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SpringerLink电子期刊(7)
Elsevier电子期刊(14)
ACS电子期刊(7)
在“
ACS电子期刊
”中,
命中:
7
条,耗时:小于0.01 秒
在所有数据库中总计命中:
28
条
1.
Rational Design of a Boron-Modified Triphenylethylene (GLL398) as an Oral Selective Estrogen Receptor Downregulator
作者:
Jiawang Liu
;
Shilong Zheng
;
Shanchun
Guo
;
Changde
Zhang
;
Qiu Zhong
;
Qiang
Zhang
;
Peng Ma
;
Elena V. Skripnikova
;
Melyssa R. Bratton
;
Thomas E. Wiese
;
Guangdi Wang
刊名:ACS Medicinal Chemistry Letters
出版年:2017
2.
Discovery of 4-Methyl-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((1-nicotinoylpiperidin-4-yl)oxy)benzamide (CHMFL-ABL/KIT-155) as a Novel Highly Potent Type II ABL/KIT Dual Kinase Inhibitor with a Distinct Hinge Binding
作者:
Qiang Wang
;
Feiyang Liu
;
Beilei Wang
;
Fengming Zou
;
Ziping Qi
;
Cheng Chen
;
Kailin Yu
;
Chen Hu
;
Shuang Qi
;
Wenchao Wang
;
Zhenquan Hu
;
Juan Liu
;
Wei Wang
;
Li Wang
;
Qianmao Liang
;
Shanchun
Zhang
;
Tao Ren
;
Qingsong Liu
;
Jing Liu
刊名:Journal of Medicinal Chemistry
出版年:2017
3.
Discovery of N-(3-((1-Isonicotinoylpiperidin-4-yl)oxy)-4-methylphenyl)-3-(trifluoromethyl)benzamide (CHMFL-KIT-110) as a Selective, Potent, and Orally Available Type II c-KIT Kinase Inhibitor for Gastrointestinal Stromal Tumors (GISTs)
作者:
Qiang Wang
;
Feiyang Liu
;
Beilei Wang
;
Fengming Zou
;
Cheng Chen
;
Xiaochuan Liu
;
Aoli Wang
;
Shuang Qi
;
Wenchao Wang
;
Ziping Qi
;
Zheng Zhao
;
Zhenquan Hu
;
Wei Wang
;
Li Wang
;
Shanchun
Zhang
;
Yuexiang Wang
;
Jing Liu
;
Qingsong Liu
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Discovery of N-((1-(4-(3-(3-((6,7-Dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I “Gatekeeper” Mutant of cKIT Kinase
作者:
Binhua Li
;
Aoli Wang
;
Juan Liu
;
Ziping Qi
;
Xiaochuan Liu
;
Kailin Yu
;
Hong Wu
;
Cheng Chen
;
Chen Hu
;
Wenchao Wang
;
Jiaxin Wu
;
Zhenquan Hu
;
Ling Ye
;
Fengming Zou
;
Feiyang Liu
;
Beilei Wang
;
Li Wang
;
Tao Ren
;
Shaojuan
Zhang
;
Mingfeng Bai
;
Shanchun
Zhang
;
Jing Liu
;
Qingsong Liu
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Fulvestrant-3 Boronic Acid (ZB716): An Orally Bioavailable Selective Estrogen Receptor Downregulator (SERD)
作者:
Jiawang Liu
;
Shilong Zheng
;
Victoria L. Akerstrom
;
Chester Yuan
;
Youning Ma
;
Qiu Zhong
;
Changde
Zhang
;
Qiang
Zhang
;
Shanchun
Guo
;
Peng Ma
;
Elena V. Skripnikova
;
Melyssa R. Bratton
;
Antonio Pannuti
;
Lucio Miele
;
Thomas E. Wiese
;
Guangdi Wang
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Discovery of 2-((3-Amino-4-methylphenyl)amino)-N-(2-methyl-5-(3-(trifluoromethyl)benzamido)phenyl)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-ABL-053) as a Potent, Selective, and Orally Available BCR-ABL/SRC/p38 Kinase Inhibitor for Chronic Myeloid Le
作者:
Xiaofei Liang
;
Xiaochuan Liu
;
Beilei Wang
;
Fengming Zou
;
Aoli Wang
;
Shuang Qi
;
Cheng Chen
;
Zheng Zhao
;
Wenchao Wang
;
Ziping Qi
;
Fengchao Lv
;
Zhenquan Hu
;
Li Wang
;
Shanchun
Zhang
;
Qingsong Liu
;
Jing Liu
刊名:Journal of Medicinal Chemistry
出版年:2016
7.
Discovery of (R)-1-(3-(4-Amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)-2-(dimethylamino)ethanone (CHMFL-FLT3-122) as a Potent and Orally Available FLT3 Kinase Inhibitor fo
作者:
Xixiang Li
;
Aoli Wang
;
Kailin Yu
;
Ziping Qi
;
Cheng Chen
;
Wenchao Wang
;
Chen Hu
;
Hong Wu
;
Jiaxin Wu
;
Zheng Zhao
;
Juan Liu
;
Fengming Zou
;
Li Wang
;
Beilei Wang
;
Wei Wang
;
Shanchun
Zhang
;
Jing Liu
;
Qingsong Liu
刊名:Journal of Medicinal Chemistry
出版年:2015
1
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