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SpringerLink电子期刊(11)
Elsevier电子期刊(26)
ACS电子期刊(9)
在“
Elsevier电子期刊
”中,
命中:
26
条,耗时:0.0329844 秒
在所有数据库中总计命中:
46
条
1.
Design and synthesis of novel N-sulfonyl-2-indoles that behave as
5
-HT
6
receptor
ligands
with significant selectivity for D
3
over D
2
receptor
s
作者:
Oscar M. Saavedra
a
;
Delphine Karila
a
;
Dominique Brossard
a
;
Anne Rojas
b
;
Delphine Dupuis
c
;
Arnaud Gohier
d
;
Clotilde Mannoury la Cour
c
;
Mark J. Millan
c
;
;
Jean-Claude Ortuno
b
;
;
Stephen Hanessian
a
;
关键词:
Benzocyclobutane
;
Indole
;
CNS
receptor
s
;
Schizophrenia
;
Antipsychotic
刊名:Bioorganic & Medicinal Chemistry
出版年:2017
2.
Convergent
18
F-labeling and evaluation of N-benzyl-phenethylamines as
5
-HT
2A
receptor
PET
ligands
作者:
Ida Nymann Petersen
a
;
Jonas Villadsen
b
;
Hanne Demant Hansen
b
;
Anders A. Jensen
a
;
Szabolcs Lehel
c
;
Nic Gillings
c
;
Matthias M. Herth
a
;
c
;
Gitte M. Knudsen
b
;
Jesper L. Kristensen
a
;
jesper.kristensen@sund.ku.dk" class="auth_mail" title="E-mail the corresponding author
关键词:
18F-labeling
;
PET
;
Serotonin
;
5
-
HT2A
receptor
agonist
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
3.
5
-HT
2
receptor
affinity, docking studies and pharmacological evaluation of a series of 1,3-disubstituted thiourea derivatives
作者:
Anna Bielenica
a
;
abielenica@wum.edu.pl" class="auth_mail" title="E-mail the corresponding author
;
Ewa Kędzierska
b
;
Michał Koliński
c
;
Sebastian Kmiecik
d
;
Andrzej Koliński
d
;
Ferdinando Fiorino
e
;
Beatrice Severino
e
;
Elisa Magli
e
;
Angela Corvino
e
;
Ilaria Rossi
f
;
Paola Massarelli
f
;
Anna E. Kozioł
g
;
Aleksandra Sawczenko
g
;
Marta Struga
h
关键词:
5
-
HT2A
receptor
ligands
;
5
-HT2C
receptor
ligands
;
Docking studies
;
Thiourea
;
CNS activity
刊名:European Journal of Medicinal Chemistry
出版年:2016
4.
Dibenzo[b,f][1,4]oxazepines and dibenzo[b,e]oxepines: Influence of the chlorine substitution pattern on the pharmacology at the H
1
R, H
4
R,
5
-HT
2A
R and other selected GPCRs
作者:
Franziska Naporra
a
;
Susanne Gobleder
a
;
Hans-Joachim Wittmann
b
;
Julia Spindler
a
;
Michael Bodensteiner
c
;
Gü
;
nther Bernhardt
b
;
Harald Hü
;
bner
d
;
Peter Gmeiner
d
;
Sigurd Elz
a
;
Andrea Strasser
b
;
andrea.strasser@chemie.uni-regensburg.de" class="auth_mail" title="E-mail the corresponding author
关键词:
Histamine H1
receptor
;
Histamine H4
receptor
;
Dual/selective H1R/H4R
ligands
;
Dual hH1R/h
5
-
HT2A
R
ligands
;
Oxazepine derivatives
;
Oxepine derivatives
刊名:Pharmacological Research
出版年:2016
5.
New halogenated tris-(phenylalkyl)amines as h
5
-HT
2B
receptor
ligands
作者:
Nirav Kapadia
a
;
b
;
Shahrear Ahmed
a
;
Wayne W. Harding
a
;
b
;
关键词:
5
-
HT2A
;
5
-HT2B
;
CNS
;
Tris-(phenylalkyl)amine
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2016
6.
Synthesis and evaluation of
18
F-labeled
5
-HT
2A
receptor
agonists as PET
ligands
作者:
Matthias M. Herth
a
;
b
;
c
;
1
;
Ida Nymann Petersen
a
;
1
;
Hanne Demant Hansen
b
;
Martin Hansen
a
;
Anders Ettrup
b
;
Anders A. Jensen
a
;
Szabolcs Lehel
c
;
Agnete Dyssegaard
b
;
Nic Gillings
c
;
Gitte M. Knudsen
b
;
Jesper L. Kristensen
a
;
jesper.kristensen@sund.ku.dk" class="auth_mail" title="E-mail the corresponding author
关键词:
PET
;
Fluorine-18
;
5
-
HT2A
R
;
Agonist
;
Cimbi-36
刊名:Nuclear Medicine and Biology
出版年:2016
7.
Synthesis, in vitro and in vivo pharmacological evaluation of serotoninergic
ligands
containing an isonicotinic nucleus
作者:
Ferdinando Fiorino
a
;
fefiorin@unina.it" class="auth_mail" title="E-mail the corresponding author
;
Antonio Ciano
a
;
Elisa Magli
a
;
Beatrice Severino
a
;
Angela Corvino
a
;
Elisa Perissutti
a
;
Francesco Frecentese
a
;
Paola Di Vaio
a
;
Angelo A. Izzo
a
;
Raffaele Capasso
a
;
Paola Massarelli
b
;
Cristina Nencini
b
;
Ilaria Rossi
b
;
Ewa Kędzierska
c
;
Jolanta Orzelska-Gò
;
rka
c
;
Anna Bielenica
d
;
Vincenzo Santagada
a
;
Giuseppe Caliendo
a
关键词:
Isonicotinamide derivatives
;
5
-HT1A
;
5
-
HT2A
and
5
-HT2C
ligands
;
Binding assays
;
In vitro assay
;
Behavioural tests
刊名:European Journal of Medicinal Chemistry
出版年:2016
8.
1,4-Disubstituted aromatic piperazines with high
5
-HT
2A
/D
2
selectivity: Quantitative structure-selectivity investigations, docking, synthesis and biological evaluation
作者:
Dorothee Mö
;
ller
a
;
Ismail Salama
a
;
b
;
ismail_mohamed@pharm.suez.edu.eg" class="auth_mail" title="E-mail the corresponding author
;
Ralf C. Kling
a
;
Harald Hü
;
bner
a
;
Peter Gmeiner
a
;
peter.gmeiner@fau.de" class="auth_mail" title="E-mail the corresponding author
关键词:
3D-QSAR
;
D2 partial agonist
;
CoMFA
;
CoMSIA
;
GPCR
;
Subtype selectivity
;
5
-
HT2A
/D2 selectivity
;
Dopamine
receptor
;
Serotonin
receptor
;
Phenylpiperazine
;
1
;
4-DAP
刊名:Bioorganic & Medicinal Chemistry
出版年:201
5
9.
Support for
5
-HT2C
receptor
functional selectivity in?vivo utilizing structurally diverse, selective
5
-HT2C
receptor
ligands
and the 2,
5
-dimethoxy-4-iodoamphetamine elicited head-twitch response model
作者:
Clinton E. Canal
a
;
b
;
c.canal@neu.edu
;
Raymond G. Booth
a
;
b
;
Drake Morgan
c
关键词:
Head-twitch response
;
DOI
;
Hallucinogen
;
C
5
7Bl/6J
;
Mouse serotonin 2C
receptor
;
Mouse serotonin 2A
receptor
;
Functional selectivity
刊名:Neuropharmacology
出版年:2013
10.
Novel pyrimidoazepine analogs as serotonin
5
-HT
2A
and
5
-HT
2C
receptor
ligands
for the treatment of obesity
作者:
Ha Yun Yang
a
;
b
;
Jinsung Tae
b
;
Yong Wan Seo
a
;
Yoon Jung Kim
a
;
c
;
Hye Yeon Im
a
;
d
;
Gil Don Choi
e
;
Heeyeong Cho
e
;
Woo-Kyu Park
e
;
Oh Seung Kwon
a
;
Yong Seo Cho
a
;
Minkyung Ko
a
;
HyunSeo Jang
a
;
Jaeick Lee
f
;
Kihang Choi
c
;
Chan-Hwa Kim
d
;
Jiyoun Lee
g
;
jlee@sungshin.ac.kr
;
Ae Nim Pae
a
;
anpae@kist.re.kr
关键词:
5
-
HT2A
antagonist
;
5
-HT2C antagonist
;
Obesity
;
Pyrimidoazepine
;
Serotonin
receptor
ligands
刊名:European Journal of Medicinal Chemistry
出版年:2013
1
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