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Elsevier电子期刊(21)
ACS电子期刊(14)
在“
ACS电子期刊
”中,
命中:
14
条,耗时:0.04997 秒
在所有数据库中总计命中:
35
条
1.
Cell Active Hydroxylactam Inhibitor
s
of Human Lactate Dehydrogena
s
e with Oral Bioavailability in Mice
作者:
Han
s
E. Purkey
;
Kirk Robarge
;
Jinhua Chen
;
Zhongguo Chen
;
Laura B. Cor
s
on
;
Charle
s
Z. Ding
;
Antonio G. DiPa
s
quale
;
Peter
S
.
Dragovich
;
Charle
s
Eigenbrot
;
Marie Evangeli
s
ta
;
Benjamin P. Fauber
;
Zhenting Gao
;
Hongxiu Ge
;
Anna Hitz
;
Qunh Ho
;
S
harada S. Labadie
;
Kwong Wah Lai
;
Wenfeng Liu
;
Yajing Liu
;
Chiho Li
;
S
huguang Ma
;
S
hiva Malek
;
Thoma
s
O’Brien
;
Jodie Pang
;
David
Peters
on
;
Laurent
S
alphati
;
S
teve Sideri
s
;
Mark Ult
s
ch
;
BinQing Wei
;
Ivana Yen
;
Qin Yue
;
Huihui Zhang
;
Aihe Zhou
刊名:AC
S
Medicinal Chemi
s
try Letter
s
出版年:2016
2.
Linker Immolation Determine
s
Cell Killing Activity of Di
s
ulfide-Linked Pyrrolobenzodiazepine Antibody–Drug Conjugate
s
作者:
Donglu Zhang
;
Thoma
s
H. Pillow
;
Yong Ma
;
Jo
s
efa dela Cruz-Chuh
;
Katherine R. Kozak
;
Jack D.
S
adow
s
ky
;
Gail D. Lewi
s
Phillip
s
;
Jun Guo
;
Martine Darwi
s
h
;
Peter
Fan
;
Jingtian Chen
;
Changrong He
;
Tao Wang
;
Hui Yao
;
Zijin Xu
;
Jinhua Chen
;
John Wai
;
Zhonghua Pei
;
Corneli
s
E. C. A. Hop
;
S
. Cyru
s
Khoja
s
teh
;
Peter
S
.
Dragovich
刊名:AC
S
Medicinal Chemi
s
try Letter
s
出版年:2016
3.
Minimizing CYP2C9 Inhibition of Expo
s
ed-Pyridine NAMPT (Nicotinamide Pho
s
phoribo
s
yltran
s
fera
s
e) Inhibitor
s
作者:
Mark Zak
;
Po-wai Yuen
;
Xiongcai Liu
;
S
nahel Patel
;
Deepak
S
ampath
;
Ja
s
on Oeh
;
Bianca M. Liederer
;
Weiru Wang
;
Thoma
s
O’Brien
;
Yang Xiao
;
Nichola
s
Skelton
;
Rongbao Hua
;
Ja
s
leen Sodhi
;
Yunli Wang
;
Lei Zhang
;
Guiling Zhao
;
Xiaozhang Zheng
;
Yen-Ching Ho
;
Kenneth W. Bair
;
Peter
S
.
Dragovich
刊名:Journal of Medicinal Chemi
s
try
出版年:2016
4.
Fragment-Ba
s
ed Identification of Amide
s
Derived from tran
s
-2-(Pyridin-3-yl)cyclopropanecarboxylic Acid a
s
Potent Inhibitor
s
of Human Nicotinamide Pho
s
phoribo
s
yltran
s
fera
s
e (NAMPT)
作者:
Anthony M. Giannetti
;
Xiaozhang Zheng
;
Nichola
s
J. Skelton
;
Weiru Wang
;
Brandon J. Bravo
;
Kenneth W. Bair
;
Timm Baumei
s
ter
;
Eric Cheng
;
Li
s
a Crocker
;
Yezhen Feng
;
Janet Gunzner-To
s
te
;
Yen-Ching Ho
;
Rongbao Hua
;
Bianca M. Liederer
;
Yongbo Liu
;
Xiaolei Ma
;
Thoma
s
O’Brien
;
Ja
s
on Oeh
;
Deepak
S
ampath
;
Youming
S
hen
;
Chengcheng Wang
;
Le
s
lie Wang
;
Hongxing Wu
;
Yang Xiao
;
Po-wai Yuen
;
Mark Zak
;
Guiling Zhao
;
Qiang Zhao
;
Peter
S
.
Dragovich
刊名:Journal of Medicinal Chemi
s
try
出版年:2014
5.
S
tructure-Ba
s
ed Di
s
covery of Novel Amide-Containing Nicotinamide Pho
s
phoribo
s
yltran
s
fera
s
e (Nampt) Inhibitor
s
作者:
Xiaozhang Zheng
;
Paul Bauer
;
Timm Baumei
s
ter
;
Alexandre J. Buckmelter
;
Maureen Caligiuri
;
Karl H. Clodfelter
;
Bing
s
ong Han
;
Yen-Ching Ho
;
Nikolai Kley
;
Jian Lin
;
Dominic J. Reynold
s
;
Geeta
S
harma
;
Cha
s
e C. Smith
;
Zhongguo Wang
;
Peter
S
.
Dragovich
;
Janet Gunzner-To
s
te
;
Bianca M. Liederer
;
Ju
s
tin Ly
;
Thoma
s
O鈥橞rien
;
Angela Oh
;
Le
s
lie Wang
;
Weiru Wang
;
Yang Xiao
;
Mark Zak
;
Guiling Zhao
;
Po-wai Yuen
;
Kenneth W. Bair
刊名:Journal of Medicinal Chemi
s
try
出版年:2013
6.
S
tructure-Ba
s
ed Identification of Urea
s
a
s
Novel Nicotinamide Pho
s
phoribo
s
yltran
s
fera
s
e (Nampt) Inhibitor
s
作者:
Xiaozhang Zheng
;
Paul Bauer
;
Timm Baumei
s
ter
;
Alexandre J. Buckmelter
;
Maureen Caligiuri
;
Karl H. Clodfelter
;
Bing
s
ong Han
;
Yen-Ching Ho
;
Nikolai Kley
;
Jian Lin
;
Dominic J. Reynold
s
;
Geeta
S
harma
;
Cha
s
e C. Smith
;
Zhongguo Wang
;
Peter
S
.
Dragovich
;
Angela Oh
;
Weiru Wang
;
Mark Zak
;
Janet Gunzner-To
s
te
;
Guiling Zhao
;
Po-wai Yuen
;
Kenneth W. Bair
刊名:Journal of Medicinal Chemi
s
try
出版年:2013
7.
Identification of C-2 Hydroxyethyl Imidazopyrrolopyridine
s
a
s
Potent JAK1 Inhibitor
s
with Favorable Phy
s
icochemical Propertie
s
and High Selectivity over JAK2
作者:
Mark Zak
;
Chri
s
topher A. Hurley
;
S
tuart I. Ward
;
Philippe Bergeron
;
Kathy Barrett
;
Mercede
s
z Balaz
s
;
Wade
S
. Blair
;
Richard Bull
;
Paroma Chakravarty
;
Chri
s
tine Chang
;
Peter
Crackett
;
Gauri De
s
hmukh
;
Ja
s
on DeVo
ss
;
Peter
S
.
Dragovich
;
Charle
s
Eigenbrot
;
Charle
s
Ellwood
;
S
imon Gaine
s
;
Nico Ghilardi
;
Paul Gibbon
s
;
S
tefan Gradl
;
Peter
Gribling
;
Chri
s
Hamman
;
Eric Har
s
tad
;
Peter
Hewitt
;
Adam John
s
on
;
Tony John
s
on
;
Jane R. Kenny
;
Michael F. T. Koehler
;
Pawan Bir Kohli
;
S
harada Labadie
;
Wyne P. Lee
;
Jiangpeng Liao
;
Marya Liimatta
;
Rohan Mendonca
;
Raman Narukulla
;
Rebecca Pulk
;
Au
s
tin Reeve
;
S
cott Savage
;
S
teven Shia
;
Micah
S
teffek
;
S
avita Ubhayakar
;
Anne van Abbema
;
Ignacio Aliaga
s
;
Barbara Avitabile-Woo
;
Yi
s
ong Xiao
;
Jing Yang
;
Janu
s
z J. Kulagow
s
ki
刊名:Journal of Medicinal Chemi
s
try
出版年:2013
8.
Di
s
covery and Optimization of C-2 Methyl Imidazopyrrolopyridine
s
a
s
Potent and Orally Bioavailable JAK1 Inhibitor
s
with Selectivity over JAK2
作者:
Mark Zak
;
Rohan Mendonca
;
Mercede
s
z Balaz
s
;
Kathy Barrett
;
Philippe Bergeron
;
Wade
S
. Blair
;
Chri
s
tine Chang
;
Gauri De
s
hmukh
;
Ja
s
on DeVo
ss
;
Peter
S
.
Dragovich
;
Charle
s
Eigenbrot
;
Nico Ghilardi
;
Paul Gibbon
s
;
S
tefan Gradl
;
Chri
s
Hamman
;
Emily J. Hanan
;
Eric Har
s
tad
;
Peter
R. Hewitt
;
Chri
s
topher A. Hurley
;
Tian Jin
;
Adam John
s
on
;
Tony John
s
on
;
Jane R. Kenny
;
Michael F. T. Koehler
;
Pawan Bir Kohli
;
Janu
s
z J. Kulagow
s
ki
;
S
harada Labadie
;
Jiangpeng Liao
;
Marya Liimatta
;
Zhonghua Lin
;
Patrick J. Lupardu
s
;
Robert J. Maxey
;
Jeremy M. Murray
;
Rebecca Pulk
;
Madeleine Rodriguez
;
S
cott Savage
;
S
teven Shia
;
Micah
S
teffek
;
S
avita Ubhayakar
;
Mark Ult
s
ch
;
Anne van Abbema
;
S
tuart I. Ward
;
Ling Xiao
;
Yi
s
ong Xiao
刊名:Journal of Medicinal Chemi
s
try
出版年:2012
9.
S
pectro
s
copic and cry
s
tallographic characterization of tricarbonylchloro(.
s
igma.2-terpyridyl)rhenium. 2D-NMR evidence for a linkage i
s
omerization reaction
作者:
Edgar R. Civitello
;
Peter
S
.
Dragovich
;
Timothy B. Karpi
s
hin
;
S
abrina G. Novick
;
Geoffrey Bierach
;
John F. O'Connell
;
and T. David We
s
tmoreland
刊名:Inorganic Chemi
s
try
出版年:1993
10.
A reaction ca
s
cade leading to 1,6-didehydro[10]annulene .fwdarw. 1,5-dehydronaphthalene cyclization initiated by thiol addition
作者:
Andrew G. Myer
s
and
Peter
S.
Dragovich
刊名:Journal of the American Chemical
S
ociety
出版年:1993
1
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