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Wiley电子期刊(2)
NATURE电子期刊(2)
ACS电子期刊(12)
SpringerLink电子期刊(9)
Elsevier电子期刊(18)
在“
ACS电子期刊
”中,
命中:
12
条,耗时:0.063968 秒
在所有数据库中总计命中:
43
条
1.
First-in-Cl
a
ss Chemic
a
l Probes
a
g
a
inst Poly(ADP-ribose) Glycohydrol
a
se (PARG) Inhibit DNA Rep
a
ir with Differenti
a
l Ph
a
rm
a
cology to Ol
a
p
a
rib
作者:
Dominic I. J
a
mes
;
K
a
te M. Smith
;
A
ll
a
n M. Jord
a
n
;
Emm
a
E. F
a
irwe
a
ther
;
Louise
A
. Griffiths
;
Nicol
a
S. H
a
milton
;
J
a
mes R. Hitchin
;
Colin P. Hutton
;
Stu
a
rt Jones
;
P
a
ul Kelly
;
A
lison E. McGon
a
gle
;
Helen Sm
a
ll
;
A
lex
a
ndr
a
I. J. Stowell
;
Julie
Tucker
;
I
a
n D. W
a
ddell
;
Bohd
a
n W
a
szkowycz
;
Don
a
ld J. Ogilvie
刊名:
A
CS Chemic
a
l Biology
出版年:2016
2.
Sm
a
ll Molecule Binding Sites on the R
a
s:SOS Complex C
a
n Be Exploited for Inhibition of R
a
s Activ
a
tion
作者:
Jon J. G. Winter
;
M
a
lcolm Anderson
;
Kevin Bl
a
des
;
Cl
a
ire Br
a
ssington
;
A
lex
a
nder L. Breeze
;
Christine Chrest
a
;
Kevin Embrey
;
G
a
ry F
a
irley
;
P
a
ul F
a
ulder
;
M. R
a
ymond V. Finl
a
y
;
J
a
son G. Kettle
;
Thorsten Now
a
k
;
Ross Overm
a
n
;
S. Joe P
a
tel
;
P
a
ul
a
Perkins
;
Lored
a
n
a
Sp
a
dol
a
;
Jon
a
th
a
n T
a
rt
;
Julie
A
.
Tucker
;
G
a
il Wrigley
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2015
3.
Structure Guided Le
a
d Gener
a
tion for M. tuberculosis Thymidyl
a
te Kin
a
se (Mtb TMK): Discovery of 3-Cy
a
nopyridone
a
nd 1,6-N
a
phthyridin-2-one
a
s Potent Inhibitors
作者:
M
a
ruti N
a
ik
;
A
n
a
ndkum
a
r R
a
ichurk
a
r
;
B
a
l
a
ch
a
ndr
a
S. B
a
ndodk
a
r
;
Begur V. V
a
run
;
Sh
a
ntik
a
Bh
a
t
;
R
a
jesh K
a
lkh
a
mbk
a
r
;
K
a
nn
a
n Murug
a
n
;
R
a
ni Menon
;
Jyothi Bh
a
t
;
Been
a
P
a
ul
;
H
a
rini Iyer
;
Syeed Hussein
;
Julie
A
.
Tucker
;
M
a
rtin Vogtherr
;
Kevin J. Embrey
;
Helen McMiken
;
Sw
a
ti Pr
a
s
a
d
;
A
dri
a
n Gill
;
Bheem
a
r
a
o G. Ug
a
rk
a
r
;
J
a
n
a
ni Venk
a
tr
a
m
a
n
;
Jon Re
a
d
;
M
a
nor
a
nj
a
n P
a
nd
a
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2015
4.
FGFR1 Kin
a
se Inhibitors: Close Regioisomers Adopt Divergent Binding Modes
a
nd Displ
a
y Distinct Biophysic
a
l Sign
a
tures
作者:
Tobi
a
s Klein
;
Julie
Tucker
;
Geoffrey
A
. Holdg
a
te
;
Rich
a
rd A. Norm
a
n
;
A
lex
a
nder L. Breeze
刊名:
A
CS Medicin
a
l Chemistry Letters
出版年:2014
5.
Homologous Critic
a
l Beh
a
vior in the Molecul
a
r Fr
a
meworks Zn(CN)2
a
nd Cd(imid
a
zol
a
te)2
作者:
Ines E. Collings
;
A
ndrew B. C
a
irns
;
A
mber L. Thompson
;
Juli
a
E. P
a
rker
;
Chiu C. T
a
ng
;
M
a
tthew G.
Tucker
;
J
a
dn
a
C
a
t
a
fest
a
;
Cl
a
ire Levelut
;
Julie
n H
a
ines
;
Vl
a
dimir Dmitriev
;
Philip P
a
ttison
;
A
ndrew L. Goodwin
刊名:The Journ
a
l of the Americ
a
n Chemic
a
l Society
出版年:2013
6.
Design
a
nd Synthesis of Novel L
a
ct
a
te Dehydrogen
a
se A Inhibitors by Fr
a
gment-B
a
sed Le
a
d Gener
a
tion
作者:
Rich
a
rd A. W
a
rd
;
Cl
a
ire Br
a
ssington
;
A
lex
a
nder L. Breeze
;
A
less
a
ndro C
a
puto
;
Sus
a
n Critchlow
;
G
a
reth D
a
vies
;
Louise Goodwin
;
Giles H
a
ss
a
ll
;
Ry
a
n Greenwood
;
Geoffrey
A
. Holdg
a
te
;
Mich
a
el Mrosek
;
Rich
a
rd A. Norm
a
n
;
Stu
a
rt Pe
a
rson
;
Jon
a
th
a
n T
a
rt
;
Julie
A
.
Tucker
;
M
a
rtin Vogtherr
;
D
a
vid Whitt
a
ker
;
Jon
a
th
a
n Wingfield
;
Jon Winter
;
Kevin Hudson
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2012
7.
Discovery of Novel Potent
a
nd Highly Selective Glycogen Synth
a
se Kin
a
se-3尾 (GSK3尾) Inhibitors for Alzheimer鈥檚 Dise
a
se: Design, Synthesis,
a
nd Ch
a
r
a
cteriz
a
tion of Pyr
a
zines
作者:
Stef
a
n Berg
;
M
a
rg
a
ret
a
Bergh
;
Sven Hellberg
;
K
a
th
a
rin
a
H枚gdin
;
Yvonne Lo-
A
lfredsson
;
Peter S枚derm
a
n
;
Stef
a
n von Berg
;
T
a
tj
a
n
a
Weigelt
;
M
a
ts Orm枚
;
Y
a
feng Xue
;
Julie
Tucker
;
J
a
n Neelissen
;
Ev
a
Jerning
;
Yvonne Nilsson
;
R
a
t
a
n Bh
a
t
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2012
8.
Thi
a
zolopyridine Ure
a
s
a
s Novel Antitubercul
a
r Agents Acting through Inhibition of DNA Gyr
a
se B
作者:
M
a
noj G. K
a
le
;
A
n
a
ndkum
a
r R
a
ichurk
a
r
;
Sh
a
hul H
a
meed P
;
D
a
vid W
a
terson
;
D
a
vid McKinney
;
M. R. M
a
njun
a
th
a
;
Ush
a
Kr
a
nthi
;
Krishn
a
Koushik
;
L
a
lit kum
a
r Jen
a
;
Vik
a
s Shinde
;
Suresh Rudr
a
p
a
tn
a
;
Shubh
a
d
a
B
a
rde
;
V
a
ish
a
li Humn
a
b
a
dk
a
r
;
Pr
a
sh
a
nti M
a
dh
a
v
a
peddi
;
H
a
lesh
a
B
a
s
a
v
a
r
a
j
a
pp
a
;
A
nirb
a
n Ghosh
;
VK R
a
my
a
;
Supreeth Gupth
a
;
Sreev
a
lli Sh
a
rm
a
;
Pr
a
k
a
sh V
a
ch
a
sp
a
ti
;
K.N. M
a
hesh Kum
a
r
;
J
a
y
a
shree Giridh
a
r
;
Jitend
a
r Reddy
;
Vijender P
a
ndug
a
;
S
a
mit G
a
nguly
;
Vij
a
yk
a
m
a
l Ahuj
a
;
Shesh
a
giri G
a
onk
a
r
;
C. N. N
a
veen Kum
a
r
;
Derek Ogg
;
Julie
A
.
Tucker
;
P.
A
nn Bori
a
ck-Sjodin
;
Sunit
a
M. de Sous
a
;
V
a
s
a
n K. S
a
mb
a
nd
a
murthy
;
S
a
ndeep R. Ghorp
a
de
刊名:Journ
a
l of Medicin
a
l Chemistry
出版年:2013
9.
A
minopyr
a
zin
a
mides: Novel
a
nd Specific GyrB Inhibitors th
a
t Kill Replic
a
ting
a
nd Nonreplic
a
ting Mycob
a
cterium tuberculosis
作者:
Pr
a
vin S. Shirude
;
Pr
a
sh
a
nti M
a
dh
a
v
a
peddi
;
Julie
A
.
Tucker
;
K
a
nn
a
n Murug
a
n
;
Vik
a
s P
a
til
;
H
a
lesh
a
B
a
s
a
v
a
r
a
j
a
pp
a
;
A
n
a
ndkum
a
r V. R
a
ichurk
a
r
;
V
a
ish
a
li Humn
a
b
a
dk
a
r
;
Syeed Hussein
;
Sreev
a
lli Sh
a
rm
a
;
V. K. R
a
my
a
;
Ch
a
nd
a
n B. N
a
r
a
y
a
n
;
T
a
njore S. B
a
lg
a
nesh
;
V
a
s
a
n K. S
a
mb
a
nd
a
murthy
刊名:
A
CS Chemic
a
l Biology
出版年:2013
10.
R
a
tion
a
l Design of M
a
teri
a
ls with Extreme Neg
a
tive Compressibility: Selective Soft-Mode Frustr
a
tion in KMn[Ag(CN)2]3
作者:
A
ndrew B. C
a
irns
;
A
mber L. Thompson
;
M
a
tthew G.
Tucker
;
Julie
n H
a
ines
;
A
ndrew L. Goodwin
刊名:The Journ
a
l of the Americ
a
n Chemic
a
l Society
出版年:2012
1
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