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SpringerLink电子期刊(1)
ACS电子期刊(6)
在“
ACS电子期刊
”中,
命中:
6
条,耗时:小于0.01 秒
在所有数据库中总计命中:
7
条
1.
Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials
作者:
T. G. Murali Dhar
;
Hai-Yun Xiao
;
Jenny Xie
;
Lois D. Lehman-McKeeman
;
Dauh-Rurng Wu
;
Marta Dabros
;
Xiaoxia Yang
;
Tracy L. Taylor
;
Xia D. Zhou
;
Elizabeth M. Heimrich
;
Rochelle Thomas
;
Kim W. McIntyre
;
Bethanne Warrack
;
Hong Shi
;
Paul C. Levesque
;
Jia L. Zhu
;
James Hennan
;
Praveen Balimane
;
Zheng Yang
;
Anthony M. Marino
;
Georgia Cornelius
;
Celia
J. D’Arienzo
;
Arvind Mathur
;
Ding Ren Shen
;
Mary Ellen Cvijic
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery and Structure–Activity Relationship (SAR) of a Series of Ethanolamine-Based Direct-Acting Agonists of Sphingosine-1-phosphate (S1P1)
作者:
John L. Gilmore
;
James E. Sheppeck II
;
Scott H. Watterson
;
Lauren Haque
;
Parag Mukhopadhyay
;
Andrew J. Tebben
;
Michael A. Galella
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Virna Borowski
;
Kathleen Gillooly
;
Tracy Taylor
;
Kim W. McIntyre
;
Bethanne Warrack
;
Paul C. Levesque
;
Julia P. Li
;
Georgia Cornelius
;
Celia
D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Luisa Salter-Cid
;
Joel C. Barrish
;
William J. Pitts
;
Percy H. Carter
;
Jenny Xie
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Potent and Selective Agonists of Sphingosine 1-Phosphate 1 (S1P1): Discovery and SAR of a Novel Isoxazole Based Series
作者:
Scott H. Watterson
;
Junqing Guo
;
Steve H. Spergel
;
Charles M. Langevine
;
Robert V. Moquin
;
Ding Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Dana Banas
;
Richard Liu
;
Suzanne J. Suchard
;
Kathleen Gillooly
;
Tracy Taylor
;
Sandra Rex-Rabe
;
David J. Shuster
;
Kim W. McIntyre
;
Georgia Cornelius
;
Celia
D’Arienzo
;
Anthony Marino
;
Praveen Balimane
;
Bethanne Warrack
;
Luisa Salter-Cid
;
Murray McKinnon
;
Joel C. Barrish
;
Percy H. Carter
;
William J. Pitts
;
Jenny Xie
;
Alaric J. Dyckman
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton’s Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked
作者:
Scott H. Watterson
;
George V. De Lucca
;
Qing Shi
;
Charles M. Langevine
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Hua Gong
;
Jun Dai
;
Shiuhang Yip
;
Peng Li
;
Dawn Sun
;
Dauh-Rurng Wu
;
Chunlei Wang
;
Yingru Zhang
;
Sarah C. Traeger
;
Mark A. Pattoli
;
Stacey Skala
;
Lihong Cheng
;
Mary T. Obermeier
;
Rodney Vickery
;
Lorell N. Discenza
;
Celia
J. D’Arienzo
;
Yifan Zhang
;
Elizabeth Heimrich
;
Kathleen M. Gillooly
;
Tracy L. Taylor
;
Claudine Pulicicchio
;
Kim W. McIntyre
;
Michael A. Galella
;
Andy J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing Chang
;
Richard Rampulla
;
Arvind Mathur
;
Luisa Salter-Cid
;
Joel C. Barrish
;
Percy H. Carter
;
Aberra Fura
;
James R. Burke
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Small Molecule Reversible Inhibitors of Bruton’s Tyrosine Kinase (BTK): Structure–Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177)
作者:
George V. De Lucca
;
Qing Shi
;
Qingjie Liu
;
Douglas G. Batt
;
Myra Beaudoin Bertrand
;
Rick Rampulla
;
Arvind Mathur
;
Lorell Discenza
;
Celia
D’Arienzo
;
Jun Dai
;
Mary Obermeier
;
Rodney Vickery
;
Yingru Zhang
;
Zheng Yang
;
Punit Marathe
;
Andrew J. Tebben
;
Jodi K. Muckelbauer
;
ChiehYing J. Chang
;
Huiping Zhang
;
Kathleen Gillooly
;
Tracy Taylor
;
Mark A. Pattoli
;
Stacey Skala
;
Daniel W. Kukral
;
Kim W. McIntyre
;
Luisa Salter-Cid
;
Aberra Fura
;
James R. Burke
;
Joel C. Barrish
;
Percy H. Carter
;
Joseph A. Tino
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1P1) Employing Ligand-Based Drug Design
作者:
Hai-Yun Xiao
;
Scott H. Watterson
;
Charles M. Langevine
;
Anurag S. Srivastava
;
Soo S. Ko
;
Yanlei Zhang
;
Robert J. Cherney
;
Wei-Wei Guo
;
John L. Gilmore
;
James E. Sheppeck II
;
Dauh-Rurng Wu
;
Peng Li
;
Duraisamy Ramasamy
;
Piramanayagam Arunachalam
;
Arvind Mathur
;
Tracy L. Taylor
;
David J. Shuster
;
Kim W. McIntyre
;
Ding-Ren Shen
;
Melissa Yarde
;
Mary Ellen Cvijic
;
Anthony M. Marino
;
Praveen V. Balimane
;
Zheng Yang
;
Dana M. Banas
;
Georgia Cornelius
;
Celia
J. D’Arienzo
;
Bethanne M. Warrack
;
Lois Lehman-McKeeman
;
Luisa M. Salter-Cid
;
Jenny Xie
;
Joel C. Barrish
;
Percy H. Carter
;
Alaric J. Dyckman
;
T. G. Murali Dhar
刊名:Journal of Medicinal Chemistry
出版年:2016
1
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