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NATURE电子期刊(1)
Elsevier电子期刊(12)
ACS电子期刊(8)
在“
Elsevier电子期刊
”中,
命中:
12
条,耗时:0.0119942 秒
在所有数据库中总计命中:
21
条
1.
Melatonin, selective and non-selective MT
1
/MT
2
receptors agonists: Differential effects on the 24-h vigilance states
作者:
Rafael Ochoa-Sanchez
;
Stefano Comai
;
Gilberto
Spadoni
;
Annalida Bedini
;
Giorgio Tarzia
;
Gabriella Gobbi
关键词:
Melatonin
;
MT1 receptor
;
MT2 receptor
;
Sleep&ndash
;
wake cycle
;
UCM924
;
UCM793
刊名:Neuroscience Letters
出版年:21 February, 2014
2.
Anxiolytic effects of the melatonin MT
2
receptor partial agonist UCM765: Comparison with melatonin and diazepam
作者:
Rafael Ochoa-Sanchez
;
Quentin Rainer
;
Stefano Comai
;
Gilberto
Spadoni
;
Annalida Bedini
;
Silvia Rivara
;
Franco Fraschini
;
Marco Mor
;
Giorgio Tarzia
;
Gabriella Gobbi
关键词:
MLT
;
melatonin
;
BZs
;
benzodiazepines
;
DZ
;
diazepam
;
4P-PDOT
;
4-phenyl-2- propionamidotetralin
;
EPMT
;
elevated plus maze test
;
NSFT
;
novelty suppressed feeding
;
OFT
;
open field test
刊名:Progress in Neuro-Psychopharmacology and Biological Psychiatry
出版年:2012
3.
Synthesis and characterization of a peripherally restricted CB
1
cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice
作者:
Jesse LoVerme
;
Andrea Duranti
;
Andrea Tontini
;
Gilberto
Spadoni
;
Marco Mor
;
Silvia Rivara
;
Nephi Stella
;
Cong Xu
;
Giorgio Tarzia
;
Daniele Piomelli
关键词:
URB447
;
Peripheral cannabinoid antagonism
;
Anti-obesity agents
;
Pyrrolic CB-antagonists
刊名:Bioorganic and Medicinal Chemistry Letters
出版年:2009
4.
Synthesis and biological activity of new melatonin dimeric derivatives
作者:
Barbara Di Giacomo
;
Annalida Bedini
;
Gilberto
Spadoni
;
Giorgio Tarzia
;
Franco Fraschini
;
Marilou Pannacci
;
Valeria Lucini
关键词:
Melatonin
;
MLT receptors
;
Biligands
;
Melatonin dimers
刊名:Bioorganic and Medicinal Chemistry
出版年:2007
5.
Reassessing the melatonin pharmacophore—Enantiomeric resolution, pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue
作者:
Silvia Rivara
;
Giuseppe Diamantini
;
Barbara Di Giacomo
;
Doriano Lamba
;
Giuseppe Gatti
;
Valeria Lucini
;
Marilou Pannacci
;
Marco Mor
;
Gilberto
Spadoni
and Giorgio Tarzia
关键词:
Melatonin
;
Conformational analysis
;
Molecular modeling
;
Enantiomeric resolution
;
X-ray crystal structure
;
Pharmacophore model
刊名:Bioorganic and Medicinal Chemistry
出版年:2006
6.
Synthesis and conformational study of 3,4-carbocyclic bridged indole melatonin and serotonin analogues
作者:
Bedini
;
Annalida
;
Giacomo
;
Barbara Di
;
Gatti
;
Giuseppe
;
Spadoni
;
Gilberto
关键词:
Melatonin
;
Serotonin
;
Conformational analysis
;
NMR coupling constants
刊名:Bioorganic & Medicinal Chemistry
出版年:2005
7.
Synthesis and structure–activity relationships of a series of pyrrole cannabinoid receptor agonists
作者:
Tarzia
;
Giorgio
;
Duranti
;
Andrea
;
Tontini
;
Andrea
;
Spadoni
;
Gilberto
;
Mor
;
Marco
;
Rivara
;
Silvia
;
et. al.
刊名:Bioorganic and Medicinal Chemistry
出版年:2003
8.
Conformation by NMR of two tetralin-based receptor ligands
作者:
Giuseppe Gatti
;
Giovanni Piersanti
;
Gilberto
Spadoni
刊名:Il Farmaco
出版年:2003
9.
Design and synthesis of melatonin receptors agonists and antagonists
作者:
Tarzia
;
Giorgio
;
Diamantini
;
Giuseppe
;
Mor
;
Marco
;
Spadoni
;
Gilberto
关键词:
Design and synthesis
;
Melatonin receptors
;
Agonists and antagonists
刊名:Il Farmaco
出版年:2000
10.
Synthesis, pharmacological characterization and QSAR studies on 2-substituted indole melatonin receptor ligands
作者:
Mor
;
Marco
;
Spadoni
;
Gilberto
;
Di Giacomo
;
Barbara
;
Diamantini
;
Giuseppe
;
Bedini
;
Annalida
;
et. al.
刊名:Bioorganic and Medicinal Chemistry
出版年:2001
1
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