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Springer电子图书(1)
SpringerLink电子期刊(14)
Elsevier电子期刊(30)
ACS电子期刊(17)
在“
ACS电子期刊
”中,
命中:
17
条,耗时:小于0.01 秒
在所有数据库中总计命中:
62
条
1.
Discovery of Aryl Sulfonamides as Isoform-Selective Inhibitors of NaV1.7 with Efficacy in Rodent Pain Models
作者:
Thilo Focken
;
Shifeng Liu
;
Navjot Chahal
;
Maxim Dauphinais
;
Michael E. Grimwood
;
Sultan Chowdhury
;
Ivan Hemeon
;
Paul Bichler
;
David Bogucki
;
Matthew Waldbrook
;
Girish Bankar
;
Luis E. Sojo
;
Clint Young
;
Sophia Lin
;
Noah Shuart
;
Rainbow Kwan
;
Jodie Pang
;
Jae H. Chang
;
Brian S. Safina
;
Daniel P. Sutherlin
;
J. P. Johnson Jr.
;
Christoph M. Dehnhardt
;
Tarek
S.
Mansour
;
Renata M. Oballa
;
Charles J. Cohen
;
C. Lee Robinette
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery of Isoquinolinone Indole Acetic Acids as Antagonists of Chemoattractant Receptor Homologous Molecule Expressed on Th2 Cells (CRTH2) for the Treatment of Allergic Inflammatory Diseases
作者:
Neelu Kaila
;
Bruce Follows
;
Louis Leung
;
Jennifer Thomason
;
Adrian Huang
;
Alessandro Moretto
;
Kristin Janz
;
Michael Lowe
;
Tarek
S.
Mansour
;
Cedric Hubeau
;
Karen Page
;
Paul Morgan
;
Susan Fish
;
Xin Xu
;
Cara Williams
;
Eddine Saiah
刊名:Journal of Medicinal Chemistry
出版年:2014
3.
Discovery of HSD-621 as a Potential Agent for the Treatment of Type 2 Diabetes
作者:
Zhao-Kui Wan
;
Eva Chenail
;
Huan-Qiu Li
;
Manus Ipek
;
Jason Xiang
;
Vipin Suri
;
Seung Hahm
;
Joel Bard
;
Kristine Svenson
;
Xin Xu
;
Xianbin Tian
;
Mengmeng Wang
;
Xiangping Li
;
Christian E. Johnson
;
Ariful Qadri
;
Darrell Panza
;
Mylene Perreault
;
Tarek
S.
Mansour
;
James F. Tobin
;
Eddine Saiah
刊名:ACS Medicinal Chemistry Letters
出版年:2013
4.
Diazine Indole Acetic Acids as Potent, Selective, and Orally Bioavailable Antagonists of Chemoattractant Receptor Homologous Molecule Expressed on Th2 Cells (CRTH2) for the Treatment of Allergic Infla
作者:
Neelu Kaila
;
Adrian Huang
;
Alessandro Moretto
;
Bruce Follows
;
Kristin Janz
;
Michael Lowe
;
Jennifer Thomason
;
Tarek
S.
Mansour
;
Cedric Hubeau
;
Karen Page
;
Paul Morgan
;
Susan Fish
;
Xin Xu
;
Cara Williams
;
Eddine Saiah
刊名:Journal of Medicinal Chemistry
出版年:2012
5.
Synthesis of Potent and Orally Efficacious 11尾-Hydroxysteroid Dehydrogenase Type 1 Inhibitor HSD-016
作者:
Zhao-Kui Wan
;
Eva Chenail
;
Huan-Qiu Li
;
Christopher Kendall
;
Youchu
;
Wang
;
Ste虂phane Gingras
;
Jason Xiang
;
Walter W. Massefski
;
Tarek
;
S.
Mansour
;
Eddine Saiah
刊名:Journal of Organic Chemistry
出版年:2011
6.
Hybrid Inhibitors of Phosphatidylinositol 3-Kinase (PI3K) and the Mammalian Target of Rapamycin (mTOR): Design, Synthesis, and Superior Antitumor Activity of Novel Wortmannin−Rapamycin Conjugate
作者:
Semiramis Ayral-Kaloustian
;
Jianxin Gu
;
Judy Lucas
;
Michael Cinque
;
Christine Gaydos
;
Arie Zask
;
Inder Chaudhary
;
Jianyao Wang
;
Li Di
;
Mairead Young
;
Mark Ruppen
;
Tarek
S.
Mansour
;
James J. Gibbons
;
Ke
刊名:Journal of Medicinal Chemistry
出版年:2010
7.
Stereoselective Synthesis of an Active Metabolite of the Potent PI3 Kinase Inhibitor PKI-179
作者:
Zecheng Chen
;
Aranapakam M. Venkatesan
;
Osvaldo Dos Santos
;
Efren Delos Santos
;
Christoph M. Dehnhardt
;
Semiramis Ayral-Kaloustian
;
Joseph Ashcroft
;
Leonard A. McDonald
;
Tarek
S.
Mansour
刊名:Journal of Organic Chemistry
出版年:2010
8.
Efficacious 11β-Hydroxysteroid Dehydrogenase Type I Inhibitors in the Diet-Induced Obesity Mouse Model
作者:
Zhao-Kui Wan
;
Eva Chenail
;
Jason Xiang
;
Huan-Qiu Li
;
Manus Ipek
;
Joel Bard
;
Kristine Svenson
;
Tarek
S.
Mansour
;
Xin Xu
;
Xianbin Tian
;
Vipin Suri
;
Seung Hahm
;
Yuzhe Xing
;
Christian E. Johnson
;
Xiangpin
刊名:Journal of Medicinal Chemistry
出版年:2009
9.
Oxidative Palladium Catalysis in SNAr Reactions Leading to Heteroaryl Ethers from Pyridotriazol-1-yloxy Heterocycles with Aryl Boronic Acids
作者:
Sumrit Wacharasindhu
;
Sujata Bardhan
;
Zhao-Kui Wan
;
Keiko Tabei
;
Tarek
S.
Mansour
*
刊名:Journal of the American Chemical Society
出版年:2009
10.
Heteroaryl Ethers by Oxidative Palladium Catalysis of Pyridotriazol-1-yloxy Pyrimidines with Arylboronic Acids
作者:
Sujata Bardhan
;
Sumrit Wacharasindhu
;
Zhao-Kui Wan
;
Tarek
S.
Mansour
刊名:Organic Letters
出版年:2009
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