh Prasad
b
;
Puran Singh Sijwali
b
关键词:
Naphthyl 1
2 ;
3-triazoles
;
Click chemistry
;
Antiplasmodial
activity
;
Cytotoxicity
;
Induced fit docking (IFD)
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
5.
Antiplasmodial
dimeric chalcone derivatives from the roots of Uvaria siamensis
作者:
Abdul-Wahab Salae
a
;
wahab_a@pkru.ac.th
;
Orapan Chairerk
a
;
Piyanut Sukkoet
a
;
Therdsak Chairat
a
;
Uma Prawat
a
;
umaprawat@pkru.ac.th
;
Pittaya Tuntiwachwuttikul
a
;
Piya Chalermglin
b
;
Somsak Ruchirawat
c
;
d
关键词:
Uvaria siamensis
;
Annonaceae
;
Dimeric chalcone
;
Antimycobacterial
;
Antiplasmodial
;
Cytotoxicity
刊名:Phytochemistry
出版年:2017
6.
Antiplasmodial
activity of Heinsia crinita (Rubiaceae) and identification of new iridoids
作者:
P. Tshisekedi Tshibangu
a
;
b
;
P. Mutwale Kapepula
a
;
b
;
M.J. Kabongo Kapinga
b
;
A. Tujibikila Mukuta
b
;
Dibungi T. Kalenda
b
;
Alembert T. Tchinda
c
;
Ange A. Mouithys-Mickalad
d
;
O. Jansen
a
;
E. Cieckiewicz
a
;
M. Tits
a
;
L. Angenot
a
;
M. Fré
;
dé
;
rich
a
;
M.frederich@ulg.ac.be
关键词:
Heinsia crinita
;
Lamalbide triacetate
;
Lamiridosin tri-acetate
;
Malaria
;
Plasmodium falciparum
刊名:Journal of Ethnopharmacology
出版年:2017
7.
4-Aminoquinoline-ferrocenyl-chalcone conjugates: Synthesis and anti-plasmodial evaluation
作者:
Amandeep Singh
a
;
Jiri Gut
b
;
Philip J. Rosenthal
b
;
Vipan Kumar
a
;
vipan_org@yahoo.com
关键词:
4-Amino-quinoline-ferrocenylchalcone
;
1
;
3-dipolar cycloaddition
;
Antiplasmodial
activities
;
Structure-activity relationship
刊名:European Journal of Medicinal Chemistry
出版年:2017
8.
New derivatives of 7-chloroquinolin-4-amine with antiprotozoal activity
作者:
Johanna Faist
a
;
johanna.faist@uni-graz.at
;
Clemens Hinteregger
a
;
Werner Seebacher
a
;
Robert Saf
b
;
Pascal Mä
;
ser
c
;
Marcel Kaiser
c
;
Robert Weis
a
关键词:
Amines
;
Antiplasmodial
activity
;
Heterocycles
;
NMR spectroscopy
;
Nucleophilic substitutions
;
Quinoline
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
9.
Dual
antiplasmodial
activity of vitamin D3 and its analog, 22-oxacalcitriol, by direct and indirect mechanisms
作者:
Kiichi Yamamoto
a
;
c
;
kyama-q3.3@mopera.net
;
Moritoshi Iwagami
b
;
Takenori Seki
a
;
Shigeyuki Kano
b
;
Nobuo Ota
a
;
Manabu Ato
c
关键词:
VD3
;
vitamin D3
;
(1α
;
25-dihydroxyvitamin D3)
;
VD
;
vitamin D
;
VDR
;
vitamin D receptor
;
KO
;
knock out
;
ZA
;
zoledronic acid
;
IFN-γ
;
interferon gamma
;
22-OCT
;
22-oxacalcitriol
;
PcAS
;
Plasmodium chabaudi AS
;
Pf
;
Plasmodium falciparum
;
PRBCs
;
parasitized red blood cells
刊名:Parasitology International
出版年:2017
10.
In vitro
antiplasmodial
and antioxidant activities of bisbenzylisoquinoline alkaloids from Alseodaphne corneri Kosterm
作者:
Azeana Zahari
1
;
Abdulwali Ablat
2
;
Yasodha Sivasothy
1
;
Jamaludin Mohamad
2
;
Muhammad I. Choudhary
3
;
Khalijah Awang
1
;
khalijah@um.edu.my" class="auth_mail" title="E-mail the corresponding author
关键词:
Bisbenzylisoquinoline
;
Laurotetanine
;
Norstephasubine
;
Antiplasmodial
;
Antioxidant
;
Oxidative stress
刊名:Asian Pacific Journal of Tropical Medicine
出版年:2016
1
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3
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7
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