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SpringerLink电子期刊(1)
NATURE电子期刊(11)
Elsevier电子期刊(7)
ACS电子期刊(25)
在“
ACS电子期刊
”中,
命中:
25
条,耗时:小于0.01 秒
在所有数据库中总计命中:
44
条
1.
Turning a Substrate Peptide into a Potent Inhibitor for the Histone Methyltransferase SETD8
作者:
Russell A. Judge
;
Haizhong Zhu
;
Anup K. Upadhyay
;
Pierre M. Bodelle
;
Charles W. Hutchins
;
Maricel Torrent
;
Violeta L. Marin
;
Wenyu Yu
;
Masoud
Vedadi
;
Fengling Li
;
Peter J. Brown
;
William N. Pappano
;
Chaohong Sun
;
Andrew M. Petros
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Discovery of Potent Pantothenamide Inhibitors of Staphylococcus aureus Pantothenate Kinase through a Minimal SAR Study: Inhibition Is Due to Trapping of the Product
作者:
Scott J. Hughes
;
Leanne Barnard
;
Katayoun Mottaghi
;
Wolfram Tempel
;
Tetyana Antoshchenko
;
Bum Soo Hong
;
Abdellah Allali-Hassani
;
David Smil
;
Masoud
Vedadi
;
Erick Strauss
;
Hee-Won Park
刊名:ACS Infectious Diseases
出版年:2016
3.
Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening
作者:
Renato Ferreira de Freitas
;
Mohammad S. Eram
;
David Smil
;
Magdalena M. Szewczyk
;
Steven Kennedy
;
Peter J. Brown
;
Vijayaratnam Santhakumar
;
Dalia Barsyte-Lovejoy
;
Cheryl H. Arrowsmith
;
Masoud
Vedadi
;
Matthieu Schapira
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Global Profiling of Acetyltransferase Feedback Regulation
作者:
David C. Montgomery
;
Julie M. Garlick
;
Rhushikesh A. Kulkarni
;
Steven Kennedy
;
Abdellah Allali-Hassani
;
Yin-Ming Kuo
;
Andrew J. Andrews
;
Hong Wu
;
Masoud
Vedadi
;
Jordan L. Meier
刊名:Journal of the American Chemical Society
出版年:2016
5.
Structure–Activity Relationship Studies for Enhancer of Zeste Homologue 2 (EZH2) and Enhancer of Zeste Homologue 1 (EZH1) Inhibitors
作者:
Xiaobao Yang
;
Fengling Li
;
Kyle D. Konze
;
Jamel Meslamani
;
Anqi Ma
;
Peter J. Brown
;
Ming-Ming Zhou
;
Cheryl H. Arrowsmith
;
H. Ümit Kaniskan
;
Masoud
Vedadi
;
Jian Jin
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2
作者:
Erik Eggert
;
Roman C. Hillig
;
Silke Koehr
;
Detlef Stöckigt
;
Jörg Weiske
;
Naomi Barak
;
Jeffrey Mowat
;
Thomas Brumby
;
Clara D. Christ
;
Antonius ter Laak
;
Tina Lang
;
Amaury E. Fernandez-Montalvan
;
Volker Badock
;
Hilmar Weinmann
;
Ingo V. Hartung
;
Dalia Barsyte-Lovejoy
;
Magdalena Szewczyk
;
Steven Kennedy
;
Fengling Li
;
Masoud
Vedadi
;
Peter J. Brown
;
Vijayaratnam Santhakumar
;
Cheryl H. Arrowsmith
;
Timo Stellfeld
;
Carlo Stresemann
刊名:Journal of Medicinal Chemistry
出版年:2016
7.
A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases
作者:
Mohammad S. Eram
;
Yudao Shen
;
Magdalena M. Szewczyk
;
Hong Wu
;
Guillermo Senisterra
;
Fengling Li
;
Kyle V. Butler
;
H. Ümit Kaniskan
;
Brandon A. Speed
;
Carlo dela Seña
;
Aiping Dong
;
Hong Zeng
;
Matthieu Schapira
;
Peter J. Brown
;
Cheryl H. Arrowsmith
;
Dalia Barsyte-Lovejoy
;
Jing Liu
;
Masoud
Vedadi
;
Jian Jin
刊名:ACS Chemical Biology
出版年:2016
8.
Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1)
作者:
Matthäus Getlik
;
David Smil
;
Carlos Zepeda-Velázquez
;
Yuri Bolshan
;
Gennady Poda
;
Hong Wu
;
Aiping Dong
;
Ekaterina Kuznetsova
;
Richard Marcellus
;
Guillermo Senisterra
;
Ludmila Dombrovski
;
Taraneh Hajian
;
Taira Kiyota
;
Matthieu Schapira
;
Cheryl H. Arrowsmith
;
Peter J. Brown
;
Masoud
Vedadi
;
Rima Al-awar
刊名:Journal of Medicinal Chemistry
出版年:2016
9.
Discovery of a Potent Class I Protein Arginine Methyltransferase Fragment Inhibitor
作者:
Renato Ferreira de Freitas
;
Mohammad S. Eram
;
Magdalena M. Szewczyk
;
Holger Steuber
;
David Smil
;
Hong Wu
;
Fengling Li
;
Guillermo Senisterra
;
Aiping Dong
;
Peter J. Brown
;
Marion Hitchcock
;
Dieter Moosmayer
;
Christian M. Stegmann
;
Ursula Egner
;
Cheryl Arrowsmith
;
Dalia Barsyte-Lovejoy
;
Masoud
Vedadi
;
Matthieu Schapira
刊名:Journal of Medicinal Chemistry
出版年:2016
10.
Correction to Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening
作者:
Renato Ferreira de Freitas
;
Mohammad S. Eram
;
David Smil
;
Magdalena M. Szewczyk
;
Steven Kennedy
;
Peter J. Brown
;
Vijayaratnam Santhakumar
;
Dalia Barsyte-Lovejoy
;
Cheryl H. Arrowsmith
;
Masoud
Vedadi
;
Matthieu Schapira
刊名:Journal of Medicinal Chemistry
出版年:2016
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