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Wiley电子期刊(1)	SpringerLink电子期刊(13)	Elsevier电子期刊(42)
Springer电子图书(2)	NATURE电子期刊(3)	ACS电子期刊(11)

在“Elsevier电子期刊”中，命中：42条，耗时：小于0.01 秒

在所有数据库中总计命中：72条

1.Context-Dependent Role of Oxidized Lipids and Lipoproteins in Inflammation

作者：Yury I. Miller¹ ; ^{yumiller@ucsd.edu} ; John Y.-J. Shyy¹

关键词：oxidized lipid ; inflammation ; toll-like receptor ; inflammasome

刊名：Trends in Endocrinology & Metabolism

出版年：2017

2.Biased agonism: An emerging paradigm in GPCR drug discovery

作者：Zoran Rankovic^a ; ^{rankovic_zoran@lilly.com" class="auth_mail" title="E-mail the corresponding author} ; Tarsis F. Brust^b ; Laura M. Bohn^b ; ^{lbohn@scripps.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：Biased ligand ; Functional selectivity ; GPCR ; Drug discovery

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

3.Evidence for biased agonists and antagonists at the endothelin receptors

作者：Janet J. Maguire ^{jjm1003@medschl.cam.ac.uk" class="auth_mail" title="E-mail the corresponding author}

关键词：G protein coupled receptors ; Endothelin ; ETA ; ETB ; Biased agonism ; Biased antagonism ; β-Arrestin ; Bosentan ; Pathway selectivity ; IRL1620

刊名：Life Sciences

出版年：2016

4.Quantification of adenosine A₁ receptor biased agonism: Implications for drug discovery

作者：Jo-Anne Baltos ; Karen J. Gregory ; Paul J. White ; Patrick M. Sexton ; Arthur Christopoulos ; ^{arthur.christopoulos@monash.edu" class="auth_mail" title="E-mail the corresponding author} ; Lauren T. May ; ^{lauren.may@monash.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：A1-FlpIn-CHO ; Chinese hamster ovary cell with FlpIn&trade ; vector stably expressing human adenosine A1 receptor ; A1AR ; adenosine A1 receptor ; A6730 ; 1 ; 3-dihydro-1-(1-((4-(6-phenyl-1H-imidazo[4 ; 5-g]quinoxalin-7-yl)phenyl)methyl)-4-piperidinyl)-2H-benzimidazol-2-one trifluoroacetate salt hydrate ; ADA ; adenosine deaminase ; Akt/PKB ; protein kinase B ; ANOVA ; analysis of variance ; AR ; adenosine receptor ; ATP ; adenosine triphosphate ; BSA ; bovine serum albumin ; CPA ; N6-cyclopentyladenosine ; ddADO ; 2&pri

刊名：Biochemical Pharmacology

出版年：2016

5.Systematic analysis of factors influencing observations of biased agonism at the mu-opioid receptor

作者：Georgina L. Thompson^a ; ^b ; J. Robert Lane^a ; Thomas Coudrat^a ; Patrick M. Sexton^a ; Arthur Christopoulos^a ; ^{arthur.christopoulos@monash.edu" class="auth_mail" title="E-mail the corresponding author} ; Meritxell Canals^a ; ^{meri.canals@monash.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：AC ; adenylyl cyclase ; α-neo ; α-neoendorphin ; β-arr1 and β-arr2 ; β-arrestin 1 and 2 ; BRET ; bioluminescence resonance energy transfer ; CHO ; Chinese hamster ovary ; DAMGO ; d-Ala2-N-MePhe4-Gly-ol enkephalin ; endo ; endomorphin ; pERK ; extracellular signal regulated kinases 1/2 phosphorylation ; GIRK ; G protein-gated inwardly rectifying K+ channel ; GPCR ; G protein-coupled receptor ; GRK ; G protein-coupled receptor kinase ; enk ; enkephalin ; MOP ; μ-opioid receptor ; PKC ; protein kinase C ; PCA ; principal compo

刊名：Biochemical Pharmacology

出版年：2016

6.Recent updates on GPCR biased agonism

作者：André ; S. Pupo^a ; ^{aspupo@ibb.unesp.br" class="auth_mail" title="E-mail the corresponding author} ; Diego A. Duarte^b ; Vanessa Lima^a ; ^b ; Larissa B. Teixeira^b ; Lucas T. Parreiras-e-Silva^b ; Claudio M. Costa-Neto^b ; ^{claudio@fmrp.usp.br" class="auth_mail" title="E-mail the corresponding author}

关键词：GPCR ; 7TMR ; Functional selectivity

刊名：Pharmacological Research

出版年：2016

7.Cardiac action of the first G protein biased small molecule apelin agonist

作者：Cai Read^a ; ¹ ; Christopher M. Fitzpatrick^b ; ¹ ; Peiran Yang^a ; ¹ ; Rhoda E. Kuc^a ; Janet J. Maguire^a ; ² ; Robert C. Glen^c ; ^d ; ² ; Richard E. Foster^b ; ² ; Anthony P. Davenport^a ; ² ; ^{apd10@medschl.cam.ac.uk" class="auth_mail" title="E-mail the corresponding author}

关键词：Apelin ; Biased agonism ; G protein coupled receptor ; Cardiovascular ; In vivo

刊名：Biochemical Pharmacology

出版年：2016

8.Label-free cell phenotypic profiling and pathway deconvolution of neurotensin receptor-1

作者：Tao Hou^a ; Liying Shi^b ; Jixia Wang^a ; Lai Wei^a ; Lala Qu^a ; Xiuli Zhang^a ; ^c ; ^{zhangxiuli@dicp.ac.cn" class="auth_mail" title="E-mail the corresponding author} ; Xinmiao Liang^a ; ^{liangxm@dicp.ac.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：Neurotensin receptor-1 ; Pathway ; Label-free cell phenotypic profiling ; Biased agonism

刊名：Pharmacological Research

出版年：2016

9.The Extracellular Surface of the GLP-1 Receptor Is a Molecular Trigger for Biased Agonism

作者：Denise Wootten¹ ; ^{denise.wootten@monash.edu" class="auth_mail" title="E-mail the corresponding author} ; Christopher A. Reynolds³ ; Kevin J. Smith³ ; Juan C. Mobarec³ ; Cassandra Koole¹ ; ⁴ ; Emilia E. Savage¹ ; Kavita Pabreja¹ ; John Simms⁵ ; Rohan Sridhar¹ ; Sebastian G.B. Furness¹ ; Mengjie Liu² ; Philip E. Thompson² ; Laurence J. Miller⁶ ; Arthur Christopoulos¹ ; Patrick M. Sexton¹ ; ^{patrick.sexton@monash.edu" class="auth_mail" title="E-mail the corresponding author}

刊名：Cell

出版年：2016

10.Key interactions by conserved polar amino acids located at the transmembrane helical boundaries in Class B GPCRs modulate activation, effector specificity and biased signalling in the glucagon-like peptide-1 receptor

作者：Denise Wootten^a ; ^{denise.wootten@monash.edu" class="auth_mail" title="E-mail the corresponding author} ; Christopher A. Reynolds^b ; Kevin J. Smith^b ; Juan C. Mobarec^b ; Sebastian G.B. Furness^a ; Laurence J. Miller^c ; Arthur Christopoulos^a ; Patrick M. Sexton^a ; ^{patrick.sexton@monash.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：cAMP ; 3&prime ; 5&prime ; -cyclic adenosine monophosphate ; CHO ; Chinese hamster ovary ; CRF1R ; corticotrophin releasing factor receptor-1 ; DMEM ; Dulbecco&rsquo ; s modified Eagle medium ; FBS ; fetal bovine serum ; GCGR ; glucagon receptor ; GLP-1 ; glucagon-like peptide-1 ; GPCR ; G protein-coupled receptor ; iCa2+ ; intracellular calcium ; pERK ; extracellular signal-regulated kinase 1 and 2 phosphorylation ; PBS ; phosphate buffered saline ; TM ; transmembrane helix

刊名：Biochemical Pharmacology

出版年：2016

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