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Wiley电子期刊(2)
Elsevier电子期刊(16)
ACS电子期刊(11)
在“
ACS电子期刊
”中,
命中:
11
条,耗时:0.0289852 秒
在所有数据库中总计命中:
29
条
1.
GSK6853, a C
h
emical Probe for In
h
ibition of t
h
e BRPF1 Bromodomain
作者:
Paul Bamboroug
h
;
H
eat
h
er A. Barnett
;
Isabelle Bec
h
er
;
Mark J. Bird
;
C
h
un-wa C
h
ung
;
Peter D. Craggs
;
Emmanuel
H
.
Demont
;
H
awa Diallo
;
David J. Fallon
;
Laurie J. Gordon
;
Paola Grandi
;
Clare I.
H
obbs
;
Edward
H
ooper-Green
h
ill
;
Emma J. Jones
;
Robert P. Law
;
Armelle Le Gall
;
David Lugo
;
Anne-Marie Mic
h
on
;
Darren J. Mitc
h
ell
;
Rab K. Prinj
h
a
;
Robert J. S
h
eppard
;
Allan J. B. Watson
;
Robert J. Watson
刊名:ACS Medicinal C
h
emistry Letters
出版年:2016
2.
Discovery of Tetra
h
ydropyrazolopyridine as Sp
h
ingosine 1-P
h
osp
h
ate Receptor 3 (S1P3)-Sparing S1P1 Agonists Active at Low Oral Doses
作者:
Emmanuel
H
.
Demont
;
James M. Bailey
;
Rino A. Bit
;
Jack A. Brown
;
Colin A. Campbell
;
Nigel Deeks
;
Simon J. Dowell
;
Colin Eldred
;
Pam Gaskin
;
James R. J. Gray
;
Andrea
H
aynes
;
David J.
H
irst
;
Duncan S.
H
olmes
;
Umes
h
Kumar
;
Mary A. Morse
;
Greg J. Osborne
;
Jessica F. Renaux
;
Gail A. L. Seal
;
C
h
ris A. Smet
h
urst
;
Simon Taylor
;
Robert Watson
;
Robert Willis
;
Jason Wit
h
erington
刊名:Journal of Medicinal C
h
emistry
出版年:2016
3.
Glyp
h
osate Loss by Runoff and Its Relations
h
ip wit
h
P
h
osp
h
orus Fertilization
作者:
Mar铆a Carolina Sasal
;
Luisina
Demont
e
;
Andrea Cislag
h
i
;
Emmanuel
A. Gabioud
;
Jos茅 D. Oszust
;
Marcelo G. Wilson
;
Nicol谩s Mic
h
lig
;
H
oracio R. Beldom茅nico
;
Mar铆a Rosa Repetti
刊名:Journal of Agricultural and Food C
h
emistry
出版年:2015
4.
Fragment-Based Discovery of Low-Micromolar ATAD2 Bromodomain In
h
ibitors
作者:
Emmanuel
H
.
Demont
;
C
h
un-wa C
h
ung
;
Rebecca C. Furze
;
Paola Grandi
;
Anne-Marie Mic
h
on
;
C
h
ris Wellaway
;
Nat
h
alie Barrett
;
Angela M. Bridges
;
Peter D. Craggs
;
H
awa Diallo
;
David P. Dixon
;
Clement Douault
;
Amanda J. Emmons
;
Emma J. Jones
;
B
h
umika V. Karams
h
i
;
Kelly Locke
;
Darren J. Mitc
h
ell
;
Bernadette
H
. Mouzon
;
Rab K. Prinj
h
a
;
Andy D. Roberts
;
Robert J. S
h
eppard
;
Robert J. Watson
;
Paul Bamboroug
h
刊名:Journal of Medicinal C
h
emistry
出版年:2015
5.
Structure-Based Optimization of Nap
h
t
h
yridones into Potent ATAD2 Bromodomain In
h
ibitors
作者:
Paul Bamboroug
h
;
C
h
un-wa C
h
ung
;
Rebecca C. Furze
;
Paola Grandi
;
Anne-Marie Mic
h
on
;
Robert J. S
h
eppard
;
H
eat
h
er Barnett
;
H
awa Diallo
;
David P. Dixon
;
Clement Douault
;
Emma J. Jones
;
B
h
umika Karams
h
i
;
Darren J. Mitc
h
ell
;
Rab K. Prinj
h
a
;
C
h
ristina Rau
;
Robert J. Watson
;
T
h
ilo Werner
;
Emmanuel
H
.
Demont
刊名:Journal of Medicinal C
h
emistry
出版年:2015
6.
Navigating CYP1A Induction and Aryl
h
ydrocarbon Receptor Agonism in Drug Discovery. A Case History wit
h
S1P1 Agonists
作者:
Simon J. Taylor
;
Emmanuel
H
.
Demont
;
James Gray
;
Nigel Deeks
;
Aarti Patel
;
Dung Nguyen
;
Maxine Taylor
;
Steve
H
ood
;
Robert J. Watson
;
Rino A. Bit
;
Fiona McClure
;
H
olly As
h
all
;
Jason Wit
h
erington
刊名:Journal of Medicinal C
h
emistry
出版年:2015
7.
1,3-Dimet
h
yl Benzimidazolones Are Potent, Selective In
h
ibitors of t
h
e BRPF1 Bromodomain
作者:
Emmanuel
H
.
Demont
;
Paul Bamboroug
h
;
C
h
un-wa C
h
ung
;
Peter D. Craggs
;
David Fallon
;
Laurie J. Gordon
;
Paola Grandi
;
Clare I.
H
obbs
;
Jameed
H
ussain
;
Emma J. Jones
;
Armelle Le Gall
;
Anne-Marie Mic
h
on
;
Darren J. Mitc
h
ell
;
Rab K. Prinj
h
a
;
Andy D. Roberts
;
Robert J. S
h
eppard
;
Robert J. Watson
刊名:ACS Medicinal C
h
emistry Letters
出版年:2014
8.
T
h
e Discovery of I-BET726 (GSK1324726A), a Potent Tetra
h
ydroquinoline ApoA1 Up-Regulator and Selective BET Bromodomain In
h
ibitor
作者:
Romain Gosmini
;
Van Loc Nguyen
;
J茅r么me Toum
;
C
h
ristop
h
e Simon
;
Jean-Marie G. Brusq
;
Gael Krysa
;
Olivier Mirguet
;
Alizon M. Riou-Eymard
;
Eric V. Boursier
;
Lionel Trottet
;
Paul Bamboroug
h
;
H
ug
h
Clark
;
C
h
un-wa C
h
ung
;
Leanne Cutler
;
Emmanuel
H
.
Demont
;
Rejbinder Kaur
;
Antonia J. Lewis
;
Mark B. Sc
h
illing
;
Peter E. Soden
;
Simon Taylor
;
Ann L. Walker
;
Matt
h
ew D. Walker
;
Rab K. Prinj
h
a
;
Edwige Nicod猫me
刊名:Journal of Medicinal C
h
emistry
出版年:2014
9.
Discovery of a Brain-Penetrant S1P3-Sparing Direct Agonist of t
h
e S1P1 and S1P5 Receptors Efficacious at Low Oral Dose
作者:
Emmanuel
H
.
Demont
;
Sandra Arpino
;
Rino A. Bit
;
Colin A. Campbell
;
Nigel Deeks
;
Sapna Desai
;
Simon J. Dowell
;
Pam Gaskin
;
James R. J. Gray
;
Lee A.
H
arrison
;
Andrea
H
aynes
;
Tom D.
H
eig
h
tman
;
Duncan S.
H
olmes
;
P
h
ilip G. Hump
h
reys
;
Umes
h
Kumar
;
Mary A. Morse
;
Greg J. Osborne
;
Terry Panc
h
al
;
Karen L. P
h
ilpott
;
Simon Taylor
;
Robert Watson
;
Robert Willis
;
Jason Wit
h
erington
刊名:Journal of Medicinal C
h
emistry
出版年:2011
10.
Investigation of t
h
e Scope of a Co-Mediated O C Ring-Contraction
作者:
Simon J. Meek
;
Fabienne Pradaux
;
Emmanuel
H
.
Demont
;
Josep
h
P. A. Harrity
刊名:Journal of Organic C
h
emistry
出版年:2007
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