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在“Elsevier电子期刊”中，命中：397条，耗时：小于0.01 秒

在所有数据库中总计命中：545条

1.An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold

作者：Srinivasulu Cherukupalli ; Rajshekhar Karpoormath ; ^{karpoormath@ukzn.ac.za} ; Balakumar Chandrasekaran ; Girish. A. Hampannavar ; Neeta Thapliyal ; Venkata Narayana Palakollu

关键词：Pyrazolo[1 ; 5-a]pyrimidine ; Anti-cancer agents ; Anti-infectious agents ; CNS agents ; Anti-inflammatory agents ; Radiopharmaceuticals

刊名：European Journal of Medicinal Chemistry

出版年：2017

2.Design, synthesis and cytotoxicity studies of novel pyrazolo[1, 5-a]pyridine derivatives

作者：Chitrakar Ravi^a ; ¹ ; Arem Qayum^b ; ¹ ; Darapaneni Chandra Mohan^a ; Shashank K. Singh^b ; ^{sksingh@iiim.ac.in} ; Subbarayappa Adimurthy^a ; ^{adimurthy@csmcri.org}

关键词：Pyrazolo[1 ; 5&ndash ; a]pyridines ; Cytotoxicity ; MCF-7 cells ; Growth inhibition ; SRB assay

刊名：European Journal of Medicinal Chemistry

出版年：2017

3.Green synthesis of novel spiro[indoline-3,4′-pyrazolo[3,4-b]pyridine]-2,3′(7′H)- dione, spiro[indeno[1,2-b]pyrazolo[4,3-e]pyridine-4,3′-indoline]-2′,3-dione, and spiro[benzo [h]pyrazolo[3,4-b]quinoline-7,3′-indoline]-2′,8(5H)-dione derivatives in aqueous medium

作者：Zhansheng Wang ; Lingli Gao ; Zhongyun Xu ; Zhi Ling ; Yaqi Qin ; Liangce Rong ; ^{lcrong@jsnu.edu.cn} ; Shu-Jiang Tu

关键词：Pyrazolo[3 ; 4-b]pyridine ; Pyrazolo[4 ; 3-e]pyridine ; Pyrazolo[3 ; 4-b]quinoline ; Aqueous medium ; Green synthesis

刊名：Tetrahedron

出版年：2017

4.Synthesis and antitumor activity of some new pyrazolo[1,5-a]pyrimidines

作者：Ashraf S. Hassan^a ; ^{ashraf_salmoon@yahoo.com} ; Mohamed F. Mady^b ; ^c ; Hanem M. Awad^d ; Taghrid S. Hafez^a

关键词：5-Amino-1H-pyrazole ; Pyrazolo[1 ; 5-a]pyrimidine ; Schiff bases ; MTT assay ; Anticancer activity ; Structure activity relationship

刊名：Chinese Chemical Letters

出版年：2017

5.Explicit treatment of active-site waters enhances quantum mechanical/implicit solvent scoring: Inhibition of CDK2 by new pyrazolo[1,5-a]pyrimidines

作者：Michaela Hylsová ; ^a ; ¹ ; Benoit Carbain^a ; ^f ; ¹ ; Jindřich Fanfrlí ; k^b ; ¹ ; Lenka Musilová ; ^a ; Susanta Haldar^b ; ^c ; Cemal Kö ; prü ; lü ; oğlu^b ; ^c ; Haresh Ajani^b ; ^c ; Pathik S. Brahmkshatriya^b ; Radek Jorda^d ; Vladimí ; r Kry&scaron ; tof^d ; Pavel Hobza^b ; ^c ; Aude Echalier^e ; ² ; Kamil Paruch^a ; ^f ; ^{paruch@chemi.muni.cz} ; Martin Lep&scaron ; í ; k^b ; ^{lepsik@uochb.cas.cz}

关键词：Cyclin-dependent kinase 2 ; ATP-competitive type I inhibitors ; Pyrazolo[1 ; 5-a]pyrimidine ; Quantum mechanical scoring ; Protein-ligand binding ; Molecular dynamics ; Water thermodynamics ; X-ray crystal structure

刊名：European Journal of Medicinal Chemistry

出版年：2017

6.Evaluation of 7-arylaminopyrazolo[1,5-a]pyrimidines as anti-Plasmodium falciparum, antimalarial, and Pf-dihydroorotate dehydrogenase inhibitors

作者：Luí ; s Felipe S.P. Azeredo^a ; ^b ; Julia P. Coutinho^c ; ^d ; Valquiria A.P. Jabor^e ; Patricia R. Feliciano^e ; Maria Cristina Nonato^e ; Carlos R. Kaiser^b ; Carla Maria S. Menezes^a ; Amanda S.O. Hammes^f ; Ernesto Raul Caffarena^f ; Lucas V.B. Hoelz^a ; Nicolli B. de Souza^c ; Glaé ; cia A.N. Pereira^c ; Isabela P. Cerá ; volo^c ; Antoniana U. Krettli^c ; ^d ; Nubia Boechat^a ; ^b ; ^{boechat@far.fiocruz.br}

关键词：Malaria ; P. falciparum ; Pyrazolo[1 ; 5-a]pyrimidine ; Dihydroorotate dehydrogenase (DHODH) ; Molecular docking

刊名：European Journal of Medicinal Chemistry

出版年：2017

7.Pyrazolo[1,5-a]pyridine-3-carboxamide hybrids: Design, synthesis and evaluation of anti-tubercular activity

作者：Xiaoyun Lu^a ; ^b ; ¹ ; ^{luxy2016@jnu.edu.cn} ; Jian Tang^b ; ^c ; ¹ ; Shengyang Cui^b ; ^c ; Baojie Wan^d ; Scott G. Franzblauc^d ; Tianyu Zhang^b ; Xiantao Zhang^e ; Ke Ding^a ; ^b

关键词：Anti-tubercular ; Hybrid ; Mtb ; Pyrazolo[1 ; 5-a]pyridine-3-carboxamide

刊名：European Journal of Medicinal Chemistry

出版年：2017

8.Derivatives of the pyrazolo[1,5-a]pyrimidine acetamide DPA-713 as translocator protein (TSPO) ligands and pro-apoptotic agents in human glioblastoma

作者：Eryn L Werry^a ; ¹ ; Victoria A. King^b ; ¹ ; Melissa L Barron^a ; Samuel D. Banister^c ; Renee Sokias^c ; Michael Kassiou^c ; ^{michael.kassiou@sydney.edu.au}

关键词：BrdU ; 5-bromo-2&prime ; -deoxyuridine ; DMEM/F12 ; Dulbecco's modified eagle's medium ; Ham's nutrient mixture F-12 ; DMSO ; dimethyl sulfoxide ; EDTA ; ethylenediaminetetraacetic acid ; LLE ; lipophilic ligand efficiency ; MEM ; minimum essential medium ; PET ; positron emission tomography ; SPECT ; single-photon emission computed tomography ; TSPO ; translocator protein

刊名：European Journal of Pharmaceutical Sciences

出版年：2017

9.Novel pyrazolo[1,5-a]pyridines with improved aqueous solubility as p110α-selective PI3 kinase inhibitors

作者：Jackie D. Kendall^a ; ^b ; ^{j.kendall@auckland.ac.nz} ; Anna C. Giddens^a ; Kit Yee Tsang^a ; Elaine S. Marshall^a ; Claire L. Lill^c ; Woo-Jeong Lee^c ; Sharada Kolekar^c ; Mindy Chao^c ; Alisha Malik^c ; Shuqiao Yu^c ; Claire Chaussade^b ; ^c ; ^d ; Christina Buchanan^b ; ^c ; Stephen M.F. Jamieson^a ; ^b ; Gordon W. Rewcastle^a ; ^b ; Bruce C. Baguley^a ; ^b ; William A. Denny^a ; ^b ; Peter R. Shepherd^b ; ^c

关键词：NKJYYWGDGSKPEW-LPYMAVHISA-N ; AOXAAEQFLNMCLC-BUVRLJJBSA-N ; WBWLQGYBHWVMKE-DHRITJCHSA-N ; MXOGXVOOBVIVJW-YDZHTSKRSA-N ; AZJHDRSPNKBZGF-MFKUBSTISA-N ; QIGFDKVDGDNYSS-LGJNPRDNSA-N ; QPTBMDPOZNSWEZ-WSDLNYQXSA-N ; OCKIBXWFWFCVNS-YDZHTSKRSA-N ; UZWYFVJGBGJHHK-OEAKJJBVSA-N ; IHHGTHQQCPWJCF-BUVRLJJBSA-N ; LAWUZULWVPIZEA-PCLIKHOPSA-N ; KJKKEUXQKMRBSJ-YZSQISJMSA-N ; PJBLMNWKWHJQJT-PCLIKHOPSA-N ; FCUSNDJMENFTMM-YZSQISJMSA-N ; JXBONZLAZJXGLS-VULFUBBASA-N ; VZUIUZAIADXPHJ-VULFUBBASA-N ; VSPKBGAMPVYLDO-VULFUBBASA-N ; VWPPTJM

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

10.Unusual Lewis-acid catalyzed formal (3+3)-cycloaddition of azomethine imines and nitrones to N-vinylpyrroles

作者：Mariia M. Efremova^a ; Rafael R. Kostikov^a ; Alexander V. Stepakov^a ; Taras L. Panikorovsky^a ; Victoriya S. Shcherbakova^b ; Andrey V. Ivanov^b ; Alexander P. Molchanov^a ; ^{a.molchanov@spbu.ru}

关键词：Pyrroles ; (3+3)-cycloadditiones ; Nitrones ; Azomethine imines ; Catalysis

刊名：Tetrahedron

出版年：2017

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