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SpringerLink电子期刊(4)
NATURE电子期刊(1)
Elsevier电子期刊(11)
ACS电子期刊(9)
在“
ACS电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
25
条
1.
Synthetic Studies on Centromere-Associated Protein-E (CENP-E) Inhibitors: 2. Application of Electrostatic Potential Map (EPM) and Structure-Based Modeling to Imidazo[1,2-a]pyridine Derivatives as Anti
作者:
Takaharu Hirayama
;
Masanori Okaniwa
;
Hiroshi Banno
;
Hiroyuki Kakei
;
Akihiro Ohashi
;
Kenichi Iwai
;
Momoko Ohori
;
Kouji Mori
;
Mika Gotou
;
Tomohiro Kawamoto
;
Akihiro Yokota
;
Tomoyasu
Ishikawa
刊名:Journal of Medicinal Chemistry
出版年:2015
2.
Structure-Based Approach for the Discovery of Pyrrolo[3,2-d]pyrimidine-Based EGFR T790M/L858R Mutant Inhibitors
作者:
Satoshi Sogabe
;
Youichi Kawakita
;
Shigeru Igaki
;
Hidehisa Iwata
;
Hiroshi Miki
;
Douglas R. Cary
;
Terufumi Takagi
;
Shinji Takagi
;
Yoshikazu Ohta
;
Tomoyasu
Ishikawa
刊名:ACS Medicinal Chemistry Letters
出版年:2013
3.
Design and Synthesis of Potent Inhibitor of Apoptosis (IAP) Proteins Antagonists Bearing an Octahydropyrrolo[1,2-a]pyrazine Scaffold as a Novel Proline Mimetic
作者:
Kentaro Hashimoto
;
Bunnai Saito
;
Naoki Miyamoto
;
Yuya Oguro
;
Daisuke Tomita
;
Zenyu Shiokawa
;
Moriteru Asano
;
Hiroyuki Kakei
;
Naohiro Taya
;
Masanori Kawasaki
;
Hiroyuki Sumi
;
Masato Yabuki
;
Kenichi Iwai
;
Sei Yoshida
;
Mie Yoshimatsu
;
Kazunobu Aoyama
;
Yohei Kosugi
;
Takashi Kojima
;
Nao Morishita
;
Douglas R. Dougan
;
Gyorgy P. Snell
;
Shinichi Imamura
;
Tomoyasu
Ishikawa
刊名:Journal of Medicinal Chemistry
出版年:2013
4.
Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives
作者:
Masanori Okaniwa
;
Masaaki Hirose
;
Takeo Arita
;
Masato Yabuki
;
Akito Nakamura
;
Terufumi Takagi
;
Tomohiro Kawamoto
;
Noriko Uchiyama
;
Akihiko Sumita
;
Shunichirou Tsutsumi
;
Tsuneaki Tottori
;
Yoshitaka Inui
;
Bi-Ching Sang
;
Jason Yano
;
Kathleen Aertgeerts
;
Sei Yoshida
;
Tomoyasu
Ishikawa
刊名:Journal of Medicinal Chemistry
出版年:2013
5.
Discovery of Potent Mcl-1/Bcl-xL Dual Inhibitors by Using a Hybridization Strategy Based on Structural Analysis of Target Proteins
作者:
Yuta Tanaka
;
Katsuji Aikawa
;
Goushi Nishida
;
Misaki Homma
;
Satoshi Sogabe
;
Shigeru Igaki
;
Yumi Hayano
;
Tomoya Sameshima
;
Ikuo Miyahisa
;
Tomohiro Kawamoto
;
Michiko Tawada
;
Yumi Imai
;
Masakazu Inazuka
;
Nobuo Cho
;
Yasuhiro Imaeda
;
Tomoyasu
Ishikawa
刊名:Journal of Medicinal Chemistry
出版年:2013
6.
Design and Synthesis of Novel DFG-Out RAF/Vascular Endothelial Growth Factor Receptor 2 (VEGFR2) Inhibitors. 1. Exploration of [5,6]-Fused Bicyclic Scaffolds
作者:
Masanori Okaniwa
;
Masaaki Hirose
;
Takashi Imada
;
Tomohiro Ohashi
;
Youko Hayashi
;
Tohru Miyazaki
;
Takeo Arita
;
Masato Yabuki
;
Kazuyo Kakoi
;
Juran Kato
;
Terufumi Takagi
;
Tomohiro Kawamoto
;
Shuhei Yao
;
Akihiko Sumita
;
Shunichirou Tsutsumi
;
Tsuneaki Tottori
;
Hideyuki Oki
;
Bi-Ching Sang
;
Jason Yano
;
Kathleen Aertgeerts
;
Sei Yoshida
;
Tomoyasu
Ishikawa
刊名:Journal of Medicinal Chemistry
出版年:2012
7.
Design and Synthesis of Pyrrolo[3,2-d]pyrimidine Human Epidermal Growth Factor Receptor 2 (HER2)/Epidermal Growth Factor Receptor (EGFR) Dual Inhibitors: Exploration of Novel Back-Pocket Binder
作者:
Youichi Kawakita
;
Hiroshi Banno
;
Tomohiro Ohashi
;
Toshiya Tamura
;
Tadashi Yusa
;
Akiko Nakayama
;
Hiroshi Miki
;
Hidehisa Iwata
;
Hidenori Kamiguchi
;
Toshimasa Tanaka
;
Noriyuki Habuka
;
Satoshi Sogabe
;
Yoshikazu Ohta
;
Tomoyasu
Ishikawa
刊名:Journal of Medicinal Chemistry
出版年:2012
8.
Design and Synthesis of Novel Human Epidermal Growth Factor Receptor 2 (HER2)/Epidermal Growth Factor Receptor (EGFR) Dual Inhibitors Bearing a Pyrrolo[3,2-d]pyrimidine Scaffold
作者:
Tomoyasu
Ishikawa
;
Masaki Seto
;
Hiroshi Banno
;
Youichi Kawakita
;
Mami Oorui
;
Takahiko Taniguchi
;
Yoshikazu Ohta
;
Toshiya Tamura
;
Akiko Nakayama
;
Hiroshi Miki
;
Hidenori Kamiguchi
;
Toshimasa Tanaka
;
Noriyuki Habuka
;
Satoshi Sogabe
;
Jason Yano
;
Kathleen Aertgeerts
;
Keiji Kamiyama
刊名:Journal of Medicinal Chemistry
出版年:2011
9.
A Second-Generation Total Synthesis of (+)-Phorboxazole A
作者:
Amos B. Smith
;
III
;
Thomas M. Razler
;
Jeffrey P. Ciavarri
;
Tomoyasu
Hirose
;
Tomoyasu
Ishikawa
;
Regina M. Meis
刊名:Journal of Organic Chemistry
出版年:2008
1
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