设为首页
收藏本站
网站地图
|
English
|
公务邮箱
About the library
Background
History
Leadership
Organization
Readers' Guide
Opening Hours
Collections
Help Via Email
Publications
Electronic Information Resources
常用资源
电子图书
期刊论文
学位会议
外文资源
特色专题
内部出版物
Elsevier电子期刊(4)
ACS电子期刊(10)
在“
ACS电子期刊
”中,
命中:
10
条,耗时:0.056972 秒
在所有数据库中总计命中:
14
条
1.
Discovery of 1-{(3R,4R)-3-[({5-Chloro-2-[(1-
m
e
t
hyl-1H-pyrazol-4-yl)a
m
ino]-7H-pyrrolo[2,3-d]pyri
m
idin-4-yl}oxy)
m
e
t
hyl]-4-
m
e
t
hoxypyrrolidin-1-yl}prop-2-en-1-one (PF-06459988), a Po
t
en
t
, WT Sparing, Irreversible Inhibi
t
or of T790M-Con
t
aining EGFR Mu
t
an
t
s
作者:
Heng
m
iao Cheng
;
Sajiv K. Nair
;
Brion W.
M
urray
;
Chau Al
m
aden
;
Si
m
on Bailey
;
Sangi
t
a Baxi
;
Doug Behenna
;
Sujin Cho-Schul
t
z
;
Deepak Dalvie
;
Dac
M
. Dinh
;
M
ar
t
in P. Edwards
;
Jun Li Feng
;
Rose Ann Ferre
;
Ke
t
an S. Gajiwala
;
M
ichelle D. He
m
kens
;
A
m
y Jackson-Fisher
;
M
ehran Jalaie
;
T
ed O. Johnson
;
Rober
t
S. Kania
;
Susan Kephar
t
;
Jennifer Lafon
t
aine
;
Be
t
h Lunney
;
Kevin K.-C. Liu
;
Zhengyu Liu
;
Jean
M
a
tt
hews
;
Asako Naga
t
a
;
Sherry Niessen
;
M
ar
t
ha A. Ornelas
;
Suvi
T
.
M
.
Orr
;
M
ason Pairish
;
Si
m
on Planken
;
Shijian Ren
;
Daniel Rich
t
er
;
Kevin Ryan
;
Neal Sach
;
Hong Shen
;
T
od S
m
eal
;
Ji
m
Solowiej
;
Sco
tt
Su
tt
on
;
Khanh
T
ran
;
Elaine
T
seng
;
Willia
m
Vernier
;
M
arlena Walls
;
Shuiwang Wang
;
Sco
tt
L. Weinrich
;
Shuibo Xin
;
Haiwei Xu
;
M
in-Jean Yin
;
M
ichael Zien
t
ek
;
Ru Zhou
;
John C. Ka
t
h
刊名:Journal of
M
edicinal Che
m
is
t
ry
出版年:2016
2.
Discovery of an in Vivo
T
ool
t
o Es
t
ablish Proof-of-Concep
t
for
M
AP4K4-Based An
t
idiabe
t
ic Trea
tm
en
t
作者:
M
ark A
mm
ira
t
i
;
Sco
tt
W. Bagley
;
Sa
m
i
t
K. Bha
tt
acharya
;
Leonard Buckbinder
;
An
t
hony A. Carlo
;
Rebecca Conrad
;
Chris
t
ian Cor
t
es
;
Rober
t
L. Dow
;
M
a
tt
hew S. Dowling
;
Ay
m
an El-Ka
tt
an
;
Kris
t
en Ford
;
Cris
t
iano R. W. Gui
m
ar茫es
;
David Hepwor
t
h
;
Wenhua Jiao
;
Jennifer LaPerle
;
Shenping Liu
;
Allyn Londregan
;
Paula
M
. Loria
;
Alan
M
. Ma
t
hiowe
t
z
;
M
ichael Munchhof
;
Suvi
T
.
M
.
Orr
;
Donna N. Pe
t
ersen
;
David A. Price
;
A
t
hanasia Skoura
;
Aaron C. S
m
i
t
h
;
Jian Wang
刊名:ACS
M
edicinal Che
m
is
t
ry Le
tt
ers
出版年:2015
3.
Discovery and Op
t
i
m
iza
t
ion of I
m
idazopyridine-Based Inhibi
t
ors of Diacylglycerol Acyl
t
ransferase 2 (DGAT2)
作者:
Ken
t
aro Fu
t
a
t
sugi
;
Daniel W. Kung
;
Suvi
T
.
M
.
Orr
;
Shawn Cabral
;
David Hepwor
t
h
;
Gary Aspnes
;
Sco
tt
Bader
;
Jianwei Bian
;
M
arkus Boeh
m
;
Philip A. Carpino
;
S
t
even B. Coffey
;
M
a
tt
hew S. Dowling
;
M
ichael Herr
;
Wenhua Jiao
;
Sophie Y. Lavergne
;
Qifang Li
;
Ronald W. Clark
;
Derek
M
. Erion
;
Kou Kou
;
Kyuha Lee
;
Brandon A. Pabs
t
;
Sylvie
M
. Perez
;
Julie Purkal
;
Csilla C. Jorgensen
;
T
heunis C. Goosen
;
Ja
m
es R. Gosse
t
;
M
ark Niosi
;
John C. Pe
tt
ersen
;
Jeffrey A. Pfefferkorn
;
Kay Ahn
;
Bryan Goodwin
刊名:Journal of
M
edicinal Che
m
is
t
ry
出版年:2015
4.
Evalua
t
ion and Syn
t
hesis of Polar Aryl- and He
t
eroaryl Spiroaze
t
idine-Piperidine Ace
t
a
m
ides as Ghrelin Inverse Agonis
t
s
作者:
Suvi
T
.
M
.
Orr
;
Ra
m
say Beveridge
;
Sa
m
i
t
K. Bha
tt
acharya
;
Ki
m
berly O. Ca
m
eron
;
S
t
even Coffey
;
Dilinie Fernando
;
David Hepwor
t
h
;
M
argare
t
V. Jackson
;
Vishal Kho
t
;
Rachel Kosa
;
Ki
m
berly Lapha
m
;
Paula
M
. Loria
;
Ki
m
F. McClure
;
Jigna Pa
t
el
;
Colin Rose
;
Ja
m
es Saenz
;
Ingrid A. S
t
ock
;
Gregory S
t
orer
;
M
aria von Volkenburg
;
Derek Vrieze
;
Guoqiang Wang
;
Jun Xiao
;
Yingxin Zhang
刊名:ACS
M
edicinal Che
m
is
t
ry Le
tt
ers
出版年:2015
5.
Discovery of 2-(6-(5-Chloro-2-
m
e
t
hoxyphenyl)-4-oxo-2-
t
hioxo-3,4-dihydropyri
m
idin-1(2H)-yl)ace
t
a
m
ide (PF-06282999): A Highly Selec
t
ive Mechanis
m
-Based Myeloperoxidase Inhibi
t
or for
t
he Trea
tm
en
t
of Car
作者:
Roger B. Ruggeri
;
Leonard Buckbinder
;
Sco
tt
W. Bagley
;
Philip A. Carpino
;
Edward L. Conn
;
M
a
tt
hew S. Dowling
;
Dilinie P. Fernando
;
Wenhua Jiao
;
Daniel W. Kung
;
Suvi
T
.
M
.
Orr
;
Ying
m
ei Qi
;
Benja
m
in N. Rocke
;
Aaron S
m
i
t
h
;
Joseph S. War
m
us
;
Yan Zhang
;
Daniel Bowles
;
Daniel W. Widlicka
;
Hea
t
her Eng
;
T
i
m
Ryder
;
Ra
m
an Shar
m
a
;
Angela Wolford
;
Carlin Okerberg
;
Karen Wal
t
ers
;
T
ris
t
an S.
M
aurer
;
Yanwei Zhang
;
Paul D. Bonin
;
Sa
m
an
t
ha N. Spa
t
h
;
Gang Xing
;
David Hepwor
t
h
;
Kay Ahn
;
A
m
i
t
S. Kalgu
t
kar
刊名:Journal of
M
edicinal Che
m
is
t
ry
出版年:2015
6.
Iden
t
ifica
t
ion of Te
t
rahydropyrido[4,3-d]pyri
m
idine A
m
ides as a New Class of Orally Bioavailable TGR5 Agonis
t
s
作者:
David W. Pio
t
rowski
;
Ken
t
aro Fu
t
a
t
sugi
;
Joseph S. War
m
us
;
Suvi
T
.
M
.
Orr
;
Kevin D. Free
m
an-Cook
;
Allyn
T
. Londregan
;
Liuqing Wei
;
Sandra
M
. Jennings
;
M
ichael Herr
;
S
t
even B. Coffey
;
Wenhua Jiao
;
Gregory S
t
orer
;
David Hepwor
t
h
;
Jian Wang
;
Sophie Y. Lavergne
;
Janice E. Chin
;
John R. Hadcock
;
M
ar
t
in B. Brenner
;
Angela C. Wolford
;
Ann
M
. Janssen
;
Nicole S. Roush
;
Joanne Bux
t
on
;
T
erri Hinchey
;
A
m
i
t
S. Kalgu
t
kar
;
Ra
m
an Shar
m
a
;
Declan A. Flynn
刊名:ACS
M
edicinal Che
m
is
t
ry Le
tt
ers
出版年:2013
7.
Discovery of PF-5190457, a Po
t
en
t
, Selec
t
ive, and Orally Bioavailable Ghrelin Recep
t
or Inverse Agonis
t
Clinical Candida
t
e
作者:
Sa
m
i
t
K. Bha
tt
acharya
;
Ki
m
Andrews
;
Ra
m
say Beveridge
;
Ki
m
berly O. Ca
m
eron
;
Chiliu Chen
;
M
a
tt
hew Dunn
;
Dilinie Fernando
;
Hua Gao
;
David Hepwor
t
h
;
V.
M
argare
t
Jackson
;
Vishal Kho
t
;
Ji
mm
y Kong
;
Rachel E. Kosa
;
Ki
m
berly Lapha
m
;
Paula
M
. Loria
;
Allyn
T
. Londregan
;
Ki
m
F. McClure
;
Suvi
T
.
M
.
Orr
;
Jigna Pa
t
el
;
Colin Rose
;
Ja
m
es Saenz
;
Ingrid A. S
t
ock
;
Gregory S
t
orer
;
M
aria VanVolkenburg
;
Derek Vrieze
;
Guoqiang Wang
;
Jun Xiao
;
Yingxin Zhang
刊名:ACS
M
edicinal Che
m
is
t
ry Le
tt
ers
出版年:2014
8.
M
echanis
m
-Based Inac
t
iva
t
ion (MBI) of Cy
t
ochro
m
e P450 Enzy
m
es: S
t
ruc
t
ure鈥揂c
t
ivi
t
y Rela
t
ionships and Discovery S
t
ra
t
egies To Mi
t
iga
t
e Drug鈥揇rug In
t
erac
t
ion Risks
作者:
Suvi
T
.
M
.
Orr
;
Sharon L. Ripp
;
T
. Eric Ballard
;
Jaclyn L. Henderson
;
Dennis O. Sco
tt
;
R. Sco
tt
Obach
;
Hao Sun
;
A
m
i
t
S. Kalgu
t
kar
刊名:Journal of
M
edicinal Che
m
is
t
ry
出版年:2012
9.
Novel Approach
t
o
t
he Lundurine Alkaloids: Syn
t
hesis of
t
he Te
t
racyclic Core
作者:
Suvi
T
.
M
.
Orr
;
Jianhua
T
ian
;
M
eike Nigge
m
ann
;
S
t
ephen F.
M
ar
t
in
刊名:Organic Le
tt
ers
出版年:2012
10.
Novel Approach
t
o
t
he Lundurine Alkaloids: Syn
t
hesis of
t
he Te
t
racyclic Core
作者:
Suvi
T
.
M
.
Orr
;
Jianhua
T
ian
;
M
eike Nigge
m
ann
;
S
t
ephen F.
M
ar
t
in
刊名:Organic Le
tt
ers
出版年:2011
1
按检索点细分(10)
题名(10)
按出版年细分(10)
2016年(1)
2015年(4)
2014年(1)
2013年(1)
2012年(2)
2011年(1)
NGLC 2004-2010.National Geological Library of China All Rights Reserved.
Add:29 Xueyuan Rd,Haidian District,Beijing,PRC. Mail Add: 8324 mailbox 100083
For exchange or info please contact us via
email
.