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SpringerLink电子期刊(1)
Elsevier电子期刊(4)
ACS电子期刊(6)
在“
ACS电子期刊
”中,
命中:
6
条,耗时:0.0189944 秒
在所有数据库中总计命中:
11
条
1.
Structure鈥揂ctivity Relationships, Pharmacokinetics, and in Vivo Activity o
f
CYP11B2 and CYP11B1 Inhibitors
作者:
Julien P. N. Papillon
;
Christopher M. Adams
;
Qi-Ying Hu
;
Changgang Lou
;
Alok K. Singh
;
Chun Zhang
;
Jose Carvalho
;
Srinivan Rajan
;
Adam Amaral
;
Michael E. Beil
;
F
umin Fu
;
Eric Gangl
;
Chii-Whei Hu
;
Arco Y. Jeng
;
Daniel LaSala
;
Guiqing Liang
;
Michael Logman
;
Wieslawa M. Maniara
;
Dean
F
.
Rigel
;
Sherri A. Smith
;
Gary M. Ksander
刊名:Journal o
f
Medicinal Chemistry
出版年:2015
2.
Discovery o
f
N-[5-(6-Chloro-3-cyano-1-methyl-1H-indol-2-yl)-pyridin-3-ylmethyl]-ethanesul
f
onamide, a Cortisol-Sparing CYP11B2 Inhibitor that Lowers Aldosterone in Human Subjects
作者:
Julien P. N. Papillon
;
Changgang Lou
;
Alok K. Singh
;
Christopher M. Adams
;
Gary M. Ksander
;
Michael E. Beil
;
Wei Chen
;
Jenni
f
er Leung-Chu
;
F
umin Fu
;
Lu Gan
;
Chii-Whei Hu
;
Arco Y. Jeng
;
Daniel LaSala
;
Guiqing Liang
;
Dean
F
.
Rigel
;
Kerry S. Russell
;
John A. Vest
;
Catherine Watson
刊名:Journal o
f
Medicinal Chemistry
出版年:2015
3.
Structure-Based Design o
f
Substituted Piperidines as a New Class o
f
Highly E
ff
icacious Oral Direct Renin Inhibitors
作者:
Takeru Ehara
;
Osamu Irie
;
Takatoshi Kosaka
;
Takanori Kanazawa
;
Werner Breitenstein
;
Philipp Grosche
;
Nils Ostermann
;
Masaki Suzuki
;
Shimpei Kawakami
;
Kazuhide Konishi
;
Yuko Hitomi
;
Atsushi Toyao
;
Hiroki Gunji
;
F
rederic Cumin
;
Nikolaus Schiering
;
Trixie Wagner
;
Dean
F
.
Rigel
;
Randy L. Webb
;
J眉rgen Maibaum
;
F
umiaki Yokokawa
刊名:ACS Medicinal Chemistry Letters
出版年:2014
4.
Discovery and in Vivo Evaluation o
f
Potent Dual CYP11B2 (Aldosterone Synthase) and CYP11B1 Inhibitors
作者:
Erik L. Meredith
;
Gary Ksander
;
Lauren G. Monovich
;
Julien P. N. Papillon
;
Qian Liu
;
Karl Miranda
;
Patrick Morris
;
Chang Rao
;
Robin Burgis
;
Michael Capparelli
;
Qi-Ying Hu
;
Alok Singh
;
Dean
F
.
Rigel
;
Arco Y. Jeng
;
Michael Beil
;
F
umin Fu
;
Chii-Whei Hu
;
Daniel LaSala
刊名:ACS Medicinal Chemistry Letters
出版年:2013
5.
The Discovery o
f
Novel Potent trans-3,4-Disubstituted Pyrrolidine Inhibitors o
f
the Human Aspartic Protease Renin
f
rom in Silico Three-Dimensional (3D) Pharmacophore Searches
作者:
Edwige Lorthiois
;
Werner Breitenstein
;
F
rederic Cumin
;
Claus Ehrhardt
;
Eric
F
rancotte
;
Edgar Jacoby
;
Nils Ostermann
;
Holger Sellner
;
Takatoshi Kosaka
;
Randy L. Webb
;
Dean
F
.
Rigel
;
Ulrich Hassiepen
;
Paul Richert
;
Trixie Wagner
;
J眉rgen Maibaum
刊名:Journal o
f
Medicinal Chemistry
出版年:2013
6.
A Novel Class o
f
Oral Direct Renin Inhibitors: Highly Potent 3,5-Disubstituted Piperidines Bearing a Tricyclic P3鈥?/b>P1 Pharmacophore
作者:
Nils Ostermann
;
Simon Ruedisser
;
Claus Ehrhardt
;
Werner Breitenstein
;
Andreas Marzinzik
;
Edgar Jacoby
;
Eric Vangrevelinghe
;
Johannes Ottl
;
Martin Klumpp
;
J. Constanze D. Hartwieg
;
F
rederic Cumin
;
Ulrich Hassiepen
;
J枚rg Trappe
;
Richard Sedrani
;
Sabine Geisse
;
Bernd Gerhartz
;
Paul Richert
;
Eric
F
rancotte
;
Trixie Wagner
;
Markus Kr枚mer
;
Takatoshi Kosaka
;
Randy L. Webb
;
Dean
F
.
Rigel
;
J眉rgen Maibaum
;
Daniel K. Baeschlin
刊名:Journal o
f
Medicinal Chemistry
出版年:2013
1
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