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Wiley电子期刊(8)	NATURE电子期刊(14)	ACS电子期刊(101)
SpringerLink电子期刊(137)	Elsevier电子期刊(648)

在“Elsevier电子期刊”中，命中：648条，耗时：小于0.01 秒

在所有数据库中总计命中：908条

1.Positional isomers of bispyridine benzene derivatives induce efficacy changes on mGlu₅ negative allosteric modulation

作者：Xavier Gó ; mez-Santacana^a ; ^b ; ^c ; ¹ ; James A.R. Dalton^b ; ^d ; Xavier Rovira^e ; ^f ; Jean Philippe Pin^e ; ^f ; Cyril Goudet^e ; ^f ; Pau Gorostiza^c ; ^g ; ^h ; Jesú ; s Giraldo^b ; ^d ; Amadeu Llebaria^a ; ^{amadeu.llebaria@iqac.csic.es}

关键词：mGlu5 ; Isomers ; Partial efficacy ; NAM ; Antagonist ; Inverse agonist

刊名：European Journal of Medicinal Chemistry

出版年：2017

2.3-Furan-2-yl-N-p-tolyl-acrylamide, a positive allosteric modulator of the α7 nicotinic receptor, reverses schizophrenia-like cognitive and social deficits in rats

作者：Agnieszka Potasiewicz^a ; Małgorzata Hołuj^a ; Tomasz Kos^a ; Piotr Popik^a ; Hugo R. Arias^b ; Agnieszka Nikiforuk^a ; ^{nikifor@if-pan.krakow.pl}

关键词：α7 Nicotinic acetylcholine receptors ; Positive allosteric modulator ; Animal model of schizophrenia ; Cognitive flexibility ; Recognition memory ; Antipsychotics

刊名：Neuropharmacology

出版年：2017

3.Characterization of P2X4 receptor agonists and antagonists by calcium influx and radioligand binding studies

作者：Aliaa Abdelrahman^a ; Vigneshwaran Namasivayam^a ; ^c ; Sonja Hinz^a ; Anke C. Schiedel^a ; Meryem Kö ; se^a ; Maggi Burton^b ; Ali El-Tayeb^a ; ¹ ; Michel Gillard^b ; Jü ; rgen Bajorath^c ; Marc de Ryck^b ; Christa E. Mü ; ller^a ; ^{christa.mueller@uni-bonn.de}

关键词：Ap3A ; diadenosine triphosphate ; Ap4A ; diadenosine tetraphosphate ; Ap5A ; diadenosine pentaphosphate ; AR-C67085MX ; 2-propylthio-β ; γ-dichloromethylene-ATP ; PSB0412 ; 2-propargylthio-β ; γ-dichloromethylene-ATP ; 5-BDBD ; 5-(3-bromophenyl)-1 ; 3-dihydro-2H-benzofuro[3 ; 2-e]-1 ; 4-diazepin-2-one ; BzATP ; 2&prime ; (3&prime ; )-O-(4-benzoylbenzoyl)adenosine 5&prime ; -triphosphate ; CHO-K1 cells ; Chinese hamster ovary cells ; HBSS ; Hank&rsquo ; s balanced salt solution ; HEPES ; 4-(2-hydroxyethyl)-1-piperazine ethanesulfoni

刊名：Biochemical Pharmacology

出版年：2017

4.The GABA_B positive allosteric modulators CGP7930 and GS39783 stimulate ERK1/2 signalling in cells lacking functional GABA_B receptors

作者：Maria C. Olianas ; ^{molianas@unica.it} ; Simona Dedoni ; Pierluigi Onali

关键词：CGP7930 (PubChem CID ; 5024764) ; GS39783 (PubChem CID ; 6604928) ; (-)-baclofen (PubChem CID ; 44602) ; SKF97541 (PubChem CID ; 5230) ; CGP55845 (PubChem CID ; 5311042) ; CGP54626 (PubChem CID ; 197584) ; phorbol 12-myristate 13 acetate (PubChem CID ; 27924) ; Go 6850 (PubChem CID ; 2396) ; 5Z-7-oxozeaenol (PubChem CID ; 9863776) ; GW5074 (PubChem CID ; 5924208)

刊名：European Journal of Pharmacology

出版年：2017

5.Novel Dopamine Therapeutics for Cognitive Deficits in Schizophrenia

作者：Amy F.T. Arnsten^a ; ^{amy.arnsten@yale.edu" class="auth_mail" title="E-mail the corresponding author} ; Ragy R. Girgis^b ; David L. Gray^c ; Richard B. Mailman^d

关键词：D1 agonist ; D2 receptors ; Executive function ; Prefrontal cortex ; Schizophrenia ; Working memory

刊名：Biological Psychiatry

出版年：2017

6.Delineation of the functional properties and the mechanism of action of TMPPAA, an allosteric agonist and positive allosteric modulator of 5-HT₃ receptors

作者：Agnes Gasiorek^a ; Sarah M. Trattnig^a ; Philip K. Ahring^b ; ¹ ; Uffe Kristiansen^a ; Bente Frø ; lund^a ; Kristen Frederiksen^c ; Anders A. Jensen^a ; ^{aaj@sund.ku.dk" class="auth_mail" title="E-mail the corresponding author}

关键词：Cys-loop receptor ; 5-HT3 receptor ; Allosteric agonist ; Allosteric modulation ; Ago-PAM ; TMPPAA

刊名：Biochemical Pharmacology

出版年：2016

7.Diverse modes of NMDA receptor positive allosteric modulation: Mechanisms and consequences

作者：David H. Hackos ; ^{hackos.david@gene.com" class="auth_mail" title="E-mail the corresponding author} ; Jesse E. Hanson ; ^{hanson.jesse@gene.com" class="auth_mail" title="E-mail the corresponding author}

关键词：PYD-106 ; CIQ ; Spermine ; Pregnenolone ; GNE-6901 ; GNE-8324 ; TCN-201 ; SGE201 ; SGE301 ; Schizophrenia

刊名：Neuropharmacology

出版年：2017

8.Integrated regulation of AMPA glutamate receptor phosphorylation in the striatum by dopamine and acetylcholine

作者：Bing Xue^a ; Elton C. Chen^b ; Nan He^a ; Dao-Zhong Jin^a ; Li-Min Mao^a ; John Q. Wang^a ; ^b ; ^c ; ^{wangjq@umkc.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：D1 ; D2 ; Muscarinic receptor ; S845 ; Protein kinase A ; Caudate putamen ; Nucleus accumbens ; Positive allosteric modulator

刊名：Neuropharmacology

出版年：2017

9.(+)-and (−)-Phenazocine enantiomers: Evaluation of their dual opioid agonist/σ₁ antagonist properties and antinociceptive effects

关键词：Sigma-1 receptor ; (+)-Phenazocine ; (&minus ; )-Phenazocine ; Mechanical antinociception ; Bifunctional ligand ; Opioid

刊名：European Journal of Medicinal Chemistry

出版年：2017

10.Metabotropic glutamate receptors and neurodegenerative diseases

作者：Fabiola M. Ribeiro^a ; Luciene B. Vieira^b ; Rita G.W. Pires^c ; Roenick P. Olmo^a ; Stephen S.G. Ferguson^d ; ^{sferguso@uottawa.ca}

关键词：AMPA ; α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid ; Aβ ; amyloid β peptide ; AD ; Alzheimer&rsquo ; s disease ; APP ; amyloid precursor protein ; BDNF ; brain derived neurotrophic factor ; BF ; basal forebrain ; CGA ; chromogranin A ; CNS ; central nervous system ; DAG ; diacylghycerol ; ERK ; extracellular signal-regulated kinase ; GABA ; gamma-aminobutyric acid ; GDNF ; glial cell line-derived neurotrophic factor ; GIRK ; inward rectifying K+ channels ; GP ; globus pallidum ; GPe ; globus pallidum externa ; GPCR ; G

刊名：Pharmacological Research

出版年：2017

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