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Elsevier电子期刊(3)
ACS电子期刊(7)
在“
ACS电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
10
条
1.
Discovery of 1-{(3R,4R)-3-[({5-Chloro-2-[(1-methyl-1H-pyrazol-4-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Potent, WT Sparing, Irreversible Inhibitor of T790M-Containing EGFR Mutants
作者:
Hengmiao Cheng
;
Sajiv K. Nair
;
Brion W. Murray
;
Chau Almaden
;
Simon Bailey
;
Sangita Baxi
;
Doug Behenna
;
Sujin Cho-Schultz
;
Deepak Dalvie
;
Dac M. Dinh
;
Martin P. Edwards
;
Jun Li Feng
;
Rose Ann Ferre
;
Ketan S. Gajiwala
;
Michelle D. Hemkens
;
Amy Jackson-Fisher
;
Mehran Jalaie
;
Ted O. Johnson
;
Robert S. Kania
;
Susan Kephart
;
Jennifer Lafontaine
;
Beth Lunney
;
Kevin K.-C. Liu
;
Zhengyu Liu
;
Jean Matthews
;
Asako Nagata
;
Sherry Niessen
;
Martha A. Ornelas
;
Suvi T. M. Orr
;
Mason
Pairish
;
Simon Planken
;
Shijian Ren
;
Daniel Richter
;
Kevin Ryan
;
Neal Sach
;
Hong Shen
;
Tod Smeal
;
Jim Solowiej
;
Scott Sutton
;
Khanh Tran
;
Elaine Tseng
;
William Vernier
;
Marlena Walls
;
Shuiwang Wang
;
Scott L. Weinrich
;
Shuibo Xin
;
Haiwei Xu
;
Min-Jean Yin
;
Michael Zientek
;
Ru Zhou
;
John C. Kath
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery of a Novel Class of Exquisitely Selective Mesenchymal-Epithelial Transition Factor (c-MET) Protein Kinase Inhibitors and Identification of the Clinical Candidate 2-(4-(1-(Quinolin-6-ylmethyl
作者:
J. Jean Cui
;
Michele McTigue
;
Mitchell Nambu
;
Michelle Tran-Dub茅
;
Mason
Pairish
;
Hong Shen
;
Lei Jia
;
Hengmiao Cheng
;
Jacqui Hoffman
;
Phuong Le
;
Mehran Jalaie
;
Gilles H. Goetz
;
Kevin Ryan
;
Neil Grodsky
;
Ya-li Deng
;
Max Parker
;
Sergei Timofeevski
;
Brion W. Murray
;
Shinji Yamazaki
;
Shirley Aguirre
;
Qiuhua Li
;
Helen Zou
;
James Christensen
刊名:Journal of Medicinal Chemistry
出版年:2012
3.
Correction to Discovery of a Novel Class of Exquisitely Selective Mesenchymal-Epithelial Transition Factor (c-MET) Protein Kinase Inhibitors and Identification of the Clinical Candidate 2-(4-(1-(Quino
作者:
J. Jean Cui
;
Michele McTigue
;
Mitchell Nambu
;
Michelle Tran-Dub茅
;
Mason
Pairish
;
Hong Shen
;
Lei Jia
;
Hengmiao Cheng
;
Jacqui Hoffman
;
Phuong Le
;
Mehran Jalaie
;
Gilles H. Goetz
;
Marcel Koenig
;
Tomas Vojkovsky
;
Fang-Jie Zhang
;
Steven Do
;
Iriny Botrous
;
Kevin Ryan
;
Neil Grodsky
;
Ya-li Deng
;
Max Parker
;
Sergei Timofeevski
;
Brion W. Murray
;
Shinji Yamazaki
;
Shirley Aguirre
;
Qiuhua Li
;
Helen Zou
;
James Christensen
刊名:Journal of Medicinal Chemistry
出版年:2012
4.
Discovery of Aryloxy Tetramethylcyclobutanes as Novel Androgen Receptor Antagonists
作者:
Chuangxing Guo
;
Angelica Linton
;
Susan Kephart
;
Martha Ornelas
;
Mason
Pairish
;
Javier Gonzalez
;
Samantha Greasley
;
Asako Nagata
;
Benjamin J. Burke
;
Martin Edwards
;
Natilie Hosea
;
Ping Kang
;
Wenyue Hu
;
Jon Engebretsen
;
David Briere
;
Manli Shi
;
Hovik Gukasyan
;
Paul Richardson
;
Kevin Dack
;
Toby Underwood
;
Patrick Johnson
;
Andrew Morell
;
Robert Felstead
;
Hidetoshi Kuruma
;
Hiroaki Matsimoto
;
Amina Zoubeidi
;
Martin Gleave
;
Gerrit Los
;
Andrea N. Fanjul
刊名:Journal of Medicinal Chemistry
出版年:2011
5.
Structure Based Drug Design of Crizotinib (PF-02341066), a Potent and Selective Dual Inhibitor of Mesenchymal鈥揈pithelial Transition Factor (c-MET) Kinase and Anaplastic Lymphoma Kinase (ALK)
作者:
J. Jean Cui
;
Michelle Tran-Dube虂
;
Hong Shen
;
Mitchell Nambu
;
Pei-Pei Kung
;
Mason
Pairish
;
Lei Jia
;
Jerry Meng
;
Lee Funk
;
Iriny Botrous
;
Michele McTigue
;
Neil Grodsky
;
Kevin Ryan
;
Ellen Padrique
;
Gordon Alton
;
Sergei Timofeevski
;
Shinji Yamazaki
;
Qiuhua Li
;
Helen Zou
;
James Christensen
;
Barbara Mroczkowski
;
Steve Bender
;
Robert S. Kania
;
Martin P. Edwards
刊名:Journal of Medicinal Chemistry
出版年:2011
6.
Systematic Structure Modifications of Imidazo[1,2-a]pyrimidine to Reduce Metabolism Mediated by Aldehyde Oxidase (AO)
作者:
Angelica Linton
;
Ping Kang
;
Martha Ornelas
;
Susan Kephart
;
Qiyue Hu
;
Mason
Pairish
;
Ying Jiang
;
Chuangxing Guo
刊名:Journal of Medicinal Chemistry
出版年:2011
7.
An Extended -Strand Mimic for a Larger Artificial
作者:
James S. Nowick
;
Mason
Pairish
;
In Quen Lee
;
Darren L. Holmes
;
and Joseph W. Ziller
刊名:Journal of the American Chemical Society
出版年:1997
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