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SpringerLink电子期刊(37)
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ACS电子期刊(84)
NATURE电子期刊(7)
Elsevier电子期刊(110)
在“
ACS电子期刊
”中,
命中:
84
条,耗时:小于0.01 秒
在所有数据库中总计命中:
239
条
1.
Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists
作者:
Anna Junker
;
Ramachandran Balasubramanian
;
Antonella Ciancetta
;
Elisa Uliassi
;
Evgeny Kiselev
;
Chiara Martiriggiano
;
Kevin Trujillo
;
Giorgi Mtchedlidze
;
Leah Birdwell
;
Kyle A. Brown
;
T. Kendall Harden
;
Kenneth
A.
Jacobson
刊名:Journal of Medicinal Chemistry
出版年:2016
2.
South (S)- and North (N)-Methanocarba-7-Deazaadenosine Analogues as Inhibitors of Human Adenosine Kinase
作者:
Kiran S. Toti
;
Danielle Osborne
;
Antonella Ciancetta
;
Detlev Boison
;
Kenneth
A.
Jacobson
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Purine (N)-Methanocarba Nucleoside Derivatives Lacking an Exocyclic Amine as Selective A3 Adenosine Receptor Agonists
作者:
Dilip K. Tosh
;
Antonella Ciancetta
;
Eugene Warnick
;
Robert O’Connor
;
Zhoumou Chen
;
Elizabeth Gizewski
;
Steven Crane
;
Zhan-Guo Gao
;
John A. Auchampach
;
Daniela Salvemini
;
Kenneth
A.
Jacobson
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Structure-Based Scaffold Repurposing for G Protein-Coupled Receptors: Transformation of Adenosine Derivatives into 5HT2B/5HT2C Serotonin Receptor Antagonists
作者:
Dilip K. Tosh
;
Antonella Ciancetta
;
Eugene Warnick
;
Steven Crane
;
Zhan-Guo Gao
;
Kenneth
A.
Jacobson
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Structure-Based Screening of Uncharted Chemical Space for Atypical Adenosine Receptor Agonists
作者:
David Rodríguez
;
Saibal Chakraborty
;
Eugene Warnick
;
Steven Crane
;
Zhan-Guo Gao
;
Robert O’Connor
;
Kenneth
A.
Jacobson
;
Jens Carlsson
刊名:ACS Chemical Biology
出版年:2016
6.
Rigidified A3 Adenosine Receptor Agonists: 1-Deazaadenine Modification Maintains High in Vivo Efficacy
作者:
Dilip K. Tosh
;
Steven Crane
;
Zhoumou Chen
;
Silvia Paoletta
;
Zhan-Guo Gao
;
Elizabeth Gizewski
;
John A. Auchampach
;
Daniela Salvemini
;
Kenneth
A.
Jacobson
刊名:ACS Medicinal Chemistry Letters
出版年:2015
7.
Molecular Docking Screening Using Agonist-Bound GPCR Structures: Probing the A2A Adenosine Receptor
作者:
David Rodr铆guez
;
Zhang-Guo Gao
;
Steven M. Moss
;
Kenneth
A.
Jacobson
;
Jens Carlsson
刊名:Journal of Chemical Information and Modeling
出版年:2015
8.
Structure-Based Design of Reactive Nucleosides for Site-Specific Modification of the A2A Adenosine Receptor
作者:
Steven M. Moss
;
P. Suresh Jayasekara
;
Silvia Paoletta
;
Zhan-Guo Gao
;
Kenneth
A.
Jacobson
刊名:ACS Medicinal Chemistry Letters
出版年:2014
9.
4-Alkyloxyimino Derivatives of Uridine-5鈥?triphosphate: Distal Modification of Potent Agonists as a Strategy for Molecular Probes of P2Y2, P2Y4, and P2Y6 Receptors
作者:
P. Suresh Jayasekara
;
Matthew O. Barrett
;
Christopher B. Ball
;
Kyle A. Brown
;
Eva Hammes
;
Ramachandran Balasubramanian
;
T. Kendall Harden
;
Kenneth
A.
Jacobson
刊名:Journal of Medicinal Chemistry
出版年:2014
10.
Synthesis and Anti-Renal Fibrosis Activity of Conformationally Locked Truncated 2-Hexynyl-N6-Substituted-(N)-Methanocarba-nucleosides as A3 Adenosine Receptor Antag
作者:
Akshata Nayak
;
Girish Chandra
;
Inah Hwang
;
Kyunglim Kim
;
Xiyan Hou
;
Hea Ok Kim
;
Pramod K. Sahu
;
Kuldeep K. Roy
;
Jakyung Yoo
;
Yoonji Lee
;
Minghua Cui
;
Sun Choi
;
Steven M. Moss
;
Khai Phan
;
Zhan-Guo Gao
;
Hunjoo Ha
;
Kenneth
A.
Jacobson
;
Lak Shin Jeong
刊名:Journal of Medicinal Chemistry
出版年:2014
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