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Wiley电子期刊(27)
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GSW全文库(12)
ACS电子期刊(160)
SpringerLink电子期刊(331)
NATURE电子期刊(103)
Elsevier电子期刊(1037)
在“
ACS电子期刊
”中,
命中:
160
条,耗时:0.0739644 秒
在所有数据库中总计命中:
1,694
条
1.
Discovery of LX2761,
a
Sodium-Dependent Glucose Cotr
a
nsporter 1 (SGLT1) Inhibitor Restricted to the Intestin
a
l Lumen, for the Tre
a
tment of Di
a
betes
作者:
Nicole C. GoodwinZhi-Ming Ding
;
Bryce
A
. H
a
rrison
;
Eric
D. Strobel
;
A
ngel
a
L. H
a
rris
;
Melind
a
Smith
;
A
ndre
a
Y. Thompson
;
Wendy Xiong
;
F
a
ik
a
Mseeh
;
Debr
a
J. Bruce
;
D
a
m
a
ris Di
a
z
;
Sum
a
Gopin
a
th
a
n
;
Ling Li
;
Emily O’Neill
;
M
a
ry Thiel
;
A
l
a
n G. E. Wilson
;
Kenneth G. C
a
rson
;
D
a
vid R. Powell
;
D
a
vid B. R
a
wlins
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2017
2.
Discovery
a
nd Optimiz
a
tion of Potent, Selective,
a
nd in Vivo Effic
a
cious 2-Aryl Benzimid
a
zole BCATm Inhibitors
作者:
Hongfeng Deng
;
Jingye Zhou
;
Flor
a
Sundersingh
;
Jeffrey
A
. Messer
;
Don
a
ld O. Somers
;
Myri
a
m Aj
a
k
a
ne
;
Christopher C.
A
rico-Muendel
;
A
rthur Belje
a
n
;
Svetl
a
n
a
L. Bely
a
nsk
a
y
a
;
Ry
a
n Bingh
a
m
;
Emily Bl
a
zensky
;
A
nne-Benedicte Boull
a
y
;
Eric
Boursier
;
Jing Ch
a
i
;
P
a
ul C
a
rter
;
Chun-W
a
Chung
;
A
l
a
in D
a
ug
a
n
;
Yun Ding
;
Kenny Herry
;
Cl
a
re Hobbs
;
Eric
Humphries
;
Christopher Kollm
a
nn
;
V
a
n Loc Nguyen
;
Edwige Nicodeme
;
S
a
r
a
h E.
Smith
;
Nerin
a
Dodic
;
Nicol
a
s Ancellin
刊名:
A
CS Medicin
a
l Chemistry Letters
出版年:2016
3.
Exploit
a
tion of
a
Novel Binding Pocket in Hum
a
n Lipoprotein-Associ
a
ted Phospholip
a
se A2 (Lp-PLA2) Discovered through X-r
a
y Fr
a
gment Screening
作者:
A
lison J.-A. Woolford
;
Joseph E. Pero
;
Sridh
a
r Ar
a
v
a
p
a
lli
;
V
a
lerio Berdini
;
Joseph E. Coyle
;
Philip J. D
a
y
;
A
ndrew M. Dodson
;
P
a
sc
a
l Grondin
;
Finn P. Holding
;
Lydi
a
Y. W. Lee
;
Peng Li
;
Eric
S. M
a
n
a
s
;
Joseph M
a
rino Jr.
;
A
gnes C. L. M
a
rtin
;
Brent W. McClel
a
nd
;
R
a
chel L. McMen
a
min
;
Christopher W. Murr
a
y
;
Christopher E. Neipp
;
Lee W. P
a
ge
;
Vipulkum
a
r K. P
a
tel
;
Florent Potv
a
in
;
Sh
a
rn
a
Rich
;
R
a
lph A. Rivero
;
Kirsten
Smith
;
Don
a
ld O. Somers
;
Lionel Trottet
;
R
a
ng
a
n
a
dh Vel
a
g
a
leti
;
Glyn Willi
a
ms
;
Ren Xie
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2016
4.
Discovery of (1S,2R,3S,4S,5R,6R)-2-
A
mino-3-[(3,4-difluorophenyl)sulf
a
nylmethyl]-4-hydroxy-bicyclo[3.1.0]hex
a
ne-2,6-dic
a
rboxylic Acid Hydrochloride (LY3020371·HCl): A Potent, Met
a
botropic Glut
a
m
a
te 2/3 Receptor Ant
a
gonist with Antidepress
a
nt-Like Activity
作者:
M
a
rk D. Ch
a
ppellRenhu
a
Li
;
Stephon C.
Smith
;
Bruce
A
. Dressm
a
n
;
Eric
G. Tromicz
a
k
;
A
llie E. Tripp
;
M
a
ri
a
-Jesus Bl
a
nco
;
T
a
ti
a
n
a
Vetm
a
n
;
Steven J. Quimby
;
J
a
mes M
a
tt
;
Thom
a
s C. Britton
;
A
d
a
m M. Fivush
;
Jeffrey M. Schkery
a
ntz
;
D
a
niel M
a
yhugh
;
Jon
A
.
Eric
kson
;
M
a
rk G. Bures
;
C
a
rlos J
a
r
a
millo
;
Mercedes C
a
rpintero
;
José Eugenio de Diego
;
M
a
rio B
a
rberis
;
Sus
a
n
a
G
a
rci
a
-Cerr
a
d
a
;
José F. Sori
a
no
;
Stephen
A
ntonys
a
my
;
Sh
a
ne Atwell
;
I
a
in M
a
cEw
a
n
;
Br
a
dley Condon
;
Christine Sougi
a
s
;
Jing W
a
ngAiping Zh
a
ng
;
Kris Conners
;
Chris Groshong
;
Stephen R. W
a
sserm
a
n
;
John W. Koss
;
Jeffrey M. Witkin
;
Xi
a
Li
;
C
a
rl Overshiner
;
Keith
A
. W
a
fford
;
Wesley Seidel
;
Xu-Sh
a
n W
a
ng
;
Beverly
A
. Heinz
;
Steven Sw
a
nson
;
John T. C
a
tlow
;
D
a
vid W. Bedwell
;
J
a
mes A. Monn
;
Ch
a
rles H. Mitch
;
P
a
ul L. Ornstein
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2016
5.
ZnCl2 C
a
pture Promotes Ethylene Polymeriz
a
tion by
a
S
a
licyl
a
ldimin
a
to Ni Complex Be
a
ring
a
Pendent 2,2′-Bipyridine Group
作者:
A
big
a
il J.
Smith
;
Eric
D. K
a
lkm
a
n
;
Z
a
ch
a
ry W. Gilbert
;
I
a
n A. Tonks
刊名:Org
a
nomet
a
llics
出版年:2016
6.
Structure-B
a
sed Design of
a
n Iminoheterocyclic β-Site Amyloid Precursor Protein Cle
a
ving Enzyme (BACE) Inhibitor th
a
t Lowers Centr
a
l Aβ in Nonhum
a
n Prim
a
tes
作者:
Mihirb
a
r
a
n M
a
nd
a
l
;
Yusheng Wu
;
Jeffrey Misi
a
szek
;
Guoqing Li
;
A
lexei Buevich
;
John P. C
a
ldwell
;
Xi
a
oxi
a
ng Liu
;
Robert D. M
a
zzol
a
;
Peter Orth
;
Corey Strickl
a
nd
;
Joh
a
nnes Voigt
;
Hongwu W
a
ng
;
Zh
a
oning Zhu
;
Xi
a
Chen
;
Mich
a
el Grzel
a
k
;
Lynn
A
. Hyde
;
Reshm
a
Kuvelk
a
r
;
Prescott T. Le
a
ch
;
Giuseppe Terr
a
cin
a
;
Lili Zh
a
ng
;
Qi Zh
a
ng
;
M
a
ri
a
S. Michener
;
Br
a
d
Smith
;
K
a
thleen Cox
;
Di
a
ne Grotz
;
Leon
a
rd F
a
vre
a
u
;
K
a
ushik Mitr
a
;
Irin
a
K
a
z
a
kevich
;
Bri
a
n A. McKittrick
;
Willi
a
m Greenlee
;
M
a
tthew E. Kennedy
;
Eric
M. P
a
rker
;
J
a
red N. Cumming
;
A
ndrew W. St
a
mford
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2016
7.
N-Methyl
a
tion
a
s
a
Str
a
tegy for Enh
a
ncing the Affinity
a
nd Selectivity of RNA-binding Peptides: Applic
a
tion to the HIV-1 Fr
a
meshift-Stimul
a
ting RNA
作者:
Thom
a
s A. Hilimire
;
Ry
a
n P. Bennett
;
Ry
a
n A. Stew
a
rt
;
P
a
blo G
a
rci
a
-Mir
a
nd
a
;
A
lex Blume
;
Jord
a
n Becker
;
N
a
th
a
n Sherer
;
Eric
D. Helms
;
S
a
muel E. Butcher
;
H
a
rold C.
Smith
;
Benj
a
min L. Miller
刊名:
A
CS Chemic
a
l Biology
出版年:2016
8.
Coordin
a
tion Geometry
a
nd Oxid
a
tion St
a
te Requirements of Corner-Sh
a
ring MnO6 Oct
a
hedr
a
for W
a
ter Oxid
a
tion C
a
t
a
lysis: An Investig
a
tion of M
a
ng
a
nite (γ-MnOOH)
作者:
P
a
ul F.
Smith
;
Benj
a
min J. Deibert
;
Shiv
a
m K
a
ushik
;
Gr
a
eme G
a
rdner
;
Shinj
a
e Hw
a
ng
;
H
a
o W
a
ng
;
J
a
f
a
r F. Al-Sh
a
r
a
b
;
Eric
G
a
rfunkel
;
L
a
ur
a
F
a
bris
;
Jing Li
;
G. Ch
a
rles Dismukes
刊名:
A
CS C
a
t
a
lysis
出版年:2016
9.
Discovery, S
A
R,
a
nd X-r
a
y Binding Mode Study of BCATm Inhibitors from
a
Novel DNA-Encoded Libr
a
ry
作者:
Hongfeng Deng
;
Jingye Zhou
;
Flor
a
S. Sundersingh
;
Jennifer Summerfield
;
Don Somers
;
Jeffrey
A
. Messer
;
A
lex
a
nder L. S
a
tz
;
Nicol
a
s Ancellin
;
Christopher C.
A
rico-Muendel
;
K
a
tie L. (S
a
rgent) Bed
a
rd
;
A
rthur Belje
a
n
;
Svetl
a
n
a
L. Bely
a
nsk
a
y
a
;
Ry
a
n Bingh
a
m
;
S
a
r
a
h E.
Smith
;
Eric
Boursier
;
P
a
ul C
a
rter
;
P
a
olo A. Centrell
a
;
M
a
tthew A. Cl
a
rk
;
Chun-w
a
Chung
;
Christopher P. D
a
vie
;
Jennifer L. Delorey
;
Yun Ding
;
G. Joseph Fr
a
nklin
;
L
a
Sh
a
dric C. Gr
a
dy
;
Kenny Herry
;
Cl
a
re Hobbs
;
Christopher S. Kollm
a
nn
;
B
a
rry A. Morg
a
n
;
L
a
ur
a
J. (Pothier) K
a
ush
a
nsky
;
Qu
a
n Zhou
刊名:
A
CS Medicin
a
l Chemistry Letters
出版年:2015
10.
Discovery of 5-
A
mino-N-(1H-pyr
a
zol-4-yl)pyr
a
zolo[1,5-
a
]pyrimidine-3-c
a
rbox
a
mide Inhibitors of IRAK4
作者:
Jongwon Lim
;
Mich
a
el D. Altm
a
n
;
J
a
mes B
a
ker
;
J
a
son D. Brub
a
ker
;
Hongmin Chen
;
Yiping Chen
;
Thierry Fischm
a
nn
;
Cr
a
ig Gibe
a
u
;
Mel
a
nie A. Kleinschek
;
Erica
Leccese
;
Ch
a
rles Lesburg
;
John K. F. M
a
cle
a
n
;
Lily Y. Moy
;
Erin F. Mulrooney
;
Jeremy Presl
a
nd
;
L
a
riss
a
R
a
khilin
a
;
Gr
a
h
a
m F.
Smith
;
Dietrich Steinhuebel
;
Ruojing Y
a
ng
刊名:
A
CS Medicin
a
l Chemistry Letters
出版年:2015
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