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Wiley电子期刊(1)
NATURE电子期刊(4)
ACS电子期刊(38)
SpringerLink电子期刊(6)
Elsevier电子期刊(38)
在“
ACS电子期刊
”中,
命中:
38
条,耗时:小于0.01 秒
在所有数据库中总计命中:
87
条
1.
A Triazolopyrimidine-Based Dihydroorotate Dehydrogenase Inhibitor with Improved Drug-like Properties for Treatment and Prevention of Malaria
作者:
Margaret A. Phillips
;
Karen L. White
;
Sreekanth Kokkonda
;
Xiaoyi Deng
;
John White
;
Farah El Mazouni
;
Kennan Marsh
;
Diana R. Tomchick
;
Krishne Manjalanagara
;
Kakali Rani Rudra
;
Grennady Wirjanata
;
Rintis Noviyanti
;
Ric N. Price
;
Jutta Marfurt
;
David M. Shackleford
;
Francis C. K. Chiu
;
Michael Campbell
;
Maria Belen Jimenez-Diaz
;
Santiago Ferrer Bazaga
;
Iñigo Angulo-Barturen
;
Maria Santos Martinez
;
Maria Lafuente-Monasterio
;
Werner Kaminsky
;
Kigbafori Silue
;
Anne-Marie Zeeman
;
Clemens Kocken
;
Didier Leroy
;
Benjamin Blasco
;
Emilie Rossignol
;
Thomas Rueckle
;
Dave Matthews
;
Jeremy N. Burrows
;
David Waterson
;
Michael J. Palmer
;
Pradipsinh K. Rathod
;
Susan
A.
Charman
刊名:ACS Infectious Diseases
出版年:2016
2.
Tetrahydro-2-naphthyl and 2-Indanyl Triazolopyrimidines Targeting Plasmodium falciparum Dihydroorotate Dehydrogenase Display Potent and Selective Antimalarial Activity
作者:
Sreekanth Kokkonda
;
Xiaoyi Deng
;
Karen L. White
;
Jose M. Coteron
;
Maria Marco
;
Laura de las Heras
;
John White
;
Farah El Mazouni
;
Diana R. Tomchick
;
Krishne Manjalanagara
;
Kakali Rani Rudra
;
Gong Chen
;
Julia Morizzi
;
Eileen Ryan
;
Werner Kaminsky
;
Didier Leroy
;
María Santos Martínez-Martínez
;
Maria Belen Jimenez-Diaz
;
Santiago Ferrer Bazaga
;
Iñigo Angulo-Barturen
;
David Waterson
;
Jeremy N. Burrows
;
Dave Matthews
;
Susan
A.
Charman
;
Margaret A. Phillips
;
Pradipsinh K. Rathod
刊名:Journal of Medicinal Chemistry
出版年:2016
3.
Revisiting the SAR of the Antischistosomal Aryl Hydantoin (Ro 13-3978)
作者:
Chunkai Wang
;
Qingjie Zhao
;
Mireille Vargas
;
Jeremy O. Jones
;
Karen L. White
;
David M. Shackleford
;
Gong Chen
;
Jessica Saunders
;
Alice C. F. Ng
;
Francis C. K. Chiu
;
Yuxiang Dong
;
Susan
A.
Charman
;
Jennifer Keiser
;
Jonathan L. Vennerstrom
刊名:Journal of Medicinal Chemistry
出版年:2016
4.
Identification of a Potential Antimalarial Drug Candidate from a Series of 2-Aminopyrazines by Optimization of Aqueous Solubility and Potency across the Parasite Life Cycle
作者:
Claire Le Manach
;
Aloysius T. Nchinda
;
Tanya Paquet
;
Diego Gonzàlez Cabrera
;
Yassir Younis
;
Ze Han
;
Sridevi Bashyam
;
Mohammed Zabiulla
;
Dale Taylor
;
Nina Lawrence
;
Karen L. White
;
Susan
A.
Charman
;
David Waterson
;
Michael J. Witty
;
Sergio Wittlin
;
Mariëtte E. Botha
;
Sindisiswe H. Nondaba
;
Janette Reader
;
Lyn-Marie Birkholtz
;
María Belén Jiménez-Díaz
;
María Santos Martínez
;
Santiago Ferrer
;
Iñigo Angulo-Barturen
;
Stephan Meister
;
Yevgeniya Antonova-Koch
;
Elizabeth A. Winzeler
;
Leslie J. Street
;
Kelly Chibale
刊名:Journal of Medicinal Chemistry
出版年:2016
5.
Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides
作者:
Stephanie Russell
;
Raphaël Rahmani
;
Amy J. Jones
;
Harriet L. Newson
;
Kevin Neilde
;
Ignacio Cotillo
;
Marzieh Rahmani Khajouei
;
Lori Ferrins
;
Sana Qureishi
;
Nghi Nguyen
;
Maria S. Martinez-Martinez
;
Donald F. Weaver
;
Marcel Kaiser
;
Jennifer Riley
;
John Thomas
;
Manu De Rycker
;
Kevin D. Read
;
Gavin R. Flematti
;
Eileen Ryan
;
Scott Tanghe
;
Ana Rodriguez
;
Susan
A.
Charman
;
Albane Kessler
;
Vicky M. Avery
;
Jonathan B. Baell
;
Matthew J. Piggott
刊名:Journal of Medicinal Chemistry
出版年:2016
6.
Trioxolane-Mediated Delivery of Mefloquine Limits Brain Exposure in a Mouse Model of Malaria
作者:
Erica M. W. Lauterwasser
;
Shaun D. Fontaine
;
Hao Li
;
Jiri Gut
;
Kasiram Katneni
;
Susan
A.
Charman
;
Philip J. Rosenthal
;
Matthew Bogyo
;
Adam R. Renslo
刊名:ACS Medicinal Chemistry Letters
出版年:2015
7.
Transformation of Poorly Water-Soluble Drugs into Lipophilic Ionic Liquids Enhances Oral Drug Exposure from Lipid Based Formulations
作者:
Yasemin Sahbaz
;
Hywel D. Williams
;
Tri-Hung Nguyen
;
Jessica Saunders
;
Leigh Ford
;
Susan
A.
Charman
;
Peter J. Scammells
;
Christopher J. H. Porter
刊名:Molecular Pharmaceutics
出版年:2015
8.
Evidence for the in Vitro Bioactivation of Aminopyrazole Derivatives: Trapping Reactive Aminopyrazole Intermediates Using Glutathione Ethyl Ester in Human Liver Microsomes
作者:
Eileen Ryan
;
Benjamin J. Morrow
;
Catherine F. Hemley
;
Jo-Anne Pinson
;
Susan
A.
Charman
;
Francis C. K. Chiu
;
Richard C. Foitzik
刊名:Chemical Research in Toxicology
出版年:2015
9.
6-Arylpyrazine-2-carboxamides: A New Core for Trypanosoma brucei Inhibitors
作者:
Rapha毛l Rahmani
;
Kung Ban
;
Amy J. Jones
;
Lori Ferrins
;
Danny Ganame
;
Melissa L. Sykes
;
Vicky M. Avery
;
Karen L. White
;
Eileen Ryan
;
Marcel Kaiser
;
Susan
A.
Charman
;
Jonathan B. Baell
刊名:Journal of Medicinal Chemistry
出版年:2015
10.
Inhibitors of Plasmodial Serine Hydroxymethyltransferase (SHMT): Cocrystal Structures of Pyrazolopyrans with Potent Blood- and Liver-Stage Activities
作者:
Matthias C. Witschel
;
Matthias Rottmann
;
Anatol Schwab
;
Ubolsree Leartsakulpanich
;
Penchit Chitnumsub
;
Michael Seet
;
Sandro Tonazzi
;
Geoffrey Schwertz
;
Frank Stelzer
;
Thomas Mietzner
;
Case McNamara
;
Frank Thater
;
C茅line Freymond
;
Aritsara Jaruwat
;
Chatchadaporn Pinthong
;
Pinpunya Riangrungroj
;
Mouhssin Oufir
;
Matthias Hamburger
;
Pascal M盲ser
;
Laura M. Sanz-Alonso
;
Susan
Charman
;
Sergio Wittlin
;
Yongyuth Yuthavong
;
Pimchai Chaiyen
;
Fran莽ois Diederich
刊名:Journal of Medicinal Chemistry
出版年:2015
1
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