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Elsevier电子期刊(1)
ACS电子期刊(3)
在“
ACS电子期刊
”中,
命中:
3
条,耗时:小于0.01 秒
在所有数据库中总计命中:
4
条
1.
Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement
作者:
Isaac E. Marx
;
Thomas
A. Dineen
;
Jessica Able
;
Christiane Bode
;
Howard Bregman
;
Margaret Chu-Moyer
;
Erin F. DiMauro
;
Bingfan Du
;
Robert S. Foti
;
Robert T. Fremeau Jr.
;
Hua Gao
;
Hakan Gunaydin
;
Brian E. Hall
;
Liyue Huang
;
Thomas
Kornecook
;
Charles R. Kreiman
;
Daniel S. La
;
Joseph Ligutti
;
Min-Hwa Jasmine Lin
;
Dong Liu
;
Jeff S. McDermott
;
Bryan D. Moyer
;
Emily A. Peterson
;
Jonathan T. Roberts
;
Paul Rose
;
Jean Wang
;
Beth D. Youngblood
;
Violeta Yu
;
Matthew M. Weiss
刊名:ACS Medicinal Chemistry Letters
出版年:2016
2.
Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors
作者:
Erin F. DiMauro
;
Stephen Altmann
;
Loren M. Berry
;
Howard Bregman
;
Nagasree Chakka
;
Margaret Chu-Moyer
;
Elma Feric Bojic
;
Robert S. Foti
;
Robert Fremeau
;
Hua Gao
;
Hakan Gunaydin
;
Angel Guzman-Perez
;
Brian E. Hall
;
Hongbing Huang
;
Michael Jarosh
;
Thomas
Kornecook
;
Josie Lee
;
Joseph Ligutti
;
Dong Liu
;
Bryan D. Moyer
;
Daniel Ortuno
;
Paul E. Rose
;
Laurie B. Schenkel
;
Kristin Taborn
;
Jean Wang
;
Yan Wang
;
Violeta Yu
;
Matthew M. Weiss
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Discovery of Clinical Candidate 1-(4-(3-(4-(1H-Benzo[d]imidazole-2-carbonyl)phenoxy)pyrazin-2-yl)piperidin-1-yl)ethanone (AMG 579), A Potent, Selective, and Efficacious Inhibitor of Phos
作者:
Essa Hu
;
Ning Chen
;
Matthew P. Bourbeau
;
Paul E. Harrington
;
Kaustav Biswas
;
Roxanne K. Kunz
;
Kristin L. Andrews
;
Samer Chmait
;
Xiaoning Zhao
;
Carl Davis
;
Ji Ma
;
Jianxia Shi
;
Dianna Lester-Zeiner
;
Jean Danao
;
Jessica Able
;
Madelyn Cueva
;
Santosh Talreja
;
Thomas
Kornecook
;
Hang Chen
;
Amy Porter
;
Randall Hungate
;
James Treanor
;
Jennifer R. Allen
刊名:Journal of Medicinal Chemistry
出版年:2014
1
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