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Elsevier电子期刊(9)
ACS电子期刊(1)
在“
Elsevier电子期刊
”中,
命中:
9
条,耗时:0.0100191 秒
在所有数据库中总计命中:
10
条
1.
Design and synthesis of 4,5,6,7‐tetrahydro‐1H‐1,2‐diazepin‐7‐one
derivatives
as a new series of Phosphodiesterase 4 (PDE4) inhibitors
作者:
Sara Guariento
a
;
Anna Karawajczyk
b
;
James A. Bull
b
;
Gessica Marchini
c
;
Martyna Bielska
b
;
Xenia Iwanowa
b
;
Olga Bruno
a
;
Paola Fossa
a
;
Fabrizio Giordanetto
b
;
fabrizio.giordanetto@deshawresearch.com
关键词:
Phosphodiesterase 4
;
PDE4 inhibitors
;
Diazepinone
derivatives
;
Compound library
刊名:Bioorganic & Medicinal Chemistry Letters
出版年:2017
2.
Imidazopyridine-fused [1,3]-
diazepinone
s part 2: Structure-activity relationships and antiproliferative activity against melanoma cells
作者:
Virginie Bellet
;
Laure Lichon
;
Dominique P. Arama
;
Audrey Gallud
;
Vincent Lisowski
;
Ludovic T. Maillard
;
Marcel Garcia
;
Jean Martinez
;
Nicolas Masurier
;
nicolas.masurier@umontpellier.fr
关键词:
Imidazo[1
;
2-a]pyridine
;
Polyfused heterocycles
;
Diazepinone
s
;
Antitumor activity
;
Melanoma
刊名:European Journal of Medicinal Chemistry
出版年:2017
3.
Novel chiral ferrocenylpyrazolo[1,5-a][1,4]diazepin-4-one
derivatives
- Synthesis, characterization and inhibition against lung cancer cells
作者:
Shi-Li Shen
a
;
Jin-Hui Shao
b
;
Ji-Zhuang Luo
b
;
Jin-Ting Liu
a
;
Jun-Ying Miao
b
;
miaojy@sdu.edu.cn
;
Bao-Xiang Zhao
a
;
bxzhao@sdu.edu.cn
;
sduzhao@hotmail.com
关键词:
Pyrazole
;
Ferrocene
;
Chiral
diazepinone
;
Lung cancer cells
;
Cell cycle arrest
;
Apoptosis
刊名:European Journal of Medicinal Chemistry
出版年:2013
4.
An efficient synthesis of pyrido-imidazodiazepinediones
作者:
Dominique P. Arama
;
Vincent Lisowski
;
Eliana Scarlata
;
Pierre Fulcrand
;
Ludovic T. Maillard
;
Jean Martinez
;
Nicolas Masurier
;
nicolas.masurier@univ-montp1.fr
关键词:
Diazepinone
s
;
Friedel&ndash
;
Crafts acylation
;
Imidazo[1
;
2-a]pyridine
;
Polyfused heterocycles
;
Urea
derivatives
刊名:Tetrahedron Letters
出版年:2013
5.
Furo- and thieno-fused 1,3-diazepine-4,6-diones
作者:
Merve Sinem Ozer
;
Gani Koza
;
Ertan Sahin
;
Metin Balci
关键词:
Benzo
diazepinone
;
Furo-diazepinedione
;
Thieno-diazepinedione
;
Curtius rearrangement
刊名:Tetrahedron Letters
出版年:27 November, 2013
6.
An efficient one-pot synthesis, structure, antimicrobial and antioxidant investigations of some novel quinolyldibenzo[b,e][1,4]
diazepinone
s
作者:
Narsidas J. Parmar
a
;
njpchemdeptspu@yahoo.co.in
;
Hitesh A. Barad
a
;
Bhavesh R. Pansuriya
a
;
Shashikant B. Teraiya
a
;
Vivek K. Gupta
b
;
Rajni Kant
b
关键词:1 ;
4-Diazepines
;
Solvent-free method
;
Antimicrobial agents
;
Quinoline
derivatives
;
Antitubercular agents
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2012
7.
Chemistry and biological activity of azoprenylated secondary metabolites
作者:
Salvatore Genovese
;
Massimo Curini
;
Francesco Epifano
关键词:
Alkaloids
;
Biological activity
;
Biosynthesis
;
Chemical synthesis
;
Microbial secondary metabolites
;
Prenylazo secondary metabolites
;
Rutaceae
刊名:Phytochemistry
出版年:2009
8.
Concise synthesis of ω-fluoroalkylated ketoesters. A building block for the synthesis of six-, seven-, and eight-membered fluoroalkyl substituted 1,2-diaza-3-one heterocycles
作者:
Wen Wan
;
Jie Hou
;
Haizhen Jiang
;
Yangli Wang
;
Shizheng Zhu
;
Hongmei Deng
;
Jian Hao
刊名:Tetrahedron
出版年:2009
9.
Imidazo-thiazine, -diazinone and -
diazepinone
derivatives
. Synthesis, structure and benzodiazepine receptor binding
作者:
Kiec-Kononowicz
;
Katarzyna
;
Karolak-Wojciechowska
;
Janina
;
Mü
;
ller
;
Christa E.
;
Schumacher
;
Britta
;
et. al.
关键词:
benzodiazepine receptor
;
GABA
A
receptor
;
imidazo[2
;
1-b]thiazines
;
imidazo[2
;
1-b]pyrimidinone
;
imidazo[2
;
1-b]
diazepinone
刊名:European Journal of Medicinal Chemistry
出版年:2001
1
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