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Elsevier电子期刊(16)
ACS电子期刊(15)
在“
ACS电子期刊
”中,
命中:
15
条,耗时:小于0.01 秒
在所有数据库中总计命中:
31
条
1.
The Discovery and Hit-to-Lead Optimization of Tricyclic Sulfonamides as Potent and Efficacious Potentiators of Glycine Receptors
作者:
Howard BregmanJeffrey R. Simard
;
Kristin L. Andrews
;
Shawn Ayube
;
Hao Chen
;
Hakan Gunaydin
;
Angel
Guzman
-
Perez
;
Jiali Hu
;
Liyue Huang
;
Xin Huang
;
Paul H. Krolikowski
;
Sonya G. Lehto
;
Richard T. Lewis
;
Klaus Michelsen
;
Pamela Pegman
;
Matthew H. Plant
;
Paul L. Shaffer
;
Yohannes Teffera
;
Shuyan Yi
;
Maosheng Zhang
;
Jacinthe Gingras
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2017
2.
Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1) Antagonists Demonstrating Potent in Vivo Activity
作者:
Laurie B. Schenkel
;
Philip R. Olivieri
;
Alessandro A. Boezio
;
Holly L. Deak
;
Renee Emkey
;
Russell F. Graceffa
;
Hakan Gunaydin
;
Angel
Guzman
-
Perez
;
Josie H. Lee
;
Yohannes Teffera
;
Weiya Wang
;
Beth D. Youngblood
;
Violeta L. Yu
;
Maosheng Zhang
;
Narender R. Gavva
;
Sonya G. Lehto
;
Stephanie Geuns-Meyer
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors
作者:
Erin F. DiMauro
;
Stephen Altmann
;
Loren M. Berry
;
Howard Bregman
;
Nagasree Chakka
;
Margaret Chu-Moyer
;
Elma Feric Bojic
;
Robert S. Foti
;
Robert Fremeau
;
Hua Gao
;
Hakan Gunaydin
;
Angel
Guzman
-
Perez
;
Brian E. Hall
;
Hongbing Huang
;
Michael Jarosh
;
Thomas Kornecook
;
Josie Lee
;
Joseph Ligutti
;
Dong Liu
;
Bryan D. Moyer
;
Daniel Ortuno
;
Paul E. Rose
;
Laurie B. Schenkel
;
Kristin Taborn
;
Jean Wang
;
Yan Wang
;
Violeta Yu
;
Matthew M. Weiss
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Structure-Based Design of 2-Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors
作者:
Hongbing Huang
;
Angel
Guzman
-
Perez
;
Lisa Acquaviva
;
Virginia Berry
;
Howard Bregman
;
Jennifer Dovey
;
Hakan Gunaydin
;
Xin Huang
;
Liyue Huang
;
Doug Saffran
;
Randy Serafino
;
Steve Schneider
;
Cindy Wilson
;
Erin F. DiMauro
刊名:ACS Medicinal Chemistry Letters
出版年:2013
5.
Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors
作者:
Howard Bregman
;
Nagasree Chakka
;
Angel
Guzman
-
Perez
;
Hakan Gunaydin
;
Yan Gu
;
Xin Huang
;
Virginia Berry
;
Jingzhou Liu
;
Yohannes Teffera
;
Liyue Huang
;
Bryan Egge
;
Erin L. Mullady
;
Steve Schneider
;
Paul S. Andrews
;
Ankita Mishra
;
John Newcomb
;
Randy Serafino
;
Craig A. Strathdee
;
Susan M. Turci
;
Cindy Wilson
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors
作者:
Zihao Hua
;
Howard Bregman
;
John L. Buchanan
;
Nagasree Chakka
;
Angel
Guzman
-
Perez
;
Hakan Gunaydin
;
Xin Huang
;
Yan Gu
;
Virginia Berry
;
Jingzhou Liu
;
Yohannes Teffera
;
Liyue Huang
;
Bryan Egge
;
Renee Emkey
;
Erin L. Mullady
;
Steve Schneider
;
Paul S. Andrews
;
Lisa Acquaviva
;
Jennifer Dovey
;
Ankita Mishra
;
John Newcomb
;
Douglas Saffran
;
Randy Serafino
;
Craig A. Strathdee
;
Susan M. Turci
;
Mary Stanton
;
Cindy Wilson
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2013
7.
Exploring Aromatic Chemical Space with NEAT: Novel and Electronically Equivalent Aromatic Template
作者:
Meihua Tu
;
Brajesh K. Rai
;
Alan M. Mathiowetz
;
Mary Didiuk
;
Jeffrey A. Pfefferkorn
;
Angel
Guzman
-
Perez
;
John Benbow
;
Cristiano R. W. Guimar茫es
;
Scot Mente
;
Matthew M. Hayward
;
Spiros Liras
刊名:Journal of Chemical Information and Modeling
出版年:2012
8.
Discovery of (S)-6-(3-Cyclopentyl-2-(4-(trifluoromethyl)-1H-imidazol-1-yl)propanamido)nicotinic Acid as a Hepatoselective Glucokinase Activator Clinical Candidate for Treating Type 2 Dia
作者:
Jeffrey A. Pfefferkorn
;
Angel
Guzman
-
Perez
;
John Litchfield
;
Robert Aiello
;
Judith L. Treadway
;
John Pettersen
;
Martha L. Minich
;
Kevin J. Filipski
;
Christopher S. Jones
;
Meihua Tu
;
Gary Aspnes
;
Hud Risley
;
Jianwei Bian
;
Benjamin D. Stevens
;
Patricia Bourassa
;
Theresa D鈥橝quila
;
Levenia Baker
;
Nicole Barucci
;
Alan S. Robertson
;
Francis Bourbonais
;
David R. Derksen
;
Margit MacDougall
;
Over Cabrera
;
Jing Chen
;
Amanda Lee Lapworth
;
James A. Landro
;
William J. Zavadoski
;
Karen Atkinson
;
Nahor Haddish-Berhane
;
Beijing Tan
;
Lili Yao
;
Rachel E. Kosa
;
Manthena V. Varma
;
Bo Feng
;
David B. Duignan
;
Ayman El-Kattan
;
Sharad Murdande
;
Shenping Liu
;
Mark Ammirati
;
John Knafels
;
Paul DaSilva-Jardine
;
Laurel Sweet
;
Spiros Liras
;
Timothy P. Rolph
刊名:Journal of Medicinal Chemistry
出版年:2012
9.
Maximizing Lipophilic Efficiency: The Use of Free-Wilson Analysis in the Design of Inhibitors of Acetyl-CoA Carboxylase
作者:
Kevin D. Freeman-Cook
;
Paul Amor
;
Scott Bader
;
Leanne M. Buzon
;
Steven B. Coffey
;
Jeffrey W. Corbett
;
Kenneth J. Dirico
;
Shawn D. Doran
;
Richard L. Elliott
;
William Esler
;
Angel
Guzman
-
Perez
;
Kevin E. Henegar
;
Janet A. Houser
;
Christopher S. Jones
;
Chris Limberakis
;
Katherine Loomis
;
Kirk McPherson
;
Sharad Murdande
;
Kendra L. Nelson
;
Dennis Phillion
;
Betsy S. Pierce
;
Wei Song
;
Eliot Sugarman
;
Susan Tapley
;
Meihua Tu
;
Zhengrong Zhao
刊名:Journal of Medicinal Chemistry
出版年:2012
10.
Functionalization of Aromatic Amino Acids via Direct C−H Activation: Generation of Versatile Building Blocks for Accessing Novel Peptide Space
作者:
Falco-Magnus Meyer
;
Spiros Liras
;
Angel
Guzman
-
Perez
;
Christian Perreault
;
Jianwei Bian
;
Keith James
刊名:Organic Letters
出版年:2010
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