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Elsevier电子期刊(5)
ACS电子期刊(1)
在“
Elsevier电子期刊
”中,
命中:
5
条,耗时:小于0.01 秒
在所有数据库中总计命中:
6
条
1.
Identification and SAR of novel pyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)
作者:
Giovanna Pescatore
;
Danila Branca
;
Fabrizio Fiore
;
Olaf Kinzel
;
Laura Llauger Bufi
;
Ester Muraglia
;
Federica Orvieto
;
Michael Rowley
;
Carlo Toniatti
;
Caterina
Torrisi
;
Philip Jones
关键词:
Pyrrolo[1
;
2-
a
]pyrazin-1(2
H
)-one
;
Poly(ADP-ribose) polymerase
;
PARP-1
;
Oncology
;
Selectivity
;
BRCA1
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
2.
Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazin-3(2H)-ones as potent poly(ADP–ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells
作者:
Federica Ferrigno
;
Danila Branca
;
Olaf Kinzel
;
Samuele Lillini
;
Laura Llauger Bufi
;
Edith Monteagudo
;
Ester Muraglia
;
Michael Rowley
;
Carsten Schultz-Fademrecht
;
Carlo Toniatti
;
Caterina
Torrisi
;
Phil
关键词:
Anticancer agents
;
PARP-1 inhibitor
;
BRCA1 deficient cancer cells
;
6-[4-Fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4
;
5-dimethylpyridazin-3(2
H
)-ones
;
Coupling reactions
;
SAR exploration
;
Pharmacokinetic properties
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
3.
Discovery and SAR of novel, potent and selective hexahydrobenzonaphthyridinone inhibitors of poly(ADP-ribose)polymerase-1 (PARP-1)
作者:
Caterina
Torrisi
;
Monica Bisbocci
;
Raffaele Ingenito
;
Jesus M. Ontoria
;
Michael Rowley
;
Carsten Schultz-Fademrecht
;
Carlo Toniatti
;
Philip Jones
关键词:
PARP
;
Cancer
;
Hexahydrobenzonaphthyridinone
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
4.
A novel base-mediated intramolecular hydroamination to build fused heteroaryl pyrazinones
作者:
Laura Llauger
;
Costanza Bergami
;
Olaf D. Kinzel
;
Samuele Lillini
;
Giovanna Pescatore
;
Caterina
Torrisi
;
Philip Jones
关键词:
Intramolecular hydroamination
;
Pyrrolopyrazinones
;
Fused-heteroaryl pyrazinones
;
DBU-mediated cyclisation
;
Isomerisation
刊名:Tetrahedron Letters
出版年:2009
5.
Lower sperm aneuploidy rate is associated with a higher pregnancy rate in unselected patients undergoing intracytoplasmic sperm injection
作者:
Calogero
;
Aldo E.
;
Burrello
;
Nunziatina
;
Grazioso
;
Caterina
;
Adele
;
De Palma
;
Torrisi
;
Carlo
;
et. al.
刊名:Fertility and Sterility
出版年:2002
1
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