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Wiley电子期刊(1)
NATURE电子期刊(2)
ACS电子期刊(16)
SpringerLink电子期刊(12)
Elsevier电子期刊(3)
在“
ACS电子期刊
”中,
命中:
16
条,耗时:小于0.01 秒
在所有数据库中总计命中:
34
条
1.
The Discovery and Hit-to-Lead Optimization of Tricyclic Sulfonamides as Potent and Efficacious Potentiators of Glycine Receptors
作者:
Howard BregmanJeffrey R. Simard
;
Kristin L. Andrews
;
Shawn Ayube
;
Hao Chen
;
Hakan Gunaydin
;
Angel Guzman-Perez
;
Jiali Hu
;
Liyue Huang
;
Xin Huang
;
Paul H. Krolikowski
;
Sonya G. Lehto
;
Richard T. Lewis
;
Klaus
Michelsen
;
Pamela Pegman
;
Matthew H. Plant
;
Paul L. Shaffer
;
Yohannes Teffera
;
Shuyan Yi
;
Maosheng Zhang
;
Jacinthe Gingras
;
Erin F. DiMauro
刊名:Journal of Medicinal Chemistry
出版年:2017
2.
Discovery of Phosphodiesterase 10A (PDE10A) PET Tracer AMG 580 to Support Clinical Studies
作者:
Essa Hu
;
Ning Chen
;
Roxanne K. Kunz
;
Dah-Ren Hwang
;
Klaus
Michelsen
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna Lester-Zeiner
;
Randall Hungate
;
James Treanor
;
Hang Chen
;
Jennifer R. Allen
刊名:ACS Medicinal Chemistry Letters
出版年:2016
3.
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase–Glucokinase Regulatory Protein (GK–GKRP) Binding: Strategic Use of a N → S (nN → σ*S–X) Interaction fo
作者:
Lewis D. Pennington
;
Michael D. Bartberger
;
Michael D. Croghan
;
Kristin L. Andrews
;
Kate S. Ashton
;
Matthew P. Bourbeau
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Christopher Fotsch
;
Joan Helmering
;
Fang-Tsao Hong
;
Randall W. Hungate
;
Steven R. Jordan
;
Ke Kong
;
Longbin Liu
;
Klaus
Michelsen
;
Carolyn Moyer
;
Nobuko Nishimura
;
Mark H. Norman
;
Andreas Reichelt
;
Aaron C. Siegmund
;
Glenn Sivits
;
Seifu Tadesse
;
Christopher M. Tegley
;
Gwyneth Van
;
Kevin C. Yang
;
Guomin Yao
;
Jiandong Zhang
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean Jr.
刊名:Journal of Medicinal Chemistry
出版年:2015
4.
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 2. Leveraging Structure-Based Drug Design to Identify Analogues with Improved Pharmacokinetic Profiles
作者:
David J. St. Jean
;
Jr.
;
Kate S. Ashton
;
Michael D. Bartberger
;
Jie Chen
;
Samer Chmait
;
Rod Cupples
;
Elizabeth Galbreath
;
Joan Helmering
;
Fang-Tsao Hong
;
Steven R. Jordan
;
Longbin Liu
;
Roxanne K. Kunz
;
Klaus
Michelsen
;
Nobuko Nishimura
;
Lewis D. Pennington
;
Steve F. Poon
;
Darren Reid
;
Glenn Sivits
;
Markian M. Stec
;
Seifu Tadesse
;
Nuria Tamayo
;
Gwyneth Van
;
Kevin C. Yang
;
Jiandong Zhang
;
Mark H. Norman
;
Christopher Fotsch
;
David J. Lloyd
;
Clarence Hale
刊名:Journal of Medicinal Chemistry
出版年:2014
5.
Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 1. Discovery of a Novel Tool Compound for in Vivo Proof-of-Concept
作者:
Kate S. Ashton
;
Kristin L. Andrews
;
Marion C. Bryan
;
Jie Chen
;
Kui Chen
;
Michelle Chen
;
Samer Chmait
;
Michael Croghan
;
Rod Cupples
;
Christopher Fotsch
;
Joan Helmering
;
Steve R. Jordan
;
Robert J. M. Kurzeja
;
Klaus
Michelsen
;
Lewis D. Pennington
;
Steve F. Poon
;
Glenn Sivits
;
Gwyneth Van
;
Steve L. Vonderfecht
;
Robert C. Wahl
;
Jiandong Zhang
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
6.
Correction to Small Molecule Disruptors of the Glucokinase鈥揋lucokinase Regulatory Protein Interaction: 1. Discovery of a Novel Tool Compound for in Vivo Proof-of-Concept
作者:
Kate S. Ashton
;
Kristin L. Andrews
;
Marian C. Bryan
;
Jie Chen
;
Kui Chen
;
Michelle Chen
;
Samer Chmait
;
Michael Croghan
;
Rod Cupples
;
Christopher Fotsch
;
Joan Helmering
;
Steve R. Jordan
;
Robert J. M. Kurzeja
;
Klaus
Michelsen
;
Lewis D. Pennington
;
Steve F. Poon
;
Glenn Sivits
;
Gwyneth Van
;
Steve L. Vonderfecht
;
Robert C. Wahl
;
Jiandong Zhang
;
David J. Lloyd
;
Clarence Hale
;
David J. St. Jean
;
Jr.
刊名:Journal of Medicinal Chemistry
出版年:2014
7.
Fragment Based Drug Discovery: Practical Implementation Based on 19F NMR Spectroscopy
作者:
John B. Jordan
;
Leszek Poppe
;
Xiaoyang Xia
;
Alan C. Cheng
;
Yax Sun
;
Klaus
Michelsen
;
Heather Eastwood
;
Paul D. Schnier
;
Thomas Nixey
;
Wenge Zhong
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
Deuterium Kinetic Isotope Effects on the Dissociation of a Protein鈥揊atty Acid Complex in the Gas Phase
作者:
Lan Liu
;
Klaus
Michelsen
;
Elena N. Kitova
;
Paul D. Schnier
;
Alex Brown
;
John S. Klassen
刊名:The Journal of the American Chemical Society
出版年:2012
9.
Energetics of Lipid Binding in a Hydrophobic Protein Cavity
作者:
Lan Liu
;
Klaus
Michelsen
;
Elena N. Kitova
;
Paul D. Schnier
;
John S. Klassen
刊名:The Journal of the American Chemical Society
出版年:2012
10.
Ordering of the N-Terminus of Human MDM2 by Small Molecule Inhibitors
作者:
Klaus
Michelsen
;
John B. Jordan
;
Jeffrey Lewis
;
Alexander M. Long
;
Evelyn Yang
;
Yosup Rew
;
Jing Zhou
;
Peter Yakowec
;
Paul D. Schnier
;
Xin Huang
;
Leszek Poppe
刊名:The Journal of the American Chemical Society
出版年:2012
1
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