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Elsevier电子期刊(9)
ACS电子期刊(7)
在“
ACS电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
16
条
1.
Discovery of 6-Amino-2-{[(1S)-1-methylbutyl]oxy}-9-[5-(1-piperidinyl)pentyl]-7,9-dihydro-8H-purin-8-one (GSK2245035), a Highly Potent and Selective Intranasal Toll-Like Receptor 7 Agonist for the Treatment of Asthma
作者:
Keith
Biggadike
;
Mahbub Ahmed
;
Doug I. Ball
;
Diane M. Coe
;
Deidre A. Dalmas Wilk
;
Chris D. Edwards
;
Bob H. Gibbon
;
Charlotte J. Hardy
;
Stephen A. Hermitage
;
Joanne O. Hessey
;
Aimee E. Hillegas
;
Stephen C. Hughes
;
Linos Lazarides
;
Xiao Q. Lewell
;
Amanda Lucas
;
David N. Mallett
;
Mark A. Price
;
Fiona M. Priest
;
Diana J. Quint
;
Poonam Shah
;
Anesh Sitaram
;
Stephen A. Smith
;
Richard Stocker
;
Naimisha A. Trivedi
;
Daphne C. Tsitoura
;
Victoria Weller
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
Discovery of a Rapidly Metabolized, Long-Acting β2 Adrenergic Receptor Agonist with a Short Onset Time Incorporating a Sulfone Group Suitable for Once-Daily Dosing
作者:
Panayiotis A. Procopiou
;
Victoria J. Barrett
;
Keith
Biggadike
;
Peter R. Butchers
;
Andrew Craven
;
Alison J. Ford
;
Stephen B. Guntrip
;
Duncan S. Holmes
;
Sara C. Hughes
;
Anne E. Jones
;
Brian E. Looker
;
Peter J. Mutch
;
Mark Ruston
;
Deborah Needham
;
Claire E. Smith
刊名:Journal of Medicinal Chemistry
出版年:2014
3.
Correlation of Skin Blanching and Percutaneous Absorption for Glucocorticoid Receptor Agonists by Matrix-Assisted Laser Desorption Ionization Mass Spectrometry Imaging and Liquid Extraction Surface An
作者:
Peter Marshall
;
Valerie Toteu-Djomte
;
Philippe Bareille
;
Hayley Perry
;
Gillian Brown
;
Mark Baumert
;
Keith
Biggadike
刊名:Analytical Chemistry
出版年:2010
4.
Synthesis and Structure−Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Metabolic Inactivation: An Antedrug Approach
作者:
Panayiotis A. Procopiou
;
Victoria J. Barrett
;
Nicola J. Bevan
;
Keith
Biggadike
;
Philip C. Box
;
Peter R. Butchers
;
Diane M. Coe
;
Richard Conroy
;
Amanda Emmons
;
Alison J. Ford
;
Duncan S. Holmes
;
Helen H
刊名:Journal of Medicinal Chemistry
出版年:2010
5.
Synthesis and Structure−Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Arylsulfonamide Groups
作者:
Panayiotis A. Procopiou
;
Victoria J. Barrett
;
Nicola J. Bevan
;
Keith
Biggadike
;
Peter R. Butchers
;
Diane M. Coe
;
Richard Conroy
;
Dean D. Edney
;
Rita N. Field
;
Alison J. Ford
;
Stephen B. Guntrip
;
Brian
刊名:Journal of Medicinal Chemistry
出版年:2009
6.
X-ray Crystal Structure of the Novel Enhanced-Affinity Glucocorticoid Agonist Fluticasone Furoate in the Glucocorticoid Receptor−Ligand Binding Domain
作者:
Keith
Biggadike
;
Randy K. Bledsoe
;
Anne M. Hassell
;
Barrie E. Kirk
;
Iain M. McLay
;
Lisa M. Shewchuk
;
Eugene L. Stewart
刊名:Journal of Medicinal Chemistry
出版年:2008
7.
Nonsteroidal Glucocorticoid Agonists: Tetrahydronaphthalenes with Alternative Steroidal A-Ring Mimetics Possessing Dissociated (Transrepression/Transactivation) Efficacy Selectivity
作者:
Keith
Biggadike
;
Mohamed Boudjelal
;
Margaret Clackers
;
Diane M. Coe
;
Derek A. Demaine
;
George W. Hardy
;
Davina Humphreys
;
Graham G. A. Inglis
;
Michael J. Johnston
;
Haydn T. Jones
;
David House
;
Richard
刊名:Journal of Medicinal Chemistry
出版年:2007
1
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