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内部出版物
Wiley电子期刊(4)
Elsevier电子期刊(6)
在“
Elsevier电子期刊
”中,
命中:
6
条,耗时:0.0249918 秒
在所有数据库中总计命中:
10
条
1.
Identification and SAR of novel pyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)
作者:
Giovanna Pescatore
;
Danila
Branca
;
Fabrizio Fiore
;
Olaf Kinzel
;
Laura Llauger Bufi
;
Ester Muraglia
;
Federica Orvieto
;
Michael Rowley
;
Carlo Toniatti
;
Caterina Torrisi
;
Philip Jones
关键词:
Pyrrolo[1
;
2-
a
]pyrazin-1(2
H
)-one
;
Poly(ADP-ribose) polymerase
;
PARP-1
;
Oncology
;
Selectivity
;
BRCA1
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
2.
Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazin-3(2H)-ones as potent poly(ADP–ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells
作者:
Federica Ferrigno
;
Danila
Branca
;
Olaf Kinzel
;
Samuele Lillini
;
Laura Llauger Bufi
;
Edith Monteagudo
;
Ester Muraglia
;
Michael Rowley
;
Carsten Schultz-Fademrecht
;
Carlo Toniatti
;
Caterina Torrisi
;
Phil
关键词:
Anticancer agents
;
PARP-1 inhibitor
;
BRCA1 deficient cancer cells
;
6-[4-Fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4
;
5-dimethylpyridazin-3(2
H
)-ones
;
Coupling reactions
;
SAR exploration
;
Pharmacokinetic properties
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2010
3.
Identification of substituted pyrazolo[1,5-a
作者:
Federica Orvieto
;
Danila
Branca
;
Claudia Giomini
;
Philip Jones
;
Uwe Koch
;
Jesus M. Ontoria
;
Maria Cecilia Palumbi
;
Michael Rowley
;
Carlo Toniatti
;
Ester Muraglia
关键词:
PARP-1 inhibitor
;
Pyrazole
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
4.
Identification of aminoethyl pyrrolo dihydroisoquinolinones as novel poly(ADP-ribose) polymerase-1 inhibitors
作者:
Danila
Branca
;
Mauro Cerretani
;
Philip Jones
;
Uwe Koch
;
Federica Orvieto
;
Maria Cecilia Palumbi
;
Michael Rowley
;
Carlo Toniatti
;
Ester Muraglia
关键词:
Parp1 Inhibitor
;
Anticancer
;
Indoles
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
5.
Discovery of N
作者:
Gabriella Dessole
;
Danila
Branca
;
Federica Ferrigno
;
Olaf Kinzel
;
Ester Muraglia
;
Maria Cecilia Palumbi
;
Michael Rowley
;
Sergio Serafini
;
Christian Steinkü
;
hler
;
Philip Jones
关键词:
Hedgehog pathway
;
Smoothened antagonists
;
N
-[(1-aryl-1
H
-indazol-5-yl)methyl]amide derivatives
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
6.
2-Trifluoroacetylthiophene oxadiazoles as potent and selective class II human histone deacetylase inhibitors
作者:
Ester Muraglia
;
Sergio Altamura
;
Danila
Branca
;
Ottavia Cecchetti
;
Federica Ferrigno
;
Maria Vittoria Orsale
;
Maria Cecilia Palumbi
;
Michael Rowley
;
Rita Scarpelli
;
Christian Steinkü
;
hler
;
Philip J
关键词:
HDAC
;
Inhibitors
;
Trifluoroacetyl
;
Oxadiazoles
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
1
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