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Elsevier电子期刊(26)
在“
Elsevier电子期刊
”中,
命中:
26
条,耗时:小于0.01 秒
在所有数据库中总计命中:
26
条
1.
Robin
Ganellin
gives his views on medicinal chemistry and drug discovery
作者:
Ganellin
;
C. Robin
关键词:
Drug Discovery
;
Cell biology
;
Chemical Biology
;
Molecular Medicine
;
medicinal chemistry
;
drug discovery
;
chemistry
;
blockbuster drugs
刊名:Drug Discovery Today
出版年:2004
2.
Molecular features of the prazosin molecule required for activation of Transport-P
作者:
Joaquim Fern
;
o Mendes da Silva
;
Marcus Walters
;
Saad Al-Damluji
;
C. Robin
Ganellin
关键词:
Transport-P
;
Prazosin
;
Peptidergic neurones
;
Quinazoline
;
Furan
;
Antidepressant
;
Amine uptake
刊名:Bioorganic and Medicinal Chemistry
出版年:2008
3.
Synthesis of novel ketoconazole derivatives as inhibitors of the human Pregnane X Receptor (PXR; NR1I2; also termed SXR, PAR)
作者:
Bhaskar C. Das
;
Ankanahlli V. Madhukumar
;
Jaime Anguiano
;
Sean Kim
;
Michael Sinz
;
Tatyana A. Zvyaga
;
Eoin C. Power
;
C. Robin
Ganellin
;
Sridhar Mani
关键词:
Pregnane X receptor
;
PXR
;
Ketoconazole
;
Azole
;
Analogs
;
Nuclear receptors
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2008
4.
Synthesis and pharmacological testing of polyaminoquinolines as blockers of the apamin-sensitive Ca
2+
-activated K
+
channel (SK
Ca
)
作者:
David I. Fletcher
;
C. Robin
Ganellin
;
Aless
;
ro Piergentili
;
Philip M. Dunn
;
Donald H. Jenkinson
关键词:
Quinoline
;
Aminoquinoline
;
Guanidine
;
Apamin
;
Potassium ion channel
;
Calcium activated
;
SK
Ca
;
SK3
;
AHP
;
After-hyperpolarization
刊名:Bioorganic and Medicinal Chemistry
出版年:2007
5.
Partial structures of ketoconazole as modulators of the large conductance calcium-activated potassium channel (BK
Ca
)
作者:
Eoin C. Power
;
C. Robin
Ganellin
and David C.H. Benton
关键词:
Potassium channels
;
Opener
;
Blocker
;
Large conductance
;
BK
Ca
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2006
6.
Structural variations of 1-(4-(phenoxymethyl)benzyl)piperidines as nonimidazole histamine H
3
receptor antagonists
作者:
Mikó
;
Tibor
;
Ligneau
;
Xavier
;
Pertz
;
Heinz H.
;
Arrang
;
Jean-Michel
;
Robin
Ganellin
;
C.
;
et. al.
关键词:
Histamine H
3
;
Antagonist
;
Nonimidazole
;
Receptor
;
Medicinal chemistry
刊名:Bioorganic and Medicinal Chemistry
出版年:2004
7.
The sleep inducing brain lipid cis-oleamide (cOA) does not modulate serotonergic transmission in the CA1 pyramidal neurons of the hippocampus in vitro
作者:
Dougalis
;
Antonios
;
Lees
;
George
;
Ganellin
;
C. Robin
关键词:
cis-Oleamide
;
cis-9
;
10 Octadeceneoamide
;
Serotonin
;
Hippocampus
;
5-HT
1A
and 5-HT
2
receptors
;
Sleep
刊名:Neuropharmacology
出版年:2004
8.
Bis-quinolinium cyclophanes: toward a pharmacophore model for the blockade of apamin-sensitive SK
Ca
channels in sympathetic neurons
作者:
Galanakis
;
Dimitrios
;
Ganellin
;
C. Robin
;
Chen
;
Jian-Quing
;
Gunasekera
;
Diyan
;
Dunn
;
Philip M.
关键词:
Quinolinium
;
Cyclophane
;
Pharmacophore
;
SK3 channel
;
Apamin
;
Conformation
;
Synperiplanar
;
Centroid
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2004
9.
Structural variations of 1-(4-(phenoxymethyl)benzyl)piperidines as nonimidazole histamine H
3
receptor antagonists
作者:
Mikó
;
Tibor
;
Ligneau
;
Xavier
;
Pertz
;
Heinz H.
;
Arrang
;
Jean-Michel
;
Robin
Ganellin
;
C.
;
et. al.
关键词:
Histamine H
3
;
Antagonist
;
Nonimidazole
;
Receptor
;
Medicinal chemistry
刊名:Bioorganic and Medicinal Chemistry
出版年:2004
10.
Defining determinant molecular properties for the blockade of the apamin-sensitive SK
Ca
channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry
作者:
Galanakis
;
Dimitrios
;
Ganellin
;
C. Robin
关键词:
Polarizability
;
QSAR
;
SK
Ca
blockers
;
Apamin
;
UCL 1848
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2004
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