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Elsevier电子期刊(38)
在“
Elsevier电子期刊
”中,
命中:
38
条,耗时:小于0.01 秒
在所有数据库中总计命中:
38
条
1.
Substrate specificity of human matriptase-2
作者:
M. Wysocka
;
N. Gruba
;
A. Miecznikowska
;
J. Popow-Stellmaszyk
;
M. G眉tschow
;
M. Stirnberg
;
N. Furtmann
;
J.
Bajorath
;
A. Lesner
;
K. Rolka
关键词:
Matriptase-2
;
Combinatorial chemistry
;
Fluorogenic substrates
;
Internally quenched substrates
刊名:Biochimie
出版年:February, 2014
2.
Evaluation of molecular model-based discovery of ecto-5¡ä-nucleotidase inhibitors on the basis of X-ray structures
作者:
Norbert Furtmann
;
J¨¹rgen
Bajorath
关键词:
Ecto-5&prime
;
-nucleotidase
;
Small molecule inhibitors
;
Docking
;
Virtual screening
;
Comparative protein models
;
X-ray structures
刊名:Bioorganic and Medicinal Chemistry
出版年:2013
3.
New chemotypes for wALADin1-like inhibitors of delta-aminolevulinic acid dehydratase from Wolbachia endobacteria
作者:
Christian S. Lentz
;
Dagmar Stumpfe
;
Juergen
Bajorath
;
Michael Famulok
;
Achim Hoerauf
;
Kenneth M. Pfarr
关键词:
Delta-aminolevulinic acid dehydratase
;
Wolbachia
;
Brugia malayi
;
Heme biosynthesis
;
wALADin
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2013
4.
Identification of sulfonic acids as efficient ecto-5鈥?nucleotidase inhibitors
作者:
Jamshed Iqbal
;
Aamer Saeed
;
Rabia Raza
;
Abdul Matin
;
Abdul Hameed
;
Norbert Furtmann
;
Joanna Lecka
;
Jean S茅vigny
;
J眉rgen
Bajorath
关键词:
Adenosine
;
Ecto-5&prime
;
-nucleotidase
;
Enzyme inhibition
;
Sulfonic acids
;
Binding mode
;
Cytotoxicity
刊名:European Journal of Medicinal Chemistry
出版年:December, 2013
5.
Activity profile relationships between structurally similar promiscuous compounds
作者:
Ye Hu
;
J眉rgen
Bajorath
关键词:
Compound activity data
;
Compound promiscuity
;
Structural similarity
;
Matched molecular pairs
;
Activity patterns
;
Activity cliffs
;
Target selectivity
刊名:European Journal of Medicinal Chemistry
出版年:November, 2013
6.
Large-scale SAR analysis
作者:
Jü
;
rgen
Bajorath
bajorath
@bit.uni-bonn.de
刊名:Drug Discovery Today: Technologies
出版年:2013
7.
Molecular crime scene investigation - dusting for fingerprints
作者:
J¨¹rgen
Bajorath
刊名:Drug Discovery Today: Technologies
出版年:2013
8.
Compound promiscuity: what can we learn from current data?
作者:
Ye Hu
;
J¨¹rgen
Bajorath
刊名:Drug Discovery Today
出版年:2013
9.
Chemoinformatics: A view of the field and current trends in method development
作者:
Martin Vogt
;
J¨¹rgen
Bajorath
关键词:
MCS
;
maximum common subgraph
;
MMP
;
matched molecular pair
;
QSAR
;
quantitative structure&ndash
;
activity relationship
;
ROC
;
receiver operating characteristic
;
SMILES
;
simplified molecular input line entry specification
;
SVM
;
support vector machine
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
10.
Chemoinformatics: Recent advances at the interfaces between computer and chemical information sciences, chemistry, and drug discovery
作者:
J¨¹rgen
Bajorath
刊名:Bioorganic and Medicinal Chemistry
出版年:2012
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