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Elsevier电子期刊(9)
在“
Elsevier电子期刊
”中,
命中:
9
条,耗时:小于0.01 秒
在所有数据库中总计命中:
9
条
1.
Synthesis, biological evaluation and molecular modeling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT
1A
receptor agonists
作者:
Silvia Franchini
a
;
Leda Ivanova Manasieva
a
;
Claudia Sorbi
a
;
Umberto M. Battisti
a
;
Paola Fossa
b
;
Elena Cichero
b
;
Nunzio Denora
c
;
Rosa Maria Iacobazzi
c
;
d
;
Antonio Cilia
e
;
Lorenza Pirona
e
;
Simone Ronsisvalle
f
;
Giuseppina
Aric
&
ograve
;
f
;
Livio Brasili
a
;
livio.brasili@unimore.it
关键词:
5-HT1A receptor
;
Agonist
;
Neuroprotection
;
BBB penetration
;
Analgesic activity
刊名:European Journal of Medicinal Chemistry
出版年:2017
2.
Multitarget opioid ligands in pain relief: New players in an old game
作者:
Rita Turnaturi
a
;
rita.turnaturi@tiscali.it" class="auth_mail" title="E-mail the corresponding author
;
Giuseppina
Aric
&
ograve
;
a
;
Giuseppe Ronsisvalle
a
;
Carmela Parenti
b
;
1
;
Lorella Pasquinucci
a
;
1
关键词:
Pain
;
MOR
;
DOR
;
KOR
;
Bifunctional ligands
;
Bivalent ligands
刊名:European Journal of Medicinal Chemistry
出版年:2016
3.
An LP1 analogue, selective MOR agonist with a peculiar pharmacological profile, used to scrutiny the ligand binding domain
作者:
Simone Ronsisvalle
a
;
s.ronsisvalle@unict.it" class="auth_mail" title="E-mail the corresponding author
;
Giuseppina
Aric
&
ograve
;
a
;
Federica Panarello
a
;
Angelo Spadaro
a
;
Lorella Pasquinucci
a
;
Maria S. Pappalardo
a
;
Carmela Parenti
b
;
Nicole Ronsisvalle
c
关键词:
MOR agonists
;
6
;
7-Benzomorphan scaffold
;
Modeling studies
;
Radioligand competition-binding assay
;
Tail-flick test
;
GPI and MVD assays
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
4.
Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives
作者:
Silvia Franchini
a
;
Umberto Maria Battisti
a
;
Adolfo Prandi
a
;
Annalisa Tait
a
;
Chiara Borsari
a
;
Elena Cichero
b
;
Paola Fossa
b
;
Antonio Cilia
c
;
Orazio Prezzavento
d
;
Simone Ronsisvalle
d
;
Giuseppina
Aric
&
ograve
;
e
;
Carmela Parenti
e
;
Livio Brasili
a
;
livio.brasili@unimore.it" class="auth_mail" title="E-mail the corresponding author
关键词:
Sigma receptors ligands
;
Sigma-1
;
Sigma-2
;
Piperidine
;
Piperazine
;
1
;
3-Dioxolane
;
Receptor-mediated analgesia
刊名:European Journal of Medicinal Chemistry
出版年:2016
5.
Evaluation of N-substituent structural variations in opioid receptor profile of LP1
作者:
Lorella Pasquinucci
a
;
Rita Turnaturi
a
;
rita.turnaturi@tiscali.it" class="auth_mail" title="E-mail the corresponding author
;
Giuseppina
Aric
&
ograve
;
a
;
Carmela Parenti
b
;
Paschalina Pallaki
c
;
Zafiroula Georgoussi
c
;
Simone Ronsisvalle
a
关键词:
Mu opioid receptor
;
6
;
7-Benzomorhan scaffold
;
Radioligand competition-binding assay
;
GPI and MVD assays
;
Tail-flick test
;
Modeling studies
刊名:Bioorganic & Medicinal Chemistry
出版年:2016
6.
The multitarget opioid ligand LP1's effects in persistent pain and in primary cell neuronal cultures
作者:
Carmela Parenti
a
;
Rita Turnaturi
b
;
Giuseppina
Aric
&
ograve
;
b
;
g
aric
o@unict.it
;
Alexandra Gramowski-Voß
;
c
;
Olaf H.-U. Schroeder
d
;
Agostino Marrazzo
b
;
Orazio Prezzavento
b
;
Simone Ronsisvalle
b
;
Giovanna M. Scoto
a
;
Giuseppe Ronsisvalle
b
;
Lorella Pasquinucci
b
关键词:
Neuropathic pain
;
Inflammatory pain
;
Opioid receptors
;
LP1
;
Micro-electrode array (MEA)
;
Electrophysiological behaviour
刊名:Neuropharmacology
出版年:2013
7.
The benzomorphan-based LP1 ligand is a suitable MOR/DOR agonist for chronic pain treatment
作者:
Lorella Pasquinucci
a
;
lpasquin@unict.it
;
Carmela Parenti
b
;
Rita Turnaturi
a
;
Giuseppina
Aric
&
ograve
;
a
;
Agostino Marrazzo
a
;
Orazio Prezzavento
a
;
Simone Ronsisvalle
a
;
Zafiroula Georgoussi
c
;
Danai-Dionysia Fourla
c
;
Giovanna M. Scoto
b
;
Giuseppe Ronsisvalle
a
关键词:
Bifunctional drugs
;
Antinociceptive tolerance
;
[35S]GTP¦ÃS binding studies
;
Tail-flick test
刊名:Life Sciences
出版年:2012
8.
Effects of intraplantar Nocistatin and (¡À)-J 113397 injections on nociceptive behavior in a rat model of inflammation
作者:
Giovanna M.
;
Scoto
a
;
;
scotog@unict.it
;
Giuseppina
;
Aric
&
ograve
;
b
;
;
g
aric
o@unict.it
;
Simone
;
Ronsisvalle
b
;
;
s.ronsisvalle@unict.it
;
Carmela
;
Parenti
a
;
;
cparenti@unict.it
关键词:
(±
;
)-J 113397
;
Nocistatin
;
Hyperalgesia
;
Allodynia
;
Inflammation
;
Rat hind paw
刊名:Pharmacology Biochemistry and Behavior
出版年:2012
9.
Corrigendum to ¡°MHV-68 producing mIFN¦Á1 is severely attenuated in vivo and effectively protects mice against challenge with wt MHV-68?[Vaccine 29 (2011) 3935-3944]
作者:
Eleonora
Aric
&
ograve
;
a
;
eleonora.
aric
o@iss.it
;
Domenica M. Monque
a
;
Giuseppina
D&rsquo
;
Agostino
a
;
Federica Moschella
a
;
Massimo Venditti
a
;
Ulrich Kalinke
b
;
Deborah J. Allen
c
;
James P. Stewart
d
;
Anthony A. Nash
c
;
Filippo Belardelli
a
;
Maria Ferrantini
a
刊名:Vaccine
出版年:2012
1
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